Process for the preparation of piperazinyl and diazepanyl benzamide derivatives

• Main Authors: GRIMM, JEFFREY S, SORGI, KIRK L, CHOUDHURY, ANUSUYA, LIU, JING, PALMER, DAVID
• Format: Patent
• Language: English
• Published: 02.06.2016
• Subjects: CHEMISTRY; HETEROCYCLIC COMPOUNDS; HUMAN NECESSITIES; HYGIENE; MEDICAL OR VETERINARY SCIENCE; METALLURGY; ORGANIC CHEMISTRY; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS

The present invention is directed to a novel process for the preparation of piperazinyl and diazepanyl benzamide derivatives, useful for the treatment of disorders and conditions mediated by a histamine receptor, preferably the H3 5 receptor.