NOVEL TYROSINE KINASE INHIBITORS

Provided are compounds of the formula (I): or a stereoisomer, tautomer, salt, hydrate or prodrug thereof that modulate tyrosine kinase activity, compositions comprising the compounds and methods of their use.

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Main Authors MIKEL, CHARLES, YAN, ZHENG, LIU, YAHUA, ZOZULYA, SERGEY, GREGOR, VLAD EDWARD, PICKENS, JASON C, THIRUVAZHI, MOHAN SANTHANAM, ZHU, TONG, KADUSHKIN, ALEXANDER, VAIRAGOUNDAR, RANENDRAN, JIANG, LUYONG, VAVILALA, GOVERDHAN REDDY, ANIKIN, ALEXEY, CHUCHOLOWSKI, ALEXANDER, KHASANOV, ALISHER, MCGRATH, DOUGLAS ERIC
Format Patent
LanguageEnglish
French
Published 24.09.2009
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Abstract Provided are compounds of the formula (I): or a stereoisomer, tautomer, salt, hydrate or prodrug thereof that modulate tyrosine kinase activity, compositions comprising the compounds and methods of their use.
AbstractList Provided are compounds of the formula (I): or a stereoisomer, tautomer, salt, hydrate or prodrug thereof that modulate tyrosine kinase activity, compositions comprising the compounds and methods of their use.
Author LIU, YAHUA
MIKEL, CHARLES
VAVILALA, GOVERDHAN REDDY
KADUSHKIN, ALEXANDER
PICKENS, JASON C
ZOZULYA, SERGEY
MCGRATH, DOUGLAS ERIC
GREGOR, VLAD EDWARD
KHASANOV, ALISHER
JIANG, LUYONG
VAIRAGOUNDAR, RANENDRAN
YAN, ZHENG
CHUCHOLOWSKI, ALEXANDER
THIRUVAZHI, MOHAN SANTHANAM
ZHU, TONG
ANIKIN, ALEXEY
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– fullname: YAN, ZHENG
– fullname: LIU, YAHUA
– fullname: ZOZULYA, SERGEY
– fullname: GREGOR, VLAD EDWARD
– fullname: PICKENS, JASON C
– fullname: THIRUVAZHI, MOHAN SANTHANAM
– fullname: ZHU, TONG
– fullname: KADUSHKIN, ALEXANDER
– fullname: VAIRAGOUNDAR, RANENDRAN
– fullname: JIANG, LUYONG
– fullname: VAVILALA, GOVERDHAN REDDY
– fullname: ANIKIN, ALEXEY
– fullname: CHUCHOLOWSKI, ALEXANDER
– fullname: KHASANOV, ALISHER
– fullname: MCGRATH, DOUGLAS ERIC
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DocumentTitleAlternate NOUVEAUX INHIBITEURS DE TYROSINE KINASE
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Snippet Provided are compounds of the formula (I): or a stereoisomer, tautomer, salt, hydrate or prodrug thereof that modulate tyrosine kinase activity, compositions...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title NOVEL TYROSINE KINASE INHIBITORS
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