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Design, Synthesis, and Structure–Activity Relationship of 2‑(Piperazin-1-yl)quinazolin-4(3H)‑one Derivatives as Active Agents against Toxoplasma gondii
Deng, Yu, Yu, Yuan-Di, Song, Chao, Xu, Guo-Yang, Xu, Yue, Ye, Chang-Ju
Published in Journal of agricultural and food chemistry (12.03.2025)
Published in Journal of agricultural and food chemistry (12.03.2025)
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The structure – Activity correlation in the family of dicationic imidazolium surfactants: Antimicrobial properties and cytotoxic effect
Voloshina, Alexandra D., Gumerova, Syumbelya K., Sapunova, Аnastasiia S., Kulik, Natalia V., Mirgorodskaya, Alla B., Kotenko, Alla A., Prokopyeva, Tatiana M., Mikhailov, Vasilii A., Zakharova, Lucia Ya, Sinyashin, Oleg G.
Published in Biochimica et biophysica acta. General subjects (01.12.2020)
Published in Biochimica et biophysica acta. General subjects (01.12.2020)
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Recent Advances in Polysaccharides Derived from the Genus Panax: Preparation Strategies, Structural Profiles, Functional Properties and Structure–Activity Relationships
Bu, Yingxuan, Liu, Yupeng, Zhu, Lingyan, Gan, Xiaona, Jiang, Shenggui, Zhang, Xiaoyu, Dilixiati, Munisa, Bai, Muwei, Zeng, Jiani, Shi, Songshan, Li, Tingzhao, Li, Bo, Wang, Shunchun, Wang, Huijun
Published in Journal of agricultural and food chemistry (27.11.2024)
Published in Journal of agricultural and food chemistry (27.11.2024)
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Structure–Activity Relationships and Therapeutic Potentials of 5‑HT7 Receptor Ligands: An Update
Modica, Maria N, Lacivita, Enza, Intagliata, Sebastiano, Salerno, Loredana, Romeo, Giuseppe, Pittalà, Valeria, Leopoldo, Marcello
Published in Journal of medicinal chemistry (11.10.2018)
Published in Journal of medicinal chemistry (11.10.2018)
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Enzyme inhibitory activities an insight into the structure–Activity relationship of biscoumarin derivatives
Faisal, Muhammad, Saeed, Aamer, Shahzad, Danish, Fattah, Tanzeela Abdul, Lal, Bhajan, Channar, Pervaiz Ali, Mahar, Jamaluddin, Saeed, Shomaila, Mahesar, Parvez Ali, Larik, Fayaz Ali
Published in European journal of medicinal chemistry (01.12.2017)
Published in European journal of medicinal chemistry (01.12.2017)
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Tyrosinase inhibitory peptides: Structure-activity relationship study on peptide chemical properties, terminal preferences and intracellular regulation of melanogenesis signaling pathways
Yap, Pei-Gee, Gan, Chee-Yuen
Published in Biochimica et biophysica acta. General subjects (01.01.2024)
Published in Biochimica et biophysica acta. General subjects (01.01.2024)
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Structure–Activity Relationship of Terpenes with Anti‐Inflammatory Profile – A Systematic Review
Santana Souza, Marilia Trindade, Almeida, Jackson Roberto Guedes da Silva, Souza Araujo, Adriano Antunes, Duarte, Marcelo Cavalcante, Gelain, Daniel Pens, Moreira, José Cláudio Fonseca, Santos, Marcio Roberto Viana, Quintans‐Júnior, Lucindo José
Published in Basic & clinical pharmacology & toxicology (01.09.2014)
Published in Basic & clinical pharmacology & toxicology (01.09.2014)
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Structure, Activity, and Function of Protein Methyltransferases
Year of Publication 2022
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Flavonols and flavones as BACE-1 inhibitors: Structure–activity relationship in cell-free, cell-based and in silico studies reveal novel pharmacophore features
Shimmyo, Yoshiari, Kihara, Takeshi, Akaike, Akinori, Niidome, Tetsuhiro, Sugimoto, Hachiro
Published in Biochimica et biophysica acta (01.05.2008)
Published in Biochimica et biophysica acta (01.05.2008)
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Serotonin 5-HT7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders
Leopoldo, Marcello, Lacivita, Enza, Berardi, Francesco, Perrone, Roberto, Hedlund, Peter B.
Published in Pharmacology & therapeutics (Oxford) (01.02.2011)
Published in Pharmacology & therapeutics (Oxford) (01.02.2011)
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Immunomodulatory Effects of Enzymatic-Synthesized α‑Galactooligosaccharides and Evaluation of the Structure–Activity Relationship
Dai, Zhuqing, Lyu, Wanyong, Xiang, Xiaoli, Tang, Yuhong, Hu, Bing, Ou, Shiyi, Zeng, Xiaoxiong
Published in Journal of agricultural and food chemistry (29.08.2018)
Published in Journal of agricultural and food chemistry (29.08.2018)
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Anti-HIV-1 activity and structure–activity-relationship study of a fucosylated glycosaminoglycan from an echinoderm by targeting the conserved CD4 induced epitope
Lian, Wu, Wu, Mingyi, Huang, Ning, Gao, Na, Xiao, Chuang, Li, Zi, Zhang, Zhigang, Zheng, Yongtang, Peng, Wenlie, Zhao, Jinhua
Published in Biochimica et biophysica acta (01.10.2013)
Published in Biochimica et biophysica acta (01.10.2013)
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Evaluation of human intestinal absorption data and subsequent derivation of a quantitative structure–activity relationship (QSAR) with the Abraham descriptors
Zhao, Yuan H., Le, Joelle, Abraham, Michael H., Hersey, Anne, Eddershaw, Peter J., Luscombe, Chris N., Boutina, Darko, Beck, Gordon, Sherborne, Brad, Cooper, Ian, Platts, James A.
Published in Journal of pharmaceutical sciences (01.06.2001)
Published in Journal of pharmaceutical sciences (01.06.2001)
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