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Published in Journal of the American Chemical Society (11.10.2017)
Published in Journal of the American Chemical Society (11.10.2017)
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Role of μ-glucosidase 2 in aberrant glycosphingolipid metabolism: model of glucocerebrosidase deficiency in zebrafish
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A chemical genetic screen reveals that iminosugar inhibitors of plant glucosylceramide synthase inhibit root growth in Arabidopsis and cereals
Rugen, Michael D, Vernet, Mathieu M J L, Hantouti, Laila, Soenens, Amalia, Andriotis, Vasilios M E, Rejzek, Martin, Brett, Paul, van den Berg, Richard J B H N, Aerts, Johannes M F G, Overkleeft, Hermen S, Field, Robert A
Published in Scientific reports (06.11.2018)
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Synthesis and evaluation of homo-bivalent GnRHR ligands
Bonger, Kimberly M., van den Berg, Richard J.B.H.N., Heitman, Laura H., IJzerman, Ad P., Oosterom, Julia, Timmers, Cornelis M., Overkleeft, Herman S., van der Marel, Gijsbert A.
Published in Bioorganic & medicinal chemistry (15.07.2007)
Published in Bioorganic & medicinal chemistry (15.07.2007)
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Nanomolar affinity, iminosugar-based chemical probes for specific labeling of lysosomal glucocerebrosidase
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Published in Bioorganic & medicinal chemistry (2010)
Published in Bioorganic & medicinal chemistry (2010)
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Synthesis and evaluation of d- gluco-pyranocyclopropyl amines as potential glucosidase inhibitors
Risseeuw, Martijn D.P., van den Berg, Richard J.B.H.N., Donker-Koopman, Wilma E., van der Marel, Gijs A., Aerts, Johannes M.F.G., Overhand, Mark, Overkleeft, Herman S.
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
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Design and synthesis of 2-acetamidomethyl derivatives of isofagomine as potential inhibitors of human lysosomal β-hexosaminidases
VAN DEN BERG, Richard J. B. H. N, DONKER-KOOPMAN, Wilma, VAN BOOM, Jacques H, AERTS, Hans M. F. G, NOORT, Daan
Published in Bioorganic & medicinal chemistry (01.03.2004)
Published in Bioorganic & medicinal chemistry (01.03.2004)
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Chemical Proteomics Reveals Antibiotic Targets of Oxadiazolones in MRSA
Bakker, Alexander T., Kotsogianni, Ioli, Mirenda, Liza, Straub, Verena M., Avalos, Mariana, van den Berg, Richard J. B. H. N., Florea, Bogdan I., van Wezel, Gilles P., Janssen, Antonius P. A., Martin, Nathaniel I., van der Stelt, Mario
Published in Journal of the American Chemical Society (18.01.2023)
Published in Journal of the American Chemical Society (18.01.2023)
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Structural basis of selective cannabinoid CB2 receptor activation
Li, Xiaoting, Chang, Hao, Bouma, Jara, de Paus, Laura V., Mukhopadhyay, Partha, Paloczi, Janos, Mustafa, Mohammed, van der Horst, Cas, Kumar, Sanjay Sunil, Wu, Lijie, Yu, Yanan, van den Berg, Richard J. B. H. N., Janssen, Antonius P. A., Lichtman, Aron, Liu, Zhi-Jie, Pacher, Pal, van der Stelt, Mario, Heitman, Laura H., Hua, Tian
Published in Nature communications (15.03.2023)
Published in Nature communications (15.03.2023)
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Glycosphingolipids-Nature, Function, and Pharmacological Modulation
Wennekes, Tom, van den Berg, Richard J. B. H. N., Boot, Rolf G., van der Marel, Gijsbert A., Overkleeft, Herman S., Aerts, Johannes M. F. G.
