Design of Radioiodinated Pharmaceuticals: Structural Features Affecting Metabolic Stability towards in Vivo Deiodination
Cavina, Lorenzo, van der Born, Dion, Klaren, Peter H. M., Feiters, Martin C., Boerman, Otto C., Rutjes, Floris P. J. T.
Published in European journal of organic chemistry (30.06.2017)
Published in European journal of organic chemistry (30.06.2017)
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Journal Article
A Universal Procedure for the [18F]Trifluoromethylation of Aryl Iodides and Aryl Boronic Acids with Highly Improved Specific Activity
van der Born, Dion, Sewing, Claudia, Herscheid, J. (Koos) D. M., Windhorst, Albert D., Orru, Romano V. A., Vugts, Danielle J.
Published in Angewandte Chemie International Edition (06.10.2014)
Published in Angewandte Chemie International Edition (06.10.2014)
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Journal Article
Microfluidic Preparation of 89Zr-Radiolabelled Proteins by Flow Photochemistry
Earley, Daniel F., Guillou, Amaury, van der Born, Dion, Poot, Alex J., Holland, Jason P.
Published in Molecules (Basel, Switzerland) (02.02.2021)
Published in Molecules (Basel, Switzerland) (02.02.2021)
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Journal Article
Efficient One-Pot Reaction of up to Eight Components by the Union of Multicomponent Reactions
Elders, Niels, van der Born, Dion, Hendrickx, Loes J.D, Timmer, Brian J.J, Krause, Alrik, Janssen, Elwin, de Kanter, Frans J.J, Ruijter, Eelco, Orru, Romano V.A
Published in Angewandte Chemie (International ed.) (27.07.2009)
Published in Angewandte Chemie (International ed.) (27.07.2009)
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Journal Article
Synthesis, biodistribution and PET studies in rats of (18)F-Labeled bridgehead fluoromethyl analogues of WAY-100635
Al Hussainy, Rana, Verbeek, Joost, van der Born, Dion, Molthoff, Carla, Booij, Jan, Herscheid, J Koos D M
Published in Nuclear medicine and biology (01.10.2012)
Published in Nuclear medicine and biology (01.10.2012)
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Journal Article
Fluorine-18 labelled building blocks for PET tracer synthesis
van der Born, Dion, Pees, Anna, Poot, Alex J, Orru, Romano V. A, Windhorst, Albert D, Vugts, Danielle J
Published in Chemical Society reviews (31.07.2017)
Published in Chemical Society reviews (31.07.2017)
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Journal Article
Ultrafast Photoclick Reaction for Selective F-18-Positron Emission Tomography Tracer Synthesis in Flow
Fu, Youxin, Helbert, Hugo, Simeth, Nadja A., Crespi, Stefano, Spoelstra, Gerbren B., van Dijl, Jan Maarten, van Oosten, Marleen, Nazario, Luiza Reali, van der Born, Dion, Luurtsema, Gert, Szymanski, Wiktor, Elsinga, Philip H., Feringa, Ben L.
Published in Journal of the American Chemical Society (14.07.2021)
Published in Journal of the American Chemical Society (14.07.2021)
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Journal Article
Ultrafast Photoclick Reaction for Selective 18 F-Positron Emission Tomography Tracer Synthesis in Flow
Fu, Youxin, Helbert, Hugo, Simeth, Nadja A., Crespi, Stefano, Spoelstra, Gerbren B., van Dijl, Jan Maarten, van Oosten, Marleen, Nazario, Luiza Reali, van der Born, Dion, Luurtsema, Gert, Szymanski, Wiktor, Elsinga, Philip H., Feringa, Ben L.
Published in Journal of the American Chemical Society (14.07.2021)
Published in Journal of the American Chemical Society (14.07.2021)
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Journal Article
Modular Medical Imaging Agents Based on Azide–Alkyne Huisgen Cycloadditions: Synthesis and Pre‐Clinical Evaluation of 18F‐Labeled PSMA‐Tracers for Prostate Cancer Imaging
Böhmer, Verena I., Szymanski, Wiktor, Berg, Keimpe‐Oeds, Mulder, Chantal, Kobauri, Piermichele, Helbert, Hugo, Born, Dion, Reeβing, Friederike, Huizing, Anja, Klopstra, Marten, Samplonius, Douwe F., Antunes, Ines F., Sijbesma, Jürgen W. A., Luurtsema, Gert, Helfrich, Wijnand, Visser, Ton J., Feringa, Ben L., Elsinga, Philip H.
