Loading…
A Dipolar Cycloaddition Reaction To Access 6‑Methyl-4,5,6,7-tetrahydro‑1H‑[1,2,3]triazolo[4,5‑c]pyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate
Chrovian, Christa C, Soyode-Johnson, Akinola, Peterson, Alexander A, Gelin, Christine F, Deng, Xiaohu, Dvorak, Curt A, Carruthers, Nicholas I, Lord, Brian, Fraser, Ian, Aluisio, Leah, Coe, Kevin J, Scott, Brian, Koudriakova, Tatiana, Schoetens, Freddy, Sepassi, Kia, Gallacher, David J, Bhattacharya, Anindya, Letavic, Michael A
Published in Journal of medicinal chemistry (11.01.2018)
Published in Journal of medicinal chemistry (11.01.2018)
Get full text
Journal Article
Loading…
A Dipolar Cycloaddition Reaction To Access 6-Methyl-4,5,6,7-tetrahydro-1H-1,2,3triazolo4,5-cpyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate
Chrovian, Christa C, Soyode-Johnson, Akinola, Peterson, Alexander A, Gelin, Christine F, Deng, Xiaohu, Dvorak, Curt A, Carruthers, Nicholas I, Lord, Brian, Fraser, Ian, Aluisio, Leah, Coe, Kevin J, Scott, Brian, Koudriakova, Tatiana, Schoetens, Freddy, Sepassi, Kia, Gallacher, David J, Bhattacharya, Anindya, Letavic, Michael A
Published in Journal of medicinal chemistry (11.01.2018)
Published in Journal of medicinal chemistry (11.01.2018)
Get full text
Journal Article
Loading…
Loading…
Organic functionalization of carbon nanostructures via 1,3-dipolar cycloadditions
Quintana, Mildred, Grzelczak, Marek, Prato, Maurizio
Published in Physica Status Solidi (b) (01.12.2010)
Published in Physica Status Solidi (b) (01.12.2010)
Get full text
Journal Article
Conference Proceeding
Loading…
Spiro‐2‐oxindoles via 1,3‐dipolar cycloadditions. A decade update
Molteni, Giorgio, Silvani, Alessandra
Published in European journal of organic chemistry (19.03.2021)
Published in European journal of organic chemistry (19.03.2021)
Get full text
Journal Article
Loading…
Loading…
Novel Glycoconjugate of 8-Fluoro Norfloxacin Derivatives as Gentamicin-resistant Staphylococcus aureus Inhibitors: Synthesis and Molecular Modelling Studies
Azad, Chandra S., Bhunia, Shome S., Krishna, Atul, Shukla, Praveen K., Saxena, Anil K.
Published in Chemical biology & drug design (01.10.2015)
Published in Chemical biology & drug design (01.10.2015)
Get full text
Journal Article
Loading…
Loading…
Anion radical [2 + 2] cycloaddition as a mechanistic probe: Stoichiometry- and concentration-dependent partitioning of electron-transfer and alkylation pathways in the reaction of the Gilman reagent Me2CuLi.LiI with bis(enones)
JINGKUI YANG, CAUBLE, David F, BERRO, Adam J, BAULD, Nathan L, KRISCHE, Michael J
Published in Journal of organic chemistry (12.11.2004)
Get full text
Published in Journal of organic chemistry (12.11.2004)
Journal Article
Loading…