Sulfur (SⅥ)-containing heterocyclic hybrids as antibacterial agents against methicillin-resistant Staphylococcus aureus (MRSA) and its SAR
[Display omitted] •Sulfur (SⅥ)-containing heterocyclic hybrids displayed potent antibacterial activity against tested MRSA strains.•Structure-activity relationship is explained in detail.•Sulfur (SⅥ)-containing heterocyclic hybrids exhibited excellent antibacterial activity with different action of...
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| Published in | Bioorganic chemistry Vol. 145; p. 107241 |
|---|---|
| Main Authors | , , , , , , |
| Format | Journal Article |
| Language | English |
| Published |
United States
Elsevier Inc
01.04.2024
|
| Subjects | |
| Online Access | Get full text |
| ISSN | 0045-2068 1090-2120 1090-2120 |
| DOI | 10.1016/j.bioorg.2024.107241 |
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| Abstract | [Display omitted]
•Sulfur (SⅥ)-containing heterocyclic hybrids displayed potent antibacterial activity against tested MRSA strains.•Structure-activity relationship is explained in detail.•Sulfur (SⅥ)-containing heterocyclic hybrids exhibited excellent antibacterial activity with different action of mechanism.•Sulfur (SⅥ)-containing heterocyclic hybrids acts as antibiofilm agents, DNA binding agents, enzyme inhibitors and showed synergistic effect with antibiotics.
The discovery of new small molecule-based inhibitors is an attractive field in medicinal chemistry. Structurally diversified heterocyclic derivatives have been investigated to combat multi-drug resistant bacterial infections and they offers several mechanism of action. Methicillin-resistant Staphylococcus aureus (MRSA) is becoming more and more deadly to humans because of its simple method of transmission, quick development of antibiotic resistance, and ability to cause hard-to-treat skin and filmy diseases. The sulfur (SVI) particularly sulfonyl and sulfonamide based heterocyclic moieties, have found to be good anti-MRSA agents. The development of new nontoxic, economical and highly active sulfur (SVI) containing derivatives has become hot research topics in drug discovery research. Presently, more than 150 FDA approved Sulfur (SVI)-based drugs are available in the market, and they are widely used to treat various types of diseases with different therapeutic potential. The present collective data provides the latest advancements in Sulfur (SVI)-hybrid compounds as antibacterial agents against MRSA. It also examines the outcomes of in-vitro and in-vivo investigations, exploring potential mechanisms of action and offering alternative perspectives on the structure–activity relationship (SAR). Sulfur (SVI)-hybrids exhibits synergistic effects with existing drugs to provide antibacterial action against MRSA |
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| AbstractList | [Display omitted]
•Sulfur (SⅥ)-containing heterocyclic hybrids displayed potent antibacterial activity against tested MRSA strains.•Structure-activity relationship is explained in detail.•Sulfur (SⅥ)-containing heterocyclic hybrids exhibited excellent antibacterial activity with different action of mechanism.•Sulfur (SⅥ)-containing heterocyclic hybrids acts as antibiofilm agents, DNA binding agents, enzyme inhibitors and showed synergistic effect with antibiotics.
The discovery of new small molecule-based inhibitors is an attractive field in medicinal chemistry. Structurally diversified heterocyclic derivatives have been investigated to combat multi-drug resistant bacterial infections and they offers several mechanism of action. Methicillin-resistant Staphylococcus aureus (MRSA) is becoming more and more deadly to humans because of its simple method of transmission, quick development of antibiotic resistance, and ability to cause hard-to-treat skin and filmy diseases. The sulfur (SVI) particularly sulfonyl and sulfonamide based heterocyclic moieties, have found to be good anti-MRSA agents. The development of new nontoxic, economical and highly active sulfur (SVI) containing derivatives has become hot research topics in drug discovery research. Presently, more than 150 FDA approved Sulfur (SVI)-based drugs are available in the market, and they are widely used to treat various types of diseases with different therapeutic potential. The present collective data provides the latest advancements in Sulfur (SVI)-hybrid compounds as antibacterial agents against MRSA. It also examines the outcomes of in-vitro and in-vivo investigations, exploring potential mechanisms of action and offering alternative perspectives on the structure–activity relationship (SAR). Sulfur (SVI)-hybrids exhibits synergistic effects with existing drugs to provide antibacterial action against MRSA The discovery of new small molecule-based inhibitors is an attractive field in medicinal chemistry. Structurally diversified heterocyclic derivatives have been investigated to combat multi-drug resistant bacterial infections and they offers several mechanism of action. Methicillin-resistant Staphylococcus aureus (MRSA) is becoming more and more deadly to humans because of its simple method of transmission, quick development of antibiotic resistance, and ability to cause hard-to-treat skin and filmy diseases. The sulfur (SVI) particularly sulfonyl and sulfonamide based heterocyclic moieties, have found to be good anti-MRSA agents. The development of new nontoxic, economical and highly active sulfur (SVI) containing derivatives has become hot research topics in drug discovery research. Presently, more than 150 FDA approved Sulfur (SVI)-based drugs are available in the market, and they are widely used to treat various types of diseases with different therapeutic potential. The present collective data provides the latest advancements in Sulfur (SVI)-hybrid compounds as antibacterial agents against MRSA. It also examines the outcomes of in-vitro and in-vivo investigations, exploring