Fused piperidine amides as modulators of ion channels

The invention relates to fused piperidine amides useful as inhibitors of ion channels for the treatment of pain. The invention also provides pharmaceutically acceptable compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various disorders.

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Bibliographic Details
Main Authors Deninno, Michael Paul, Conroy, Erica Lynn, Hurley, Dennis James, Silina, Alina, Pierre, Fabrice Jean Denis, Zhou, Jinglan, Uy, Johnny, Frieman, Bryan A, Anderson, Corey, Groothenhuis, Peter Diederik Jan, Hadida-Ruah, Sara Sabina
Format Patent
LanguageEnglish
Published 28.11.2019
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Abstract The invention relates to fused piperidine amides useful as inhibitors of ion channels for the treatment of pain. The invention also provides pharmaceutically acceptable compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various disorders.
AbstractList The invention relates to fused piperidine amides useful as inhibitors of ion channels for the treatment of pain. The invention also provides pharmaceutically acceptable compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various disorders.
Author Anderson, Corey
Conroy, Erica Lynn
Groothenhuis, Peter Diederik Jan
Hadida-Ruah, Sara Sabina
Hurley, Dennis James
Deninno, Michael Paul
Silina, Alina
Uy, Johnny
Pierre, Fabrice Jean Denis
Frieman, Bryan A
Zhou, Jinglan
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– fullname: Hurley, Dennis James
– fullname: Silina, Alina
– fullname: Pierre, Fabrice Jean Denis
– fullname: Zhou, Jinglan
– fullname: Uy, Johnny
– fullname: Frieman, Bryan A
– fullname: Anderson, Corey
– fullname: Groothenhuis, Peter Diederik Jan
– fullname: Hadida-Ruah, Sara Sabina
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Snippet The invention relates to fused piperidine amides useful as inhibitors of ion channels for the treatment of pain. The invention also provides pharmaceutically...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title Fused piperidine amides as modulators of ion channels
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