Structure-Based Design of Irreversible Human KAT II Inhibitors: Discovery of New Potency-Enhancing Interactions - Tuttle, Jamison B; Anderson, Marie; Bechle, Bruce M; Campbell, Brian M; Chang, Cheng; Dounay, Amy B; Evrard, Edelweiss; Fonseca, Kari R; Gan, Xinmin; Ghosh, Somraj; Horner, Weldon; James, Larry C; et al. (ACS medicinal chemistry letters, 2013)
Keywords: Letter; dose response modeling; irreversible inhibition; kynurenine amino transferase; hydroxamic acid; schizophrenia; kynurenic acid; in vivo microdialysis; aryl hydrocarbon receptor