Small Molecule Ligands of the BET-like Bromodomain, SmBRD3, Affect Schistosoma mansoni Survival, Oviposition, and Development
Schiedel, Matthias, McArdle, Darius J. B., Padalino, Gilda, Chan, Anthony K. N., Forde-Thomas, Josephine, McDonough, Michael, Whiteland, Helen, Beckmann, Manfred, Cookson, Rosa, Hoffmann, Karl F., Conway, Stuart J.
Published in Journal of medicinal chemistry (14.12.2023)
Published in Journal of medicinal chemistry (14.12.2023)
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Journal Article
Anti-schistosomal activities of quinoxaline-containing compounds: From hit identification to lead optimisation
Padalino, Gilda, El-Sakkary, Nelly, Liu, Lawrence J., Liu, Chenxi, Harte, Danielle S.G., Barnes, Rachel E., Sayers, Edward, Forde-Thomas, Josephine, Whiteland, Helen, Bassetto, Marcella, Ferla, Salvatore, Johnson, George, Jones, Arwyn T., Caffrey, Conor R., Chalmers, Iain, Brancale, Andrea, Hoffmann, Karl F.
Published in European journal of medicinal chemistry (15.12.2021)
Published in European journal of medicinal chemistry (15.12.2021)
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Journal Article
Flukicidal effects of abietane diterpenoid derived analogues against the food borne pathogen Fasciola hepatica
Chakroborty, Anand, Pritchard, Deiniol, Bouillon, Marc E., Cervi, Anna, Cookson, Alan, Wild, Charlotte, Fenn, Caroline, Payne, Joseph, Holdsworth, Peter, Capner, Colin, O’Neill, Jenna, Padalino, Gilda, Forde-Thomas, Josephine, Gupta, Sandeep, Smith, Brendan G., Fisher, Maggie, Lahmann, Martina, Baird, Mark S., Hoffmann, Karl F.
Published in Veterinary parasitology (01.09.2022)
Published in Veterinary parasitology (01.09.2022)
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Journal Article
Using ChEMBL to Complement Schistosome Drug Discovery
Padalino, Gilda, Coghlan, Avril, Pagliuca, Giampaolo, Forde-Thomas, Josephine E, Berriman, Matthew, Hoffmann, Karl F
Published in Pharmaceutics (28.04.2023)
Published in Pharmaceutics (28.04.2023)
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Journal Article
The repositioning of epigenetic probes/inhibitors identifies new anti-schistosomal lead compounds and chemotherapeutic targets
Whatley, Kezia C L, Padalino, Gilda, Whiteland, Helen, Geyer, Kathrin K, Hulme, Benjamin J, Chalmers, Iain W, Forde-Thomas, Josephine, Ferla, Salvatore, Brancale, Andrea, Hoffmann, Karl F
Published in PLoS neglected tropical diseases (01.11.2019)
Published in PLoS neglected tropical diseases (01.11.2019)
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Journal Article
Schistosoma mansoni venom allergen-like protein 6 (SmVAL6) maintains tegumental barrier function
Perally, Samirah, Geyer, Kathrin K., Farani, Priscila S.G., Chalmers, Iain W., Fernandez-Fuentes, Narcis, Maskell, Daniel R., Hulme, Benjamin J., Forde-Thomas, Josephine, Phillips, Dylan, Farias, Leonardo P., Collins, James J., Hoffmann, Karl F.
Published in International journal for parasitology (01.03.2021)
Published in International journal for parasitology (01.03.2021)
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Journal Article
Quorum sensing N-Acyl homoserine lactones are a new class of anti-schistosomal
Whiteland, Helen, Crusco, Alessandra, Bloemberg, Lisa W, Tibble-Howlings, Jamie, Forde-Thomas, Josephine, Coghlan, Avril, Murphy, Patrick J, Hoffmann, Karl F
Published in PLoS neglected tropical diseases (01.10.2020)
Published in PLoS neglected tropical diseases (01.10.2020)
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Journal Article
Antischistosomal Properties of Sclareol and Its Heck-Coupled Derivatives: Design, Synthesis, Biological Evaluation, and Untargeted Metabolomics
Crusco, Alessandra, Whiteland, Helen, Baptista, Rafael, Forde-Thomas, Josephine E, Beckmann, Manfred, Mur, Luis A. J, Nash, Robert J, Westwell, Andrew D, Hoffmann, Karl F
Published in ACS infectious diseases (12.07.2019)
Published in ACS infectious diseases (12.07.2019)
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Journal Article
Modified Hederagenin Derivatives Demonstrate Ex Vivo Anthelmintic Activity against Fasciola hepatica
Chakroborty, Anand, Pritchard, Deiniol R, Bouillon, Marc E, Cervi, Anna, Kraehenbuehl, Rolf, Wild, Charlotte, Fenn, Caroline, Holdsworth, Peter, Capner, Colin, Padalino, Gilda, Forde-Thomas, Josephine E, Payne, Joseph, Smith, Brendan G, Fisher, Maggie, Lahmann, Martina, Baird, Mark S, Hoffmann, Karl F
Published in Pharmaceutics (03.07.2023)
Published in Pharmaceutics (03.07.2023)
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Journal Article
An Abies procera-derived tetracyclic triterpene containing a steroid-like nucleus core and a lactone side chain attenuates in vitro survival of both Fasciola hepatica and Schistosoma mansoni
Whiteland, Helen L., Chakroborty, Anand, Forde-Thomas, Josephine E., Crusco, Alessandra, Cookson, Alan, Hollinshead, Jackie, Fenn, Caroline A., Bartholomew, Barbara, Holdsworth, Peter A., Fisher, Maggie, Nash, Robert J., Hoffmann, Karl F.
