AZAINDOLE-ETHYLAMINE DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR BINDING AGENTS

• Main Author: NAGEL, ARTHUR ADAM
• Format: Patent
• Language: English; French
• Published: 02.10.2001
• Edition: 6
• Subjects: CHEMISTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HYGIENE; MEDICAL OR VETERINARY SCIENCE; METALLURGY; ORGANIC CHEMISTRY; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS

Disclosed are compounds that are useful in the treatment of conditions associated with depletion of nicotine receptors in mammals, the compounds having formula I: (wherein X is; a) -CH2NR1R2; b) ; or c) ; where R, R1, and R2 are independently selected from hydrogen and C1-C6 alkyl; R3 is selected fr...