Novel heterocyclic compounds as HSP90-inhibitors

NOVEL HETEROCYCLIC COMPOUNDS AS HSP90-INHIBITORS Abstract Novel heterocyclic compounds are described and demonstrated to have utility as Heat Shock Protein 90 (HSP90) inhibiting agent. Method of synthesis and use of such 5 compounds are also described.

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Main Authors SHI, JIANDONG, BOEHM, MARCUS F, KASIBHATLA, SRINIVAS R, LE BRAZIDEC, JEAN-YVES, BIAMONTE, MARCO A, HONG, KEVIN D, ZHANG, LIN, HURST, DAVID
Format Patent
LanguageEnglish
Published 01.09.2011
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Abstract NOVEL HETEROCYCLIC COMPOUNDS AS HSP90-INHIBITORS Abstract Novel heterocyclic compounds are described and demonstrated to have utility as Heat Shock Protein 90 (HSP90) inhibiting agent. Method of synthesis and use of such 5 compounds are also described.
AbstractList NOVEL HETEROCYCLIC COMPOUNDS AS HSP90-INHIBITORS Abstract Novel heterocyclic compounds are described and demonstrated to have utility as Heat Shock Protein 90 (HSP90) inhibiting agent. Method of synthesis and use of such 5 compounds are also described.
Author HONG, KEVIN D
SHI, JIANDONG
HURST, DAVID
ZHANG, LIN
LE BRAZIDEC, JEAN-YVES
BIAMONTE, MARCO A
BOEHM, MARCUS F
KASIBHATLA, SRINIVAS R
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– fullname: BIAMONTE, MARCO A
– fullname: HONG, KEVIN D
– fullname: ZHANG, LIN
– fullname: HURST, DAVID
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Snippet NOVEL HETEROCYCLIC COMPOUNDS AS HSP90-INHIBITORS Abstract Novel heterocyclic compounds are described and demonstrated to have utility as Heat Shock Protein 90...
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SubjectTerms ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
Title Novel heterocyclic compounds as HSP90-inhibitors
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