Validation of the zebrafish pentylenetetrazol seizure model: locomotor versus electrographic responses to antiepileptic drugs
Afrikanova, Tatiana, Serruys, Ann-Sophie K, Buenafe, Olivia E M, Clinckers, Ralph, Smolders, Ilse, de Witte, Peter A M, Crawford, Alexander D, Esguerra, Camila V
Published in PloS one (14.01.2013)
Published in PloS one (14.01.2013)
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Pharmacological characterization of an antisense knockdown zebrafish model of Dravet syndrome: inhibition of epileptic seizures by the serotonin agonist fenfluramine
Zhang, Yifan, Kecskés, Angéla, Copmans, Daniëlle, Langlois, Mélanie, Crawford, Alexander D, Ceulemans, Berten, Lagae, Lieven, de Witte, Peter A M, Esguerra, Camila V
Published in PloS one (12.05.2015)
Published in PloS one (12.05.2015)
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An Emerging Role for Sigma-1 Receptors in the Treatment of Developmental and Epileptic Encephalopathies
Martin, Parthena, Reeder, Thadd, Sourbron, Jo, de Witte, Peter A M, Gammaitoni, Arnold R, Galer, Bradley S
Published in International journal of molecular sciences (05.08.2021)
Published in International journal of molecular sciences (05.08.2021)
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Using Zebrafish as a Disease Model to Study Fibrotic Disease
Wang, Xixin, Copmans, Daniëlle, de Witte, Peter A. M.
Published in International journal of molