Pharmacological characterization of GLPG1972/S201086, a potent and selective small-molecule inhibitor of ADAMTS5
Clement-Lacroix, P., Little, C.B., Smith, M.M., Cottereaux, C., Merciris, D., Meurisse, S., Mollat, P., Touitou, R., Brebion, F., Gosmini, R., De Ceuninck, F., Botez, I., Lepescheux, L., van der Aar, E., Christophe, T., Vandervoort, N., Blanqué, R., Comas, D., Deprez, P., Amantini, D.
Published in Osteoarthritis and cartilage (01.02.2022)
Published in Osteoarthritis and cartilage (01.02.2022)
Get full text
Journal Article
Anti‐rheumatic activities of histone deacetylase (HDAC) inhibitors in vivo in collagen‐induced arthritis in rodents
Lin, H‐S, Hu, C‐Y, Chan, H‐Y, Liew, Y‐Y, Huang, H‐P, Lepescheux, L, Bastianelli, E, Baron, R, Rawadi, G, Clément‐Lacroix, P
Published in British journal of pharmacology (01.04.2007)
Published in British journal of pharmacology (01.04.2007)
Get full text
Journal Article
OP0258 Efficacy of the highly selective adamts-5 inhibitor glpg1972 in the rat meniscectomy model
Lepescheux, L., Clement-Lacroix, P., Merciris, D., Meurisse, S., Borgonovi, M., Cottereaux, C., Mollat, P., Brebion, F., Gosmini, R., De Ceuninck, F., Botez, I., van der Aar, E., Christophe, T., Vandervoort, N., Blanqué, R., Comas, D., Deprez, P., Amantini, D.
Published in Annals of the rheumatic diseases (01.06.2018)
Published in Annals of the rheumatic diseases (01.06.2018)
Get full text
Journal Article
Deletion of estrogen receptors reveals a regulatory role for estrogen receptors-β in bone remodeling in females but not in males
SIMS, N. A, DUPONT, S, KRUST, A, CLEMENT-LACROIX, P, MINET, D, RESCHE-RIGON, M, GAILLARD-KELLY, M, BARON, R
Published in Bone (New York, N.Y.) (2002)
Published in Bone (New York, N.Y.) (2002)
Get full text
Journal Article
GLPG1972: a potent, selective, orally available adamts-5 inhibitor for the treatment of OA
Clement-Lacroix, P, Little, C, Meurisse, S, Blanqué, R, Mollat, P, Brebion, F, Gosmini, R, De Ceuninck, F, Botez, I, Lepescheux, L, van der Aar, E, Christophe, T, Vandervoort, N, Cottereaux, C, Comas, D, Deprez, P, Amantini, D
Published in Osteoarthritis and cartilage (01.04.2017)
Published in Osteoarthritis and cartilage (01.04.2017)
Get full text
Journal Article
New cartilage quality evaluation using bio-indentation: effect of a tool dmoad compound active in the rat MNX model
Lavet, C, Clement-Lacroix, P, Merciris, D, Meurisse, S, Lepescheux, L, Gaillard, V, Pastoureau, P, Deprez, P, Amantini, D, Ammann, P
Published in Osteoarthritis and cartilage (01.04.2016)
Published in Osteoarthritis and cartilage (01.04.2016)
Get full text
Journal Article
THU0116 Biological Effects of the JAK1 Selective Inhibitor GLPG0634 on Inflammation Markers in Arthritic Mice
Vayssiere, B., de Vos, S., Merciris, D., Auberval, M., Dupont, S., Vandeghinste, N., Lepescheux, L., Clement-Lacroix, P., Delerive, P., van Rompaey, L., Brys, R., Galien, R.
Published in Annals of the rheumatic diseases (01.06.2013)
Published in Annals of the rheumatic diseases (01.06.2013)
Get full text
Journal Article
Androgen replacement therapy improves function in male rat muscles independently of hypertrophy and activation of the Akt/mTOR pathway
Hourdé, C., Jagerschmidt, C., Clément-Lacroix, P., Vignaud, A., Ammann, P., Butler-Browne, G. S., Ferry, A.
