ENTRY INHIBITORS OF THE HIV VIRUS
The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors...
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| Main Authors | , , , |
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| Format | Patent |
| Language | English French |
| Published |
27.11.2012
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| Subjects | |
| Online Access | Get full text |
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| Abstract | The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors with other anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS. The compounds of formula (I) have the following structure: (I). |
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| AbstractList | The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors with other anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS. The compounds of formula (I) have the following structure: (I). |
| Author | WIGERINCK, PIET TOM BERT PAUL MICHIELS, LIEVE EMMA JAN VAN ACKER, KOENRAAD LODEWIJK AUGUST TAHRI, ABDELLAH |
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| DocumentTitleAlternate | INHIBITEURS DE LA PENETRATION DU VIRUS VIH |
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| RelatedCompanies | TIBOTEC PHARMACEUTICALS LTD |
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| Snippet | The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions,... |
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| SubjectTerms | ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| Title | ENTRY INHIBITORS OF THE HIV VIRUS |
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