Stereocontrolled synthesis of 5-azaspiro[2.3]hexane derivatives as conformationally "frozen" analogues of L-glutamic acid
Bechi, Beatrice, Amantini, David, Tintori, Cristina, Botta, Maurizio, Fabio, Romano di
Published in Beilstein journal of organic chemistry (14.05.2014)
Published in Beilstein journal of organic chemistry (14.05.2014)
Get full text
Journal Article
Synthesis and structure–activity relationship of N-(3-azabicyclo[3.1.0]hex-6-ylmethyl)-5-(2-pyridinyl)-1,3-thiazol-2-amines derivatives as NPY Y5 antagonists
Biagetti, Matteo, Leslie, Colin Philip, Mazzali, Angelica, Seri, Catia, Pizzi, Domenica Antonia, Bentley, Jonathan, Genski, Thorsten, Fabio, Romano Di, Zonzini, Laura, Caberlotto, Laura
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Get full text
Journal Article
Role of orexin-1 receptor mechanisms on compulsive food consumption in a model of binge eating in female rats
Piccoli, Laura, Micioni Di Bonaventura, Maria Vittoria, Cifani, Carlo, Costantini, Vivian J A, Massagrande, Mario, Montanari, Dino, Martinelli, Prisca, Antolini, Marinella, Ciccocioppo, Roberto, Massi, Maurizio, Merlo-Pich, Emilio, Di Fabio, Romano, Corsi, Mauro
Published in Neuropsychopharmacology (New York, N.Y.) (01.08.2012)
Published in Neuropsychopharmacology (New York, N.Y.) (01.08.2012)
Get full text
Journal Article
Prdm16-mediated H3K9 methylation controls fibro-adipogenic progenitors identity during skeletal muscle repair
Biferali, Beatrice, Bianconi, Valeria, Perez, Daniel Fernandez, Kronawitter, Sophie Pöhle, Marullo, Fabrizia, Maggio, Roberta, Santini, Tiziana, Polverino, Federica, Biagioni, Stefano, Summa, Vincenzo, Toniatti, Carlo, Pasini, Diego, Stricker, Sigmar, Di Fabio, Romano, Chiacchiera, Fulvio, Peruzzi, Giovanna, Mozzetta, Chiara
Published in Science advances (01.06.2021)
Published in Science advances (01.06.2021)
Get full text
Journal Article
Efficient synthesis of a novel euchromatic histone methyl transferase 2 (G9a) inhibitor
Gornati, Davide, Sinisi, Roberta, Bertuolo, Stefania, De Matteo, Marilenia, Di Fabio, Romano
Published in Results in Chemistry (01.01.2022)
Published in Results in Chemistry (01.01.2022)
Get full text
Journal Article
Stereoselective Synthesis of 3-Substituted Tetrahydropyrazinoisoquinolines via Intramolecular Cyclization of Enantiomerically Enriched Dihydro-2H-pyrazines
Reginato, Gianna, Catalani, Maria Pia, Pezzati, Bernardo, Di Fabio, Romano, Bernardelli, Andrea, Curcuruto, Ornella, Moro, Elisa, Pozzan, Alfonso, Mordini, Alessandro
Published in Organic letters (06.02.2015)
Published in Organic letters (06.02.2015)
Get full text
Journal Article
Discovery process and pharmacological characterization of a novel dual orexin 1 and orexin 2 receptor antagonist useful for treatment of sleep disorders
Di Fabio, Romano, Pellacani, Annalisa, Faedo, Stefania, Roth, Adelheid, Piccoli, Laura, Gerrard, Philip, Porter, Rod A., Johnson, Christopher N., Thewlis, Kevin, Donati, Daniele, Stasi, Luigi, Spada, Simone, Stemp, Geoffrey, Nash, David, Branch, Clive, Kindon, Leanda, Massagrande, Mario, Poffe, Alessandro, Braggio, Simone, Chiarparin, Elisabetta, Marchioro, Carla, Ratti, Emiliangelo, Corsi, Mauro
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Get full text
Journal Article
Discovery of NBI-77860/GSK561679, a potent corticotropin-releasing factor (CRF 1) receptor antagonist with improved pharmacokinetic properties
Tellew, John E., Lanier, Marion, Moorjani, Manisha, Lin, Emily, Luo, Zhiyong, Slee, Deborah H., Zhang, Xiaohu, Hoare, Sam R.J., Grigoriadis, Dimitri E., Denis, Yves St, Fabio, Romano Di, Modugno, Enza Di, Saunders, John, Williams, John P.
