Oxadiazole derivatives active on sphingosine-1-phosphate (S1P)

The present application discloses oxadiazole based compounds of Formula (I) active on sphingosine-1-phosphate (S1P) in particular useful to treat lupus erythematosus. A is phenyl or a 5 or 6-membered heteroaryl ring; R

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Main Authors JOHNSON, CHRISTOPHER NORBERT, SKIDMORE, JOHN, DEMONT, EMMANUEL HUBERT, HEER, JAG PAUL, HURST, DAVID NIGEL, WALL, IAN DAVID, WITHERINGTON, JASON, HEIGHTMAN, THOMAS DANIEL
Format Patent
LanguageEnglish
Published 26.09.2013
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Abstract The present application discloses oxadiazole based compounds of Formula (I) active on sphingosine-1-phosphate (S1P) in particular useful to treat lupus erythematosus. A is phenyl or a 5 or 6-membered heteroaryl ring; R
AbstractList The present application discloses oxadiazole based compounds of Formula (I) active on sphingosine-1-phosphate (S1P) in particular useful to treat lupus erythematosus. A is phenyl or a 5 or 6-membered heteroaryl ring; R
Author DEMONT, EMMANUEL HUBERT
HEIGHTMAN, THOMAS DANIEL
WALL, IAN DAVID
SKIDMORE, JOHN
HEER, JAG PAUL
WITHERINGTON, JASON
HURST, DAVID NIGEL
JOHNSON, CHRISTOPHER NORBERT
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– fullname: DEMONT, EMMANUEL HUBERT
– fullname: HEER, JAG PAUL
– fullname: HURST, DAVID NIGEL
– fullname: WALL, IAN DAVID
– fullname: WITHERINGTON, JASON
– fullname: HEIGHTMAN, THOMAS DANIEL
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Snippet The present application discloses oxadiazole based compounds of Formula (I) active on sphingosine-1-phosphate (S1P) in particular useful to treat lupus...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title Oxadiazole derivatives active on sphingosine-1-phosphate (S1P)
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