Allosteric Modulation of the Adenosine A1 Receptor. Synthesis and Biological Evaluation of Novel 2-Amino-3-benzoylthiophenes as Allosteric Enhancers of Agonist Binding
van der Klein, Pieter A. M, Kourounakis, Angeliki P, IJzerman, Ad P
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Elucidation of structure-activity relationships of 2-amino-3-benzoylthiophenes: Study of their allosteric enhancing vs. antagonistic activity on adenosine A1 receptors
Kourounakis, Angeliki P., Van der Klein, Pieter A.M., Ijzerman, Ad P.
Published in Drug development research (01.04.2000)
Published in Drug development research (01.04.2000)
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Synthesis of a methyl heptaglucoside: Analogue of the phytoalexin elicitor from phytophtora megasperma
Verduyn, R., Douwes, M., van der Klein, P.A.M., Mösinger, E.M., van der Marel, G.A., van Boom, J.H.
Published in Tetrahedron (13.08.1993)
Published in Tetrahedron (13.08.1993)
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Phenyl-substituted N6-phenyladenosines and N6-phenyl-5′-N-ethylcarboxamidoadenosines with high activity at human adenosine A2B receptors
de Zwart, Maarten, de Groote, Miriam, van der Klein, Pieter A.M., van Dun, Stephanie, Bronsing, Robert, von Frijtag Drabbe Künzel, Jacobien K., Ijzerman, Ad P.
Published in Drug development research (01.02.2000)
Published in Drug development research (01.02.2000)
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A NEW AND VERSATILE PHOSPHONYLATION APPROACH
VANDERKLEIN, PAM, DREEF, CE, VANDERMAREL, GA, VANBOOM, JH
Published in Tetrahedron letters (01.01.1989)
Published in Tetrahedron letters (01.01.1989)
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