Novel Antagonists Acting at the P2Y 1 Purinergic Receptor:  Synthesis and Conformational Analysis Using Potentiometric and Nuclear Magnetic Resonance Titration Techniques

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Published inJournal of medicinal chemistry Vol. 45; no. 4; pp. 962 - 972
Main Authors Raboisson, Pierre, Baurand, Anthony, Cazenave, Jean-Pierre, Gachet, Christian, Retat, Myriam, Spiess, Bernard, Bourguignon, Jean-Jacques
Format Journal Article
LanguageEnglish
Published 01.02.2002
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Author Gachet, Christian
Retat, Myriam
Baurand, Anthony
Spiess, Bernard
Bourguignon, Jean-Jacques
Cazenave, Jean-Pierre
Raboisson, Pierre
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  givenname: Jean-Jacques
  surname: Bourguignon
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  organization: Laboratoire de Pharmacochimie de la Communication Cellulaire, UMR 7081 du CNRS, Faculté de Pharmacie, Université Louis Pasteur, 74, Route du Rhin, 67401 Illkirch Cedex, France, and Laboratoire de Biologie et de Pharmacologie de l'Hémostase et de la Thrombose, Etablissement Français du Sang-Alsace, U.311 de l'INSERM, 10, Rue Spielmann, BP 36, 67065 Strasbourg Cedex, France
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Title Novel Antagonists Acting at the P2Y 1 Purinergic Receptor:  Synthesis and Conformational Analysis Using Potentiometric and Nuclear Magnetic Resonance Titration Techniques
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