Published in Chemistry : a European journal (21.08.2020)
Published in Chemistry : a European journal (21.08.2020)
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Journal Article
Ultrafast Photoclick Reaction for Selective 18F‑Positron Emission Tomography Tracer Synthesis in Flow
Fu, Youxin, Helbert, Hugo, Simeth, Nadja A, Crespi, Stefano, Spoelstra, Gerbren B, van Dijl, Jan Maarten, van Oosten, Marleen, Nazario, Luiza Reali, van der Born, Dion, Luurtsema, Gert, Szymanski, Wiktor, Elsinga, Philip H, Feringa, Ben L
Published in Journal of the American Chemical Society (14.07.2021)
Published in Journal of the American Chemical Society (14.07.2021)
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Journal Article
Modular Medical Imaging Agents Based on Azide-Alkyne Huisgen Cycloadditions: Synthesis and Pre-Clinical Evaluation of 18 F-Labeled PSMA-Tracers for Prostate Cancer Imaging
Böhmer, Verena I, Szymanski, Wiktor, van den Berg, Keimpe-Oeds, Mulder, Chantal, Kobauri, Piermichele, Helbert, Hugo, van der Born, Dion, Reeβing, Friederike, Huizing, Anja, Klopstra, Marten, Samplonius, Douwe F, Antunes, Ines F, Sijbesma, Jürgen W A, Luurtsema, Gert, Helfrich, Wijnand, Visser, Ton J, Feringa, Ben L, Elsinga, Philip H
Published in Chemistry : a European journal (21.08.2020)
Published in Chemistry : a European journal (21.08.2020)
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Journal Article
Corrigendum: Modular Medical Imaging Agents Based on Azide–Alkyne Huisgen Cycloadditions: Synthesis and Pre‐Clinical Evaluation of 18F‐Labeled PSMA‐Tracers for Prostate Cancer Imaging
Böhmer, Verena I., Szymanski, Wiktor, Berg, Keimpe‐Oeds, Mulder, Chantal, Kobauri, Piermichele, Helbert, Hugo, Born, Dion, Reeβing, Friederike, Huizing, Anja, Klopstra, Marten, Samplonius, Douwe F., Antunes, Ines F., Sijbesma, Jürgen W. A., Luurtsema, Gert, Helfrich, Wijnand, Visser, Ton J., Feringa, Ben L., Elsinga, Philip H.
Published in Chemistry : a European journal (21.04.2021)
Published in Chemistry : a European journal (21.04.2021)
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Journal Article
Microfluidic Preparation of 89 Zr-Radiolabelled Proteins by Flow Photochemistry
Earley, Daniel F, Guillou, Amaury, van der Born, Dion, Poot, Alex J, Holland, Jason P
Published in Molecules (Basel, Switzerland) (02.02.2021)
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Published in Molecules (Basel, Switzerland) (02.02.2021)
Journal Article
Efficient synthesis of [18F]trifluoromethane and its application in the synthesis of PET tracersElectronic supplementary information (ESI) available: Synthesis and characterisation of reference compounds and experimental details. See DOI: 10.1039/c3cc37833k
van der Born, Dion, Herscheid, J. (Koos) D. M, Orru, Romano V. A, Vugts, Danielle J
Year of Publication 16.04.2013
Year of Publication 16.04.2013
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Journal Article
Tumour imaging by Positron Emission Tomography using fluorinase generated 5-[18 F]fluoro-5-deoxyribose as a novel tracer
Dall'Angelo, Sergio, Bandaranayaka, Nouchali, Windhorst, Albert D, Vugts, Danielle J, van der Born, Dion, Onega, Mayca, Schweiger, Lutz F, Zanda, Matteo, O'Hagan, David
Published in Nuclear medicine and biology (01.05.2013)
Published in Nuclear medicine and biology (01.05.2013)
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Journal Article
Design, synthesis and in vitro evaluation of bridgehead fluoromethyl analogs of N-{2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl}-N-(pyridin-2-yl) cyclohexanecarboxamide (WAY-100635) for the 5-HT1A receptor
Al Hussainy, Rana, Verbeek, Joost, van der Born, Dion, Booij, Jan, Herscheid, J. (Koos) D. M.
Published in European journal of medicinal chemistry (01.12.2011)
Published in European journal of medicinal chemistry (01.12.2011)
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Journal Article
Design, Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of Bridgehead Iodinated Analogues of N-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-N-(pyridin-2-yl)cyclohexanecarboxamide (WAY-100635) as Potential SPECT Ligands for the 5-HT1A Receptor
Al Hussainy, Rana, Verbeek, Joost, van der Born, Dion, Braker, Anton H, Leysen, Josée E, Knol, Remco J, Booij, Jan, Herscheid, J. (Koos) D. M
Published in Journal of medicinal chemistry (26.05.2011)
Published in Journal of medicinal chemistry (26.05.2011)
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Journal Article
Design, synthesis and in vitro evaluation of bridgehead fluoromethyl analogs of N-{2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl}- N-(pyridin-2-yl)cyclohexanecarboxamide (WAY-100635) for the 5-HT 1A receptor
Al Hussainy, Rana, Verbeek, Joost, van der Born, Dion, Booij, Jan, Herscheid, J(Koos) D.M.
Published in European journal of medicinal chemistry (2011)
Published in European journal of medicinal chemistry (2011)
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Journal Article
Design, Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of Bridgehead Iodinated Analogues of N -{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}- N -(pyridin-2-yl)cyclohexanecarboxamide (WAY-100635) as Potential SPECT Ligands for the 5-HT 1A Receptor
Al Hussainy, Rana, Verbeek, Joost, van der Born, Dion, Braker, Anton H., Leysen, Josée E., Knol, Remco J., Booij, Jan, Herscheid, J. (Koos) D. M.
Published in Journal of medicinal chemistry (26.05.2011)
Published in Journal of medicinal chemistry (26.05.2011)
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Journal Article