Structure-Activity Studies on the Corticotropin Releasing Factor Antagonist Astressin, leading to a Minimal Sequence necessary for Antagonistic Activity
Rijkers, Dirk T.S, Kruijtzer, John A.W, van Oostenbrugge, Marja, Ronken, Eric, den Hartog, Jack A.J, Liskamp, Rob M.J
Published in Chembiochem : a European journal of chemical biology (05.03.2004)
Published in Chembiochem : a European journal of chemical biology (05.03.2004)
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Design and Synthesis of an orally active GPIIb/IIIa antagonist based on a phenylpiperazine scaffold
van Maarseveen, Jan H, den Hartog, Jack A.J, Tipker, Koos, Reinders, Jan-Hendrik, Brakkee, Joost, Schön, Uwe, Kehrbach, Wolfgang, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
Published in Bioorganic & medicinal chemistry letters (16.06.1998)
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A straightforward synthesis of 1,3-dichloro-5,8-dihydroisoquinoline by consecutive Stille cross-coupling and metathesis reactions
van den Hoogenband, Adri, den Hartog, Jack A.J., Faber-Hilhorst, Nancy, Lange, Jos H.M., Terpstra, Jan Willem
Published in Tetrahedron letters (02.09.2009)
Published in Tetrahedron letters (02.09.2009)
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Synthesis and biological activity of N-terminal lipidated and/or fluorescently labeled conjugates of astressin as corticotropin releasing factor antagonists
Rijkers, Dirk T.S., den Hartog, Jack A.J., Liskamp, Rob M.J.
Published in Bioorganic & medicinal chemistry (01.10.2004)
Published in Bioorganic & medicinal chemistry (01.10.2004)
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Journal Article
An optimized solid phase synthesis strategy- including on-resin lactamization-of astressin, its retro-, inverso-, and retro-inverso isomers as corticotropin releasing factor antagonists
Rijkers, Dirk T. S., den Hartog, Jack A. J., Liskamp, Rob M. J.
Published in Biopolymers (01.02.2002)
Published in Biopolymers (01.02.2002)
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Journal Article
Two novel syntheses of the histamine H 3 antagonist thioperamide
Lange, Jos H.M., Wals, Henri C., den Hoogenband, Adri van, de Kuilen, Aalt van, den Hartog, Jack A.J.
Published in Tetrahedron (1995)
Published in Tetrahedron (1995)
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NEW METHODS FOR THE SYNTHESIS OF 2-ARYLPYRROLES
KRUSE, CG, BOUW, JP, VANHES, R, VANDEKUILEN, A, DENHARTOG, JAJ
Published in Heterocycles (01.12.1987)
Published in Heterocycles (01.12.1987)
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Conformational Analysis of the Nucleotides A2′‐5′A, A2′‐5′A2′‐5′A and A2′‐5′U from Nuclear Magnetic Resonance and Circular Dichroism Studies
DOORNBOS, Johannes, HARTOG, Jack A. J., BOOM, Jacques H. v., ALTONA, Cornelis
Published in European journal of biochemistry (01.05.1981)
Published in European journal of biochemistry (01.05.1981)
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Chemical synthesis of a messenger ribonucleic acid fragment: AUGUUCUUCUUCUUCUUC
den Hartog, J A, Wille, G, Scheublin, R A, van Boom, J H
Published in Biochemistry (Easton) (02.03.1982)
Published in Biochemistry (Easton) (02.03.1982)
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Piperazinophenyl- and piperazinophenyloxy-carboxylic acid derivatives as well as processes and intermediates for their preparation and medicaments containing these compounds
ANTEL, JOCHEN, KRUSE, C.G, BIELENBERG, GERHARD-WILHELM, ZIEGLER, DIETER, KEHRBACH, WOLFGANG, VAN MAARSEVEEN, J.H, REINDERS, JAN-HENDRIK, DEN HARTOG, JACK A.J, SCHOEN, UWE
Year of Publication 04.10.2001
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Year of Publication 04.10.2001
Patent
DERIVADOS DE ACIDOS PIPERAZINO-FENIL- Y PIPERAZINO-FENILOXI-CARBOXILICOS, ASI COMO PROCEDIMIENTOS Y PRODUCTOS INTERMEDIOS PARA SU PREPARACION Y MEDICAMENTOS QUE CONTIENEN ESTOS COMPUESTOS
ANTEL, JOCHEN, KRUSE, C.G, KEHRBACH, WOLFGANG, VAN MAARSEVEEN, J.H, DEN HARTOG, JACK A.J, SCHON, UWE
Year of Publication 01.12.2001
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Year of Publication 01.12.2001
Patent
Piperazinophenyl- und Piperazinophenyloxy-carbonsäure-Derivate sowie Verfahren und Zwischenprodukte zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
SCHOEN, UWE., 31303 BURGDORF, DE, HARTOG, JACK A.J. DEN., WEESP, NL, REINDERS, JAN-HENDRIK., HILVERSUM, NL, KEHRBACH, WOLFGANG., 30173 HANNOVER, DE, ANTEL, JOCHEN., 31848 BAD MUENDER, DE, BIELENBERG, GERHARD-WILHELM., 31061 ALFELD, DE, ZIEGLER, DIETER., 30966 HEMMINGEN, DE, MAARSEVEEN, JAN HERMAN VAN., AMERSFOORT, NL, KRUSE, CHRIS G.., AMERSFOORT, NL
Year of Publication 25.06.1998
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Year of Publication 25.06.1998
Patent
Piperazinophenyl- and piperazinophenyloxy-carboxylic acid derivatives as well as processes and intermediates for their preparation and medicaments containing these compounds
ANTEL, JOCHEN, KRUSE, C.G, BIELENBERG, GERHARD-WILHELM, ZIEGLER, DIETER, KEHRBACH, WOLFGANG, VAN MAARSEVEEN, J.H, REINDERS, JAN-HENDRIK, DEN HARTOG, JACK A.J, SCHOEN, UWE
Year of Publication 24.06.1998
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Year of Publication 24.06.1998
Patent