Published in International journal for parasitology -- drugs and drug resistance (01.12.2018)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2018)
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Journal Article
Structural Requirements for Dihydrobenzoxazepinone Anthelmintics: Actions against Medically Important and Model Parasites: Trichuris muris, Brugia malayi, Heligmosomoides polygyrus, and Schistosoma mansoni
Partridge, Frederick A, Bataille, Carole J.R, Forman, Ruth, Marriott, Amy E, Forde-Thomas, Josephine, Häberli, Cécile, Dinsdale, Ria L, O’Sullivan, James D.B, Willis, Nicky J, Wynne, Graham M, Whiteland, Helen, Archer, John, Steven, Andrew, Keiser, Jennifer, Turner, Joseph D, Hoffmann, Karl F, Taylor, Mark J, Else, Kathryn J, Russell, Angela J, Sattelle, David B
Published in ACS infectious diseases (14.05.2021)
Published in ACS infectious diseases (14.05.2021)
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Journal Article
Chemical modulation of Schistosoma mansoni lysine specific demethylase 1 (SmLSD1) induces wide-scale biological and epigenomic changes
Padalino, Gilda, Celatka, Cassandra A, Rienhoff, Jr, Hugh Y, Kalin, Jay H, Cole, Philip A, Lassalle, Damien, Forde-Thomas, Josephine, Chalmers, Iain W, Brancale, Andrea, Grunau, Christoph, Hoffmann, Karl F
Published in Wellcome open research (2023)
Published in Wellcome open research (2023)
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Journal Article
Plasmacytoid Dendritic Cells Facilitate Th Cell Cytokine Responses throughout Schistosoma mansoni Infection
Webb, Lauren M, Phythian-Adams, Alexander T, Costain, Alice H, Brown, Sheila L, Lundie, Rachel J, Forde-Thomas, Josephine, Cook, Peter C, Jackson-Jones, Lucy H, Marley, Angela K, Smits, Hermelijn H, Hoffmann, Karl F, Tait Wojno, Elia D, MacDonald, Andrew S
Published in ImmunoHorizons (30.08.2021)
Published in ImmunoHorizons (30.08.2021)
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Journal Article
Aberrant spindle dynamics and cytokinesis in Dictyostelium discoideum cells that lack glycogen synthase kinase 3
Harwood, Adrian J., Forde-Thomas, Josephine E., Williams, Hazel, Samereier, Matthias, Müller-Taubenberger, Annette
Published in European journal of cell biology (01.06.2013)
Published in European journal of cell biology (01.06.2013)
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Journal Article
The repositioning of epigenetic probes/inhibitors identifies new anti-schistosomal lead compounds and chemotherapeutic targets
Whatley, Kezia, Padalino, Gilda, Whiteland, Helen, Geyer, Kathrin, Hulme, Benjamin, Chalmers, Iain, de-Thomas, Josephine, Ferla, Salvatore, Brancale, Andrea, Hoffmann, Karl F
Published in bioRxiv (08.08.2019)
Published in bioRxiv (08.08.2019)
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Paper
Structural requirements for dihydrobenzoxazepinone anthelmintics: actions against medically important and model parasites - Trichuris muris, Brugia malayi, Heligmosomoides polygyrus and Schistosoma mansoni
Partridge, Frederick A, Bataille, Carole Jr, man, Ruth, Marriott, Amy E, de-Thomas, Josephine, Häberli, Cécile, Dinsdale, Ria L, James Db O’sullivan, Willis, Nicky J, Wynne, Graham M, Whiteland, Helen, Archer, John, Andrew, Steven, Keiser, Jennifer, Turner, Joseph D, Hoffmann, Karl F, Taylor, Mark J, Else, Kathryn J, Russell, Angela J, Sattelle, David B
Published in bioRxiv (07.01.2021)
Published in bioRxiv (07.01.2021)
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