Novel substituted thiophenepyrimidinone derivatives as inhibitors of 17beta-hydroxysteroid dehydrogenase

This invention relates to novel substituted thiophenepyrimidinone derivatives and their use in therapy, especially for use in the treatment and/or prevention of a steroid hormone dependent diseases or disorder, such as steroid hormone dependent diseases or disorders requiring inhibition of 17ß-hydro...

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Main Authors PASI KOSKIMIES, JOSEF MESSINGER, OLLI TANELI PENTIKAINEN, HEINRICH-HUBERT THOLE, PAULI SAARENKETO, BETTINA HUSEN, LEENA HIRVELA, PEKKA LEHTOVUORI, JOHANNA KIVINIEMI, MIKKO UNKILA, LILA PIRKKALA, BARTHOLOMEUS JOHANNES VAN STEEN
Format Patent
LanguageEnglish
Published 22.06.2006
Subjects
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
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Abstract This invention relates to novel substituted thiophenepyrimidinone derivatives and their use in therapy, especially for use in the treatment and/or prevention of a steroid hormone dependent diseases or disorder, such as steroid hormone dependent diseases or disorders requiring inhibition of 17ß-hydroxysteroid dehydrogenase enzymes.
AbstractList This invention relates to novel substituted thiophenepyrimidinone derivatives and their use in therapy, especially for use in the treatment and/or prevention of a steroid hormone dependent diseases or disorder, such as steroid hormone dependent diseases or disorders requiring inhibition of 17ß-hydroxysteroid dehydrogenase enzymes.
Author JOHANNA KIVINIEMI
BETTINA HUSEN
BARTHOLOMEUS JOHANNES VAN STEEN
LEENA HIRVELA
HEINRICH-HUBERT THOLE
LILA PIRKKALA
PAULI SAARENKETO
PEKKA LEHTOVUORI
PASI KOSKIMIES
OLLI TANELI PENTIKAINEN
MIKKO UNKILA
JOSEF MESSINGER
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– fullname: PAULI SAARENKETO
– fullname: BETTINA HUSEN
– fullname: LEENA HIRVELA
– fullname: PEKKA LEHTOVUORI
– fullname: JOHANNA KIVINIEMI
– fullname: MIKKO UNKILA
– fullname: LILA PIRKKALA
– fullname: BARTHOLOMEUS JOHANNES VAN STEEN
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Snippet This invention relates to novel substituted thiophenepyrimidinone derivatives and their use in therapy, especially for use in the treatment and/or prevention...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
Title Novel substituted thiophenepyrimidinone derivatives as inhibitors of 17beta-hydroxysteroid dehydrogenase
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