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
Get full text
Journal Article
Discovery Process and Pharmacological Characterization of 2-(S)-(4-Fluoro-2-methylphenyl)piperazine-1-carboxylic Acid [1-(R)-(3,5-Bis-trifluoromethylphenyl)ethyl]methylamide (Vestipitant) as a Potent, Selective, and Orally Active NK1 Receptor Antagonist
Di Fabio, Romano, Griffante, Cristiana, Alvaro, Giuseppe, Pentassuglia, Giorgio, Pizzi, Domenica A, Donati, Daniele, Rossi, Tino, Guercio, Giuseppe, Mattioli, Mario, Cimarosti, Zadeo, Marchioro, Carla, Provera, Stefano, Zonzini, Laura, Montanari, Dino, Melotto, Sergio, Gerrard, Philip A, Trist, David G, Ratti, Emiliangelo, Corsi, Mauro
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
Get full text
Journal Article
Synthesis and Pharmacological Characterization of Novel Druglike Corticotropin-Releasing Factor 1 Antagonists
Fabio, Romano Di, St-Denis, Yves, Sabbatini, Fabio M, Andreotti, Daniele, Arban, Roberto, Bernasconi, Giovanni, Braggio, Simone, Blaney, Frank E, Capelli, Anna M, Castiglioni, Emiliano, Modugno, Enza Di, Donati, Daniele, Fazzolari, Elettra, Ratti, Emiliangelo, Feriani, Aldo, Contini, Stefania, Gentile, Gabriella, Ghirlanda, Damiano, Provera, Stefano, Marchioro, Carla, Roberts, Karen L, Mingardi, Anna, Mattioli, Mario, Nalin, Arnaldo, Pavone, Francesca, Spada, Simone, Trist, David G, Worby, Angela
Published in Journal of medicinal chemistry (11.12.2008)
Published in Journal of medicinal chemistry (11.12.2008)
Get full text
Journal Article
From pyrroles to 1 -oxo -2,3,4,9 -tetrahydro -1H-β -carbolines : A new class of orally bioavailable mGluR1 antagonists
DI FABIO, Romano, MICHELI, Fabrizio, TRANQUILLINI, Maria Elvira, VITULLI, Giovanni, ALVARO, Giuseppe, CAVANNI, Paolo, DONATI, Daniele, GAGLIARDI, Tatiana, FONTANA, Gabriele, GIOVANNINI, Riccardo, MAFFEIS, Micaela, MINGARDI, Anna
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
Get full text
Journal Article
Stereospecific synthesis and structure–activity relationships of unsymmetrical 4,4-diphenylbut-3-enyl derivatives of nipecotic acid as GAT-1 inhibitors
Pizzi, Domenica A., Leslie, Colin P., Fabio, Romano Di, Seri, Catia, Bernasconi, Giovanni, Squaglia, Michela, Carnevale, Gennaro, Falchi, Alessandro, Greco, Elisabetta, Mangiarini, Laura, Negri, Michele
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Get full text
Journal Article
Dopamine D 3 receptor antagonists: The quest for a potentially selective PET ligand. Part one: Lead identification
Holmes, Ian P., Micheli, Fabrizio, Gaines, Simon, Lorthioir, Olivier, Watson, Steve P., Fabio, Romano Di, Gentile, Gabriella, Heidbreder, Christian, Savoia, Chiara, Worby, Angela
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Get full text
Journal Article
Triazolyl Azabicyclo[3.1.0]hexanes: a Class of Potent and Selective Dopamine D 3 Receptor Antagonists
Bonanomi, Giorgio, Braggio, Simone, Capelli, Anna Maria, Checchia, Anna, Di Fabio, Romano, Marchioro, Carla, Tarsi, Luca, Tedesco, Giovanna, Terreni, Silvia, Worby, Angela, Heibreder, Christian, Micheli, Fabrizio
Published in ChemMedChem (03.05.2010)
Published in ChemMedChem (03.05.2010)
Get full text
Journal Article
New fused benzazepine as selective D 3 receptor antagonists. Synthesis and biological evaluation. Part one: [h]-fused tricyclic systems
Micheli, Fabrizio, Bonanomi, Giorgio, Braggio, Simone, Capelli, Anna Maria, Celestini, Paolo, Damiani, Federica, Fabio, Romano Di, Donati, Daniele, Gagliardi, Stefania, Gentile, Gabriella, Hamprecht, Dieter, Petrone, Marcella, Radaelli, Stefano, Tedesco, Giovanna, Terreni, Silvia, Worby, Angela, Heidbreder, Christian
Published in Bioorganic & medicinal chemistry letters (01.02.2008)
Published in Bioorganic & medicinal chemistry letters (01.02.2008)
Get full text
Journal Article
Pyrrolo[1,2- a]pyrazine and pyrazolo[1,5- a]pyrazine: Novel, potent, and selective series of Vasopressin 1b receptor antagonists
Arban, Roberto, Bianchi, Federica, Buson, Alberto, Cremonesi, Susanna, Fabio, Romano Di, Gentile, Gabriella, Micheli, Fabrizio, Pasquarello, Alessandra, Pozzan, Alfonso, Tarsi, Luca, Terreni, Silvia, Tonelli, Federica
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Get full text
Journal Article
Triazolyl Azabicyclo[3.1.0]hexanes: a Class of Potent and Selective Dopamine D3 Receptor Antagonists
Bonanomi, Giorgio, Braggio, Simone, Capelli, Anna Maria, Checchia, Anna, Di Fabio, Romano, Marchioro, Carla, Tarsi, Luca, Tedesco, Giovanna, Terreni, Silvia, Worby, Angela, Heibreder, Christian, Micheli, Fabrizio
Published in ChemMedChem (03.05.2010)
Published in ChemMedChem (03.05.2010)
Get full text
Journal Article
Azabicyclo[3.1.0]hexane-1-carbohydrazides as Potent and Selective GHSR1a Ligands Presenting a Specific in vivo Behavior
Sabbatini, Fabio Maria, Melotto, Sergio, Bernasconi, Giovanni, Bromidge, Steve M., D'Adamo, Lucilla, Rinaldi, Marilisa, Savoia, Chiara, Mundi, Claudia, Di Francesco, Carla, Zonzini, Laura, Costantini, Vivian J. A., Perini, Benedetta, Valerio, Enzo, Pozzan, Alfonso, Perdonà, Elisabetta, Visentini, Filippo, Corsi, Mauro, Di Fabio, Romano
Published in ChemMedChem (04.11.2011)
Published in ChemMedChem (04.11.2011)
Get full text
Journal Article