항-191P4D12 항체 약물 컨쥬게이트를 포함하는 약제학적 조성물 및 이의 사용 방법
VAN SCHRAVENDIJK MARIE ROSE, SUN YINGQING, MCGARVEY ORLA, RATNASWAMY GAYATHRI
Year of Publication 17.08.2021
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Year of Publication 17.08.2021
Patent
Structural Basis of Src Tyrosine Kinase Inhibition with a New Class of Potent and Selective Trisubstituted Purine-based Compounds
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Published in Chemical biology & drug design (01.01.2006)
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A ligand-reversible dimerization system for controlling protein–protein interactions
Rollins, C T, Rivera, V M, Woolfson, D N, Keenan, T, Hatada, M, Adams, S E, Andrade, L J, Yaeger, D, van Schravendijk, M R, Holt, D A, Gilman, M, Clackson, T
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Published in Proceedings of the National Academy of Sciences - PNAS (20.06.2000)
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Shakespeare, William, Yang, Michael, Bohacek, Regine, Cerasoli, Franklin, Stebbins, Karin, Sundaramoorthi, Raji, Azimioara, Mihai, Vu, Chi, Pradeepan, Selvi, Metcalf, Chester, Haraldson, Chad, Merry, Taylor, Dalgarno, David, Narula, Surinder, Hatada, Marcos, Lu, Xiaode, van Schravendijk, Marie Rose, Adams, Susan, Violette, Shelia, Smith, Jeremy, Guan, Wei, Bartlett, Catherine, Herson, Jay, Iuliucci, John, Weigele, Manfred, Sawyer, Tomi
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Published in Proceedings of the National Academy of Sciences - PNAS (15.08.2000)
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Bone-Targeted 2,6,9-Trisubstituted purines: novel inhibitors of Src tyrosine kinase for the treatment of bone diseases
Wang, Yihan, Metcalf, Chester A., Shakespeare, William C., Sundaramoorthi, Raji, Keenan, Terence P., Bohacek, Regine S., van Schravendijk, Marie Rose, Violette, Shiela M., Narula, Surinder S., Dalgarno, David C., Haraldson, Chad, Keats, Jeffrey, Liou, Shuenn, Mani, Ukti, Pradeepan, Selvi, Ram, Mary, Adams, Susan, Weigele, Manfred, Sawyer, Tomi K.
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Lipophilic bis-arylsulfonates as inhibitors of the CD4-gp120 interaction
Patch, Raymond J., Roberts, John C., Huai Gao, Zhan Shi, Gopalsamy, Ariamala, Kongsjahju, Azis, Daniels, Kevin, Kowalczyk, Paul J., van Schravendijk, Marie-Rose, Gordon, Kristin A., Pallai, Peter V.
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The characterization of two monoclonal antibodies which react with high molecular weight antigens of asexual Plasmodium falciparum
Handunnetti, Shiroma M., Pasloske, Brittan L., van Schravendijk, Marie-Rose, Aguiar, Joao C., Taraschi, Theodore F., Gormley, Jill Ann, Howard, Russell J.
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Vu, Chi B, Corpuz, Evelyn G, Merry, Taylor J, Pradeepan, Selvaluxmi G, Bartlett, Catherine, Bohacek, Regine S, Botfield, Martyn C, Eyermann, Charles J, Lynch, Berkley A, MacNeil, Ian A, Ram, Mary K, van Schravendijk, Marie Rose, Violette, Shelia, Sawyer, Tomi K
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SAR of Carbon-Linked, 2-Substituted Purines: Synthesis and Characterization of AP23451 as a novel Bone-Targeted Inhibitor of Src Tyrosine Kinase With In Vivo Anti-Resorptive Activity
Shakespeare, William C, Wang, Yihan, Bohacek, Regine, Keenan, Terry, Sundaramoorthi, Raji, Metcalf, Chet III, Dilauro, Anne, Roeloffzen, Sonya, Liu, Shuangying, Saltmarsh, Jennifer, Paramanathan, Guru, Dalgarno, David, Narula, Surinder, Pradeepan, Selvi, van Schravendijk, Marie Rose, Keats, Jeff, Ram, Mary, Liou, Shuenn, Adams, Susan, Wardwell, Scott, Bogus, Julie, Iuliucci, John, Weigele, Manfred, Xing, Lianping, Boyce, Brendan, Sawyer, Tomi K
Published in Chemical biology & drug design (01.02.2008)
Published in Chemical biology & drug design (01.02.2008)
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Investigating Protein−Ligand Interactions with a Mutant FKBP Possessing a Designed Specificity Pocket
Yang, Wu, Rozamus, Leonard W, Narula, Surinder, Rollins, Carl T, Yuan, Ruth, Andrade, Lawrence J, Ram, Mary K, Phillips, Thomas B, van Schravendijk, Marie Rose, Dalgarno, David, Clackson, Tim, Holt, Dennis A
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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