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G-quadruplexes in human promoters: A challenge for therapeutic applications
Rigo, Riccardo, Palumbo, Manlio, Sissi, Claudia
Published in Biochimica et biophysica acta. General subjects (01.05.2017)
Published in Biochimica et biophysica acta. General subjects (01.05.2017)
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One stone two birds: Introducing piperazine into a series of nucleoside derivatives as potent and selective PRMT5 inhibitors
Li, Huaxuan, Yang, Hong, Liu, Li, Zheng, Jiahong, Shi, Qiongyu, Li, Bang, Wang, Xingcan, Zhang, Ying, Zhou, Ruilin, Zhang, Jian, Chen, Zhong-Zhu, Wang, Chang-Yun, Wang, Yuanxiang, Huang, Xun, Liu, Zhiqing
Published in European journal of medicinal chemistry (05.01.2025)
Published in European journal of medicinal chemistry (05.01.2025)
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Structure-function analyses of microsomal triglyceride transfer protein missense mutations in abetalipoproteinemia and hypobetalipoproteinemia subjects
Walsh, Meghan T., Di Leo, Enza, Okur, Ilyas, Tarugi, Patrizia, Hussain, M. Mahmood
Published in Biochimica et biophysica acta (01.11.2016)
Published in Biochimica et biophysica acta (01.11.2016)
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Isomerization of aspartyl residues in crystallins and its influence upon cataract
Fujii, Noriko, Takata, Takumi, Fujii, Norihiko, Aki, Kenzo
Published in Biochimica et biophysica acta (01.01.2016)
Published in Biochimica et biophysica acta (01.01.2016)
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PI-2620 Lead Optimization Highlights the Importance of Off-Target Assays to Develop a PET Tracer for the Detection of Pathological Aggregated Tau in Alzheimer’s Disease and Other Tauopathies
Kroth, Heiko, Oden, Felix, Molette, Jerome, Schieferstein, Hanno, Gabellieri, Emanuele, Mueller, Andre, Berndt, Mathias, Sreenivasachary, Nampally, Serra, Andreia Monica, Capotosti, Francesca, Schmitt-Willich, Heribert, Hickman, David, Pfeifer, Andrea, Dinkelborg, Ludger, Stephens, Andrew
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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The prion protein and its ligands: Insights into structure-function relationships
Shafiq, Mohsin, Da Vela, Stefano, Amin, Ladan, Younas, Neelam, Harris, David A., Zerr, Inga, Altmeppen, Hermann C., Svergun, Dmitri, Glatzel, Markus
Published in Biochimica et biophysica acta. Molecular cell research (01.06.2022)
Published in Biochimica et biophysica acta. Molecular cell research (01.06.2022)
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Proteases—From Basic Structure to Function to Drug Design as Targeted Therapy
Year of Publication 2021
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Phenotypic and biochemical analysis of an international cohort of individuals with variants in NAA10 and NAA15
Cheng, Hanyin, Gottlieb, Leah, Marchi, Elaine, Kleyner, Robert, Bhardwaj, Puja, Rope, Alan F, Rosenheck, Sarah, Moutton, Sébastien, Philippe, Christophe, Eyaid, Wafaa, Alkuraya, Fowzan S, Toribio, Janet, Mena, Rafael, Prada, Carlos E, Stessman, Holly, Bernier, Raphael, Wermuth, Marieke, Kauffmann, Birgit, Blaumeiser, Bettina, Kooy, R Frank, Baralle, Diana, Mancini, Grazia M S, Conway, Simon J, Xia, Fan, Chen, Zhao, Meng, Linyan, Mihajlovic, Ljubisa, Marmorstein, Ronen, Lyon, Gholson J
Published in Human molecular genetics (01.09.2019)
Published in Human molecular genetics (01.09.2019)
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Abstract 1359: Identification of a novel class of compounds as proteasome inhibitors: Synthesis and structure activity relationship studies of PI-1833 library
