METHODS OF SYNTHESIZING FACTOR XA INHIBITORS

Described herein are novel methods of preparing a compound of Formula II or a pharmaceutically acceptable salt thereof. In some embodiments, the method is for preparing betrixaban or a pharmaceutically acceptable salt thereof. Also described are compositions comprising substantially pure betrixaban...

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Main Authors SONG, ZHIGUO JAKE, PANDEY, ANJALI, RATO, JOSE, LEITAO, EMILIA P. T
Format Patent
LanguageEnglish
French
Published 14.07.2011
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Abstract Described herein are novel methods of preparing a compound of Formula II or a pharmaceutically acceptable salt thereof. In some embodiments, the method is for preparing betrixaban or a pharmaceutically acceptable salt thereof. Also described are compositions comprising substantially pure betrixaban free base or salt thereof.
AbstractList Described herein are novel methods of preparing a compound of Formula II or a pharmaceutically acceptable salt thereof. In some embodiments, the method is for preparing betrixaban or a pharmaceutically acceptable salt thereof. Also described are compositions comprising substantially pure betrixaban free base or salt thereof.
Author RATO, JOSE
SONG, ZHIGUO JAKE
PANDEY, ANJALI
LEITAO, EMILIA P. T
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DocumentTitleAlternate PROCEDES DE SYNTHESE D'INHIBITEURS DU FACTEUR XA
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RelatedCompanies PORTOLA PHARMACEUTICALS, INC
MILLENNIUM PHARMACEUTICALS, INC
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Snippet Described herein are novel methods of preparing a compound of Formula II or a pharmaceutically acceptable salt thereof. In some embodiments, the method is for...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title METHODS OF SYNTHESIZING FACTOR XA INHIBITORS
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