Synthesis and evaluation of two new candidate high-affinity full agonist PET radioligands for imaging 5-HT1B receptors - Lindberg, Anton; Lu, Shuiyu; Nag, Sangram; Schou, Magnus; Liow, Jeih-San; Zoghbi, Sami S.; Frankland, Michael P.; Gladding, Robert L.; Morse, Cheryl L.; Takano, Akihiro; Amini, Nahid; Elmore, Charles S.; et al. (Nuclear medicine and biology, 2019)
Keywords: Affinity; Agonist; Agonists; Anxiety; Binding; Brain; Carbon monoxide; Carbon-11; Carbonylation; Efflux; Experiments; Headache; Intravenous administration; Mental depression; Methylation; Migraine; Neuroimaging; Parameter identification; Pharmacology; Physiochemistry; Positron emission; Positron emission tomography; Precursors; Pretreatment; Primates; Radioactivity; Radiochemistry; Radioisotopes; Radioligand; Receptors; Serotonin; Serotonin S1 receptors; Serotonin subtype 1B receptor; Tomography; Serotonin subtype 1B receptor; Agonist; Carbonylation; Radioligand; Carbon-11