Ozcan, Sevil, Aslamuzzaman, Kazi, Marsilio, Frank, Daniel, Kenyon, Brooks, Wesley, Guida, Wayne, Lawrence, Harshani, Sebti, Said
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Amiselimod, a novel sphingosine 1‐phosphate receptor‐1 modulator, has potent therapeutic efficacy for autoimmune diseases, with low bradycardia risk
Sugahara, Kunio, Maeda, Yasuhiro, Shimano, Kyoko, Mogami, Akira, Kataoka, Hirotoshi, Ogawa, Kei, Hikida, Kumiko, Kumagai, Hiroshi, Asayama, Mahoko, Yamamoto, Toshinobu, Harada, Tomohiko, Ni, Pingping, Inoue, Shinsuke, Kawaguchi, Atsuhiro
Published in British journal of pharmacology (01.01.2017)
Published in British journal of pharmacology (01.01.2017)
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Novel mitochondrial and DNA damaging fluorescent Calix[4]arenes bearing isatin groups as aromatase inhibitors: Design, synthesis and anticancer activity
Oguz, Alev, Saglik, Begum Nurpelin, Oguz, Mehmet, Ozturk, Bahadir, Yilmaz, Mustafa
Published in Bioorganic & medicinal chemistry (15.01.2024)
Published in Bioorganic & medicinal chemistry (15.01.2024)
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Structural insights into the activation mechanisms of human HtrA serine proteases
Zurawa-Janicka, Dorota, Wenta, Tomasz, Jarzab, Miroslaw, Skorko-Glonek, Joanna, Glaza, Przemyslaw, Gieldon, Artur, Ciarkowski, Jerzy, Lipinska, Barbara
Published in Archives of biochemistry and biophysics (01.05.2017)
Published in Archives of biochemistry and biophysics (01.05.2017)
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Carbon-based metal-free oxygen reduction reaction electrocatalysts: past, present and future
An, Fu, Bao, Xiao-qing, Deng, Xiao-yang, Ma, Zi-zai, Wang, Xiao-guang
Published in New carbon materials (01.04.2022)
Published in New carbon materials (01.04.2022)
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Tandem application of ligand-based virtual screening and G4-OAS assay to identify novel G-quadruplex-targeting chemotypes
Musumeci, Domenica, Amato, Jussara, Zizza, Pasquale, Platella, Chiara, Cosconati, Sandro, Cingolani, Chiara, Biroccio, Annamaria, Novellino, Ettore, Randazzo, Antonio, Giancola, Concetta, Pagano, Bruno, Montesarchio, Daniela
Published in Biochimica et biophysica acta. General subjects (01.05.2017)
Published in Biochimica et biophysica acta. General subjects (01.05.2017)
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Dynamic membrane interactions of antibacterial and antifungal biomolecules, and amyloid peptides, revealed by solid-state NMR spectroscopy
Naito, Akira, Matsumori, Nobuaki, Ramamoorthy, Ayyalusamy
Published in Biochimica et biophysica acta. General subjects (01.02.2018)
Published in Biochimica et biophysica acta. General subjects (01.02.2018)
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Crucial role for the VWF A1 domain in binding to type IV collagen
Flood, Veronica H., Schlauderaff, Abraham C., Haberichter, Sandra L., Slobodianuk, Tricia L., Jacobi, Paula M., Bellissimo, Daniel B., Christopherson, Pamela A., Friedman, Kenneth D., Gill, Joan Cox, Hoffmann, Raymond G., Montgomery, Robert R.
Published in Blood (02.04.2015)
Published in Blood (02.04.2015)
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Binding Sites for Acylated Trehalose Analogs of Glycolipid Ligands on an Extended Carbohydrate Recognition Domain of the Macrophage Receptor Mincle
Feinberg, Hadar, Rambaruth, Neela D.S., Jégouzo, Sabine A.F., Jacobsen, Kristian M., Djurhuus, Rasmus, Poulsen, Thomas B., Weis, William I., Taylor, Maureen E., Drickamer, Kurt
Published in The Journal of biological chemistry (30.09.2016)
Published in The Journal of biological chemistry (30.09.2016)
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