Published in Angewandte Chemie (International ed.) (09.11.2009)
Published in Angewandte Chemie (International ed.) (09.11.2009)
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Discovery of a Photoaffinity Probe that Captures the Active Conformation of the Cannabinoid CB2 Receptor
De Paus, Laura V., An, Yu, Janssen, Antonius P. A., Berg, Richard J. B. H. N., Heitman, Laura H., Stelt, Mario
Published in Chembiochem : a European journal of chemical biology (02.04.2024)
Published in Chembiochem : a European journal of chemical biology (02.04.2024)
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Role of β-glucosidase 2 in aberrant glycosphingolipid metabolism: model of glucocerebrosidase deficiency in zebrafish
Lelieveld, Lindsey T, Mirzaian, Mina, Kuo, Chi-Lin, Artola, Marta, Ferraz, Maria J, Peter, Remco E A, Akiyama, Hisako, Greimel, Peter, van den Berg, Richard J B H N, Overkleeft, Herman S, Boot, Rolf G, Meijer, Annemarie H, Aerts, Johannes M F G
Published in Journal of lipid research (01.11.2019)
Published in Journal of lipid research (01.11.2019)
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Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding
Deng, Hui, Kooijman, Sander, van den Nieuwendijk, Adrianus M. C. H, Ogasawara, Daisuke, van der Wel, Tom, van Dalen, Floris, Baggelaar, Marc P, Janssen, Freek J, van den Berg, Richard J. B. H. N, den Dulk, Hans, Cravatt, Benjamin F, Overkleeft, Herman S, Rensen, Patrick C. N, van der Stelt, Mario
Published in Journal of medicinal chemistry (12.01.2017)
Published in Journal of medicinal chemistry (12.01.2017)
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Synthesis of Glycosylated 1‐Deoxynojirimycins Starting from Natural and Synthetic Disaccharides
Liu, Bing, van Mechelen, Jeanine, van den Berg, Richard J. B. H. N., van den Nieuwendijk, Adrianus M. C. H., Aerts, Johannes M. F. G., van der Marel, Gijsbert A., Codée, Jeroen D. C., Overkleeft, Herman S.
Published in European journal of organic chemistry (10.01.2019)
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Identification and Development of Biphenyl Substituted Iminosugars as Improved Dual Glucosylceramide Synthase/Neutral Glucosylceramidase Inhibitors
Ghisaidoobe, Amar T, van den Berg, Richard J. B. H. N, Butt, Saleem S, Strijland, Anneke, Donker-Koopman, Wilma E, Scheij, Saskia, van den Nieuwendijk, Adrianus M. C. H, Koomen, Gerrit-Jan, van Loevezijn, Arnold, Leemhuis, Mark, Wennekes, Tom, van der Stelt, Mario, van der Marel, Gijsbert A, van Boeckel, Constant A. A, Aerts, Johannes M. F. G, Overkleeft, Herman S
Published in Journal of medicinal chemistry (13.11.2014)
Published in Journal of medicinal chemistry (13.11.2014)
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Two-step activity-based protein profiling of diacylglycerol lipase
van Rooden, Eva J., Kreekel, Roy, Hansen, Thomas, Janssen, Antonius P. A., van Esbroeck, Annelot C. M., den Dulk, Hans, van den Berg, Richard J. B. H. N., Codee, Jeroen D. C., van der Stelt, Mario
Published in Organic & biomolecular chemistry (2018)
Published in Organic & biomolecular chemistry (2018)
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Development of Adamantan-1-yl-methoxy-Functionalized 1-Deoxynojirimycin Derivatives as Selective Inhibitors of Glucosylceramide Metabolism in Man
Wennekes, Tom, van den Berg, Richard J. B. H. N, Donker, Wilma, van der Marel, Gijsbert A, Strijland, Anneke, Aerts, Johannes M. F. G, Overkleeft, Herman S
Published in Journal of organic chemistry (16.02.2007)
Published in Journal of organic chemistry (16.02.2007)
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Synthesis of a Panel of Carbon-13-Labelled (Glyco)Sphingolipids
Wisse, Patrick, Gold, Henrik, Mirzaian, Mina, Ferraz, Maria J., Lutteke, Ginger, van den Berg, Richard J. B. H. N., van den Elst, Hans, Lugtenburg, Johan, van der Marel, Gijsbert A., Aerts, Johannes M. F. G., Codée, Jeroen D. C., Overkleeft, Herman S.
Published in European journal of organic chemistry (01.04.2015)
Published in European journal of organic chemistry (01.04.2015)
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Synthesis of 6‑Hydroxysphingosine and α‑Hydroxy Ceramide Using a Cross-Metathesis Strategy
Wisse, Patrick, de Geus, Mark A. R, Cross, Gen, van den Nieuwendijk, Adrianus M. C. H, van Rooden, Eva J, van den Berg, Richard J. B. H. N, Aerts, Johannes M. F. G, van der Marel, Gijsbert A, Codée, Jeroen D. C, Overkleeft, Herman S
Published in Journal of organic chemistry (17.07.2015)
Published in Journal of organic chemistry (17.07.2015)
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ortho-Carborane-Modified N-Substituted Deoxynojirimycins
Hoogendoorn, Sascha, Mock, Elliot D., Strijland, Anneke, Donker-Koopman, Wilma E., van den Elst, Hans, van den Berg, Richard J. B. H. N., Aerts, Johannes M. F. G., van der Marel, Gijsbert A., Overkleeft, Herman S.
Published in European journal of organic chemistry (01.07.2015)
Published in European journal of organic chemistry (01.07.2015)
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