Published in Acta Physiologica (01.04.2009)
Published in Acta Physiologica (01.04.2009)
Get full text
Journal Article
Up-regulation of a set of genes in breast cancer bone metastases discloses predisposition to generate metastases also in visceral organs
Rucci, N, Capulli, M, Angelucci, A, Martella, F, Bologna, M, Ventura, L, Moreschini, O, Driouch, K, Landemaine, T, Lidereau, R, Clement-Lacroix, P, Garcia, T, Ricevuto, E, Teti, A
Published in Bone (New York, N.Y.) (01.05.2011)
Published in Bone (New York, N.Y.) (01.05.2011)
Get full text
Journal Article
Osteoblasts are a new target for prolactin: analysis of bone formation in prolactin receptor knockout mice
Clément-Lacroix, P, Ormandy, C, Lepescheux, L, Ammann, P, Damotte, D, Goffin, V, Bouchard, B, Amling, M, Gaillard-Kelly, M, Binart, N, Baron, R, Kelly, P A
Published in Endocrinology (Philadelphia) (01.01.1999)
Published in Endocrinology (Philadelphia) (01.01.1999)
Get full text
Journal Article
Deletion of a Single Allele of the Dkk1 Gene Leads to an Increase in Bone Formation and Bone Mass
Morvan, Frederic, Boulukos, Kim, Clément‐Lacroix, Philippe, Roman, Sergio Roman, Suc‐Royer, Isabelle, Vayssière, Béatrice, Ammann, Patrick, Martin, Patrick, Pinho, Sonia, Pognonec, Philippe, Mollat, Patrick, Niehrs, Christof, Baron, Roland, Rawadi, Georges
Published in Journal of bone and mineral research (01.06.2006)
Published in Journal of bone and mineral research (01.06.2006)
Get full text
Journal Article
Thyroid Hormone Excess Rather Than Thyrotropin Deficiency Induces Osteoporosis in Hyperthyroidism
Bassett, J. H. Duncan, O’Shea, Patrick J, Sriskantharajah, Srividya, Rabier, Bénédicte, Boyde, Alan, Howell, Peter G. T, Weiss, Roy E, Roux, Jean-Paul, Malaval, Luc, Clement-Lacroix, Phillipe, Samarut, Jacques, Chassande, Olivier, Williams, Graham R
Published in Molecular endocrinology (Baltimore, Md.) (01.05.2007)
Published in Molecular endocrinology (Baltimore, Md.) (01.05.2007)
Get full text
Journal Article
437 IL-17C inhibition reduces skin inflammation in IL23-induced psoriasis mouse model
Marsais, F., Auberval, M., Lavazais, S., Lepescheux, L., Clement-Lacroix, P., Dupont, S., Haertle, S., Steidl, S., Brys, R., Vandeghinste, N.
Published in Journal of investigative dermatology (01.10.2017)
Published in Journal of investigative dermatology (01.10.2017)
Get full text
Journal Article
ADAMTS-5 inhibition with the potent and highly selective inhibitor GLPG1972 results in strong disease-modifying OA drug effects in the rat meniscectomy model
Clement-Lacroix, P., Meurisse, S., Lepescheux, L., Merciris, D., Borgonovi, M., Cottereaux, C., Mollat, P., Brebion, F., Gosmini, R., De Ceuninck, F., Botez, I., Christophe, T., van der Aar, E.E., Vandervoort, N., Blanqué, R., Comas, D., Deprez, P., Amantini, D.
Published in Osteoarthritis and cartilage (01.04.2018)
Published in Osteoarthritis and cartilage (01.04.2018)
Get full text
Journal Article
Increased expression of a set of genes enriched in oxygen binding function discloses a predisposition of breast cancer bone metastases to generate metastasis spread in multiple organs
Capulli, Mattia, Angelucci, Adriano, Driouch, Keltouma, Garcia, Teresa, Clement-Lacroix, Philippe, Martella, Francesco, Ventura, Luca, Bologna, Mauro, Flamini, Stefano, Moreschini, Oreste, Lidereau, Rosette, Ricevuto, Enrico, Muraca, Maurizio, Teti, Anna, Rucci, Nadia
Published in Journal of bone and mineral research (01.11.2012)
Published in Journal of bone and mineral research (01.11.2012)
Get full text
Journal Article
IRAK4 inhibition dampens pathogenic processes driving inflammatory skin diseases
Lavazais, Stéphanie, Jargosch, Manja, Dupont, Sonia, Labéguère, Frédéric, Menet, Christel, Jagerschmidt, Catherine, Ohm, Frenz, Kupcsik, Laszlo, Parent, Isabelle, Cottereaux, Céline, Marsais, Florence, Oste, Line, Van de Water, An, Christophe, Thierry, De Vos, Steve, Fallon, Padraic, Lauffer, Felix, Clément-Lacroix, Philippe, Eyerich, Kilian, Brys, Reginald
Published in Science translational medicine (15.02.2023)
Published in Science translational medicine (15.02.2023)
Get more information
Journal Article
Lrp5-Independent Activation of Wnt Signaling by Lithium Chloride Increases Bone Formation and Bone Mass in Mice
Philippe Clément-Lacroix, Minrong Ai, Frederic Morvan, Sergio Roman-Roman, Béatrice Vayssière, Cecille Belleville, Kenneth Estrera, Warman, Matthew L., Baron, Roland, Georges Rawadi, Prockop, Darwin J.
Published in Proceedings of the National Academy of Sciences - PNAS (29.11.2005)
Published in Proceedings of the National Academy of Sciences - PNAS (29.11.2005)
Get full text
Journal Article
Bone homeostasis in growth hormone receptor-null mice is restored by IGF-I but independent of Stat5
Sims, N A, Clément-Lacroix, P, Da Ponte, F, Bouali, Y, Binart, N, Moriggl, R, Goffin, V, Coschigano, K, Gaillard-Kelly, M, Kopchick, J, Baron, R, Kelly, P A
Published in The Journal of clinical investigation (01.11.2000)
Published in The Journal of clinical investigation (01.11.2000)
Get full text
Journal Article