On the basis of sex: male vs. female rat adenosine A1/A2A receptor affinity
Janse van Rensburg, Helena D, Terre'Blanche, Gisella, Van der Walt, Mietha M
Published in BMC research notes (10.08.2023)
Published in BMC research notes (10.08.2023)
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Journal Article
1,3,7-Triethyl-substituted xanthines—possess nanomolar affinity for the adenosine A1 receptor
Van der Walt, Mietha M., Terre’Blanche, Gisella
Published in Bioorganic & medicinal chemistry (15.10.2015)
Published in Bioorganic & medicinal chemistry (15.10.2015)
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Journal Article
Imidazo[1,2-α]pyridines possess adenosine A1 receptor affinity for the potential treatment of cognition in neurological disorders
Lefin, Roslyn, van der Walt, Mietha M., Milne, Pieter J., Terre'Blanche, Gisella
Published in Bioorganic & medicinal chemistry letters (01.09.2017)
Published in Bioorganic & medicinal chemistry letters (01.09.2017)
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Journal Article
Evaluation of chemical constituents of Rooibos (Aspalathus linearis) and Honeybush (Cyclopia intermedia) as adenosine A1/A2A receptor ligands
Gouws, Liezel, Janse van Rensburg, Helena D., Terre’Blanche, Gisella, Van der Walt, Mietha M.
Published in Medicinal chemistry research (01.12.2023)
Published in Medicinal chemistry research (01.12.2023)
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Journal Article
Methoxy substituted 2-benzylidene-1-indanone derivatives as A and/or A AR antagonists for the potential treatment of neurological conditions
Janse van Rensburg, Helena D, Legoabe, Lesetja J, Terre'Blanche, Gisella, Van der Walt, Mietha M
Published in MedChemComm (20.02.2019)
Published in MedChemComm (20.02.2019)
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Journal Article
Methoxy substituted 2-benzylidene-1-indanone derivatives as A 1 and/or A 2A AR antagonists for the potential treatment of neurological conditions
Janse van Rensburg, Helena D, Legoabe, Lesetja J, Terre'Blanche, Gisella, Van der Walt, Mietha M
Published in MedChemComm (20.02.2019)
Published in MedChemComm (20.02.2019)
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Journal Article
Discovery of 1,3-diethyl-7-methyl-8-(phenoxymethyl)-xanthine derivatives as novel adenosine A1 and A2A receptor antagonists
Harmse, Rozanne, van der Walt, Mietha M., Petzer, Jacobus P., Terre’Blanche, Gisella
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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Journal Article
Discovery of 1,3-diethyl-7-methyl-8-(phenoxymethyl)-xanthine derivatives as novel adenosine A 1 and A 2A receptor antagonists
Harmse, Rozanne, van der Walt, Mietha M, Petzer, Jacobus P, Terre'Blanche, Gisella
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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Journal Article
8-(3-phenylpropyl)-1,3,7-triethylxanthine is a synthetic caffeine substitute with stronger metabolic modulator activity
Carrageta, David F., Dias, Tânia R., Jarak, Ivana, Alves, Marco G., Oliveira, Pedro F., Van der Walt, Mietha M., Terre'Blanche, Gisella, Monteiro, Mariana P., Silva, Branca M.
Published in Toxicology in vitro (01.12.2018)
Published in Toxicology in vitro (01.12.2018)
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Journal Article
Methoxy substituted 2-benzylidene-1-indanone derivatives as A1 and/or A2A AR antagonists for the potential treatment of neurological conditions
Helena D Janse van Rensburg, Legoabe, Lesetja J, Terre'Blanche, Gisella, Mietha M Van der Walt
Published in MedChemComm (01.02.2019)
Published in MedChemComm (01.02.2019)
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Journal Article
The adenosine A(2A) antagonistic properties of selected C8-substituted xanthines
Van der Walt, Mietha M, Terre'Blanche, Gisella, Petzer, Anél, Lourens, Anna C U, Petzer, Jacobus P
Published in Bioorganic chemistry (01.08.2013)
Published in Bioorganic chemistry (01.08.2013)
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