The First Structure–Activity Relationship Studies for Designer Receptors Exclusively Activated by Designer Drugs - Chen, Xin; Choo, Hyunah; Huang, Xi-Ping; Yang, Xiaobao; Stone, Orrin; Roth, Bryan L; Jin, Jian (ACS chemical neuroscience, 2015)
Keywords: Acetylcholine - pharmacology; Animals; Cholinergic Agonists - pharmacology; Clozapine - analogs & derivatives; Clozapine - pharmacology; Designer Drugs; Dibenzazepines - pharmacology; Humans; Ligands; Receptor, Muscarinic M3 - chemistry; Receptor, Muscarinic M3 - drug effects; Serotonin Antagonists - pharmacology; Signal Transduction - drug effects; Structure-Activity Relationship; neuronal activation; CNO; SAR; hM3Dq; perlapine; DREADD