EQUILIBRATIVE NUCLEOSIDE TRANSPORTER ENT1 INHIBITORS
The present invention is related to novel compounds of formula (I) having equilibrative nucleoside transporter ENT1 inhibiting properties, pharmaceutical compositions comprising these compounds, chemical processes for preparing these compounds and their use in the treatment of diseases linked to the...
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| Main Authors | , , , , |
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| Format | Patent |
| Language | English French |
| Published |
10.01.2017
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The present invention is related to novel compounds of formula (I) having equilibrative nucleoside transporter ENT1 inhibiting properties, pharmaceutical compositions comprising these compounds, chemical processes for preparing these compounds and their use in the treatment of diseases linked to the inhibition of ENT1 receptors in animals, in particular humans.
L'invention porte sur de nouveaux composés de formule (I) présentant des propriétés inhibant le transporteur équilibrant des nucléosides ENT1, sur des préparations pharmaceutiques les comprenant, et sur leurs procédés de préparation, et d'utilisation pour le traitement de maladies de l'animal et en particulier de l'homme, liées à l'inhibition des récepteurs du ENT1. |
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| AbstractList | The present invention is related to novel compounds of formula (I) having equilibrative nucleoside transporter ENT1 inhibiting properties, pharmaceutical compositions comprising these compounds, chemical processes for preparing these compounds and their use in the treatment of diseases linked to the inhibition of ENT1 receptors in animals, in particular humans.
L'invention porte sur de nouveaux composés de formule (I) présentant des propriétés inhibant le transporteur équilibrant des nucléosides ENT1, sur des préparations pharmaceutiques les comprenant, et sur leurs procédés de préparation, et d'utilisation pour le traitement de maladies de l'animal et en particulier de l'homme, liées à l'inhibition des récepteurs du ENT1. |
| Author | BOSMANS, JEAN-PAUL RENE MARIE ANDRE PIETERS, SERGE MARIA ALOYSIUS DE CLEYN, MICHEL ANNA JOZEF BERTHELOT, DIDIER JEAN-CLAUDE VERBIST, BIE MARIA PIETER |
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| DocumentTitleAlternate | INHIBITEURS DU TRANSPORTEUR EQUILIBRANT DES NUCLEOSIDES ENT1 |
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| RelatedCompanies | JANSSEN PHARMACEUTICA NV |
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| Snippet | The present invention is related to novel compounds of formula (I) having equilibrative nucleoside transporter ENT1 inhibiting properties, pharmaceutical... |
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| Title | EQUILIBRATIVE NUCLEOSIDE TRANSPORTER ENT1 INHIBITORS |
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