4, 5-DIARYLTHIAZOLE DERIVATIVES AS CB-1 LIGANDS

The present invention relates to compounds of formula (I): in which R1 and R2 independently represent phenyl, thienyl or pyridyl and R3 represents a group -X-Y-NR4R5 in which X is CO or SO2; Y is absent or represents NH and the other substituente are as defined in the description and their use in th...

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Main Authors ANNA, INGRID, KRISTINA BERGGREN, JOHAN, MICHAEL WILSTERMANN, STIG, JONAS BOSTROM, PETER GREASLEY, STIG, THOMAS ELEBRING, LINDA FALLEFORS
Format Patent
LanguageEnglish
Published 22.07.2004
Edition7
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Abstract The present invention relates to compounds of formula (I): in which R1 and R2 independently represent phenyl, thienyl or pyridyl and R3 represents a group -X-Y-NR4R5 in which X is CO or SO2; Y is absent or represents NH and the other substituente are as defined in the description and their use in the treatment of obesity, psychiatric and neurological disorders and to pharmaceutical compositions containing them.
AbstractList The present invention relates to compounds of formula (I): in which R1 and R2 independently represent phenyl, thienyl or pyridyl and R3 represents a group -X-Y-NR4R5 in which X is CO or SO2; Y is absent or represents NH and the other substituente are as defined in the description and their use in the treatment of obesity, psychiatric and neurological disorders and to pharmaceutical compositions containing them.
Author JOHAN, MICHAEL WILSTERMANN
ANNA, INGRID, KRISTINA BERGGREN
STIG, THOMAS ELEBRING
PETER GREASLEY
STIG, JONAS BOSTROM
LINDA FALLEFORS
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– fullname: PETER GREASLEY
– fullname: STIG, THOMAS ELEBRING
– fullname: LINDA FALLEFORS
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Snippet The present invention relates to compounds of formula (I): in which R1 and R2 independently represent phenyl, thienyl or pyridyl and R3 represents a group...
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SubjectTerms CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Title 4, 5-DIARYLTHIAZOLE DERIVATIVES AS CB-1 LIGANDS
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