potential mechanisms of action and offering alternative perspectives on the structure-activity relationship (SAR). Sulfur (SVI)-hybrids exhibits synergistic effects with existing drugs to provide antibacterial action against MRSA.The discovery of new small molecule-based inhibitors is an attractive field in medicinal chemistry. Structurally diversified heterocyclic derivatives have been investigated to combat multi-drug resistant bacterial infections and they offers several mechanism of action. Methicillin-resistant Staphylococcus aureus (MRSA) is becoming more and more deadly to humans because of its simple method of transmission, quick development of antibiotic resistance, and ability to cause hard-to-treat skin and filmy diseases. The sulfur (SVI) particularly sulfonyl and sulfonamide based heterocyclic moieties, have found to be good anti-MRSA agents. The development of new nontoxic, economical and highly active sulfur (SVI) containing derivatives has become hot research topics in drug discovery research. Presently, more than 150 FDA approved Sulfur (SVI)-based drugs are available in the market, and they are widely used to treat various types of diseases with different therapeutic potential. The present collective data provides the latest advancements in Sulfur (SVI)-hybrid compounds as antibacterial agents against MRSA. It also examines the outcomes of in-vitro and in-vivo investigations, exploring potential mechanisms of action and offering alternative perspectives on the structure-activity relationship (SAR). Sulfur (SVI)-hybrids exhibits synergistic effects with existing drugs to provide antibacterial action against MRSA. The discovery of new small molecule-based inhibitors is an attractive field in medicinal chemistry. Structurally diversified heterocyclic derivatives have been investigated to combat multi-drug resistant bacterial infections and they offers several mechanism of action. Methicillin-resistant Staphylococcus aureus (MRSA) is becoming more and more deadly to humans because of its simple method of transmission, quick development of antibiotic resistance, and ability to cause hard-to-treat skin and filmy diseases. The sulfur (S ) particularly sulfonyl and sulfonamide based heterocyclic moieties, have found to be good anti-MRSA agents. The development of new nontoxic, economical and highly active sulfur (S ) containing derivatives has become hot research topics in drug discovery research. Presently, more than 150 FDA approved Sulfur (S )-based drugs are available in the market, and they are widely used to treat various types of diseases with different therapeutic potential. The present collective data provides the latest advancements in Sulfur (S )-hybrid compounds as antibacterial agents against MRSA. It also examines the outcomes of in-vitro and in-vivo investigations, exploring potential mechanisms of action and offering alternative perspectives on the structure-activity relationship (SAR). Sulfur (S )-hybrids exhibits synergistic effects with existing drugs to provide antibacterial action against MRSA. |
| ArticleNumber | 107241 |
| Author | Xue, Fan Verma, Santosh Kumar Verma, Rameshwari Rangappa, Kanchugarakoppal S. Verma, Shekhar Rangappa, Shobith Sharath Kumar, Kothanahally S. |
| Author_xml | – sequence: 1 givenname: Santosh Kumar surname: Verma fullname: Verma, Santosh Kumar organization: School of New Energy, Yulin University, Yulin 719000, Shaanxi, PR China – sequence: 2 givenname: Shobith surname: Rangappa fullname: Rangappa, Shobith organization: Adichunchanagiri Institute for Molecular Medicine, Adichunchanagiri Institute of Medical Sciences, Adichunchanagiri University, B. G. Nagar 571448, India – sequence: 3 givenname: Rameshwari surname: Verma fullname: Verma, Rameshwari email: rbaghe19@yulinu.edu.cn organization: School of New Energy, Yulin University, Yulin 719000, Shaanxi, PR China – sequence: 4 givenname: Fan surname: Xue fullname: Xue, Fan organization: Shaanxi Key Laboratory of Low Metamorphic Coal Clean Utilization, Yulin University, Yulin 719000, PR China – sequence: 5 givenname: Shekhar surname: Verma fullname: Verma, Shekhar organization: Department of Pharmacy, Guru Ghasidas Central University, Bilaspur 495009, Chhattisgarh, India – sequence: 6 givenname: Kothanahally S. surname: Sharath Kumar fullname: Sharath Kumar, Kothanahally S. email: sharu.shivaramu@gmail.com organization: Department of Studies in Chemistry, Manasagangotri, University of Mysore, Mysuru 570006, India – sequence: 7 givenname: Kanchugarakoppal S. surname: Rangappa fullname: Rangappa, Kanchugarakoppal S. email: rangappaks@yahoo.com organization: Department of Studies in Chemistry, Manasagangotri, University of Mysore, Mysuru 570006, India |
| BackLink | https://www.ncbi.nlm.nih.gov/pubmed/38437761$$D View this record in MEDLINE/PubMed |
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| Keywords | NR SAR WTA HTS MIC Sulfur (SVI)-hybrids SASF ESKAPE Antibacterial agents MBC SuFEx SD Azoles DFT S. aureus PABA MRSA LTA DOC ESF MDR PK ALH Sulfur (S(VI))-hybrids |
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•Sulfur (SⅥ)-containing heterocyclic hybrids displayed potent antibacterial activity against tested MRSA strains.•Structure-activity... The discovery of new small molecule-based inhibitors is an attractive field in medicinal chemistry. Structurally diversified heterocyclic derivatives have been... |
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| SubjectTerms | Anti-Bacterial Agents - chemistry Anti-Bacterial Agents - pharmacology Antibacterial agents Azoles Humans Methicillin-Resistant Staphylococcus aureus Microbial Sensitivity Tests MRSA SAR Structure-Activity Relationship Sulfur (SVI)-hybrids Sulfur - pharmacology |
| Title | Sulfur (SⅥ)-containing heterocyclic hybrids as antibacterial agents against methicillin-resistant Staphylococcus aureus (MRSA) and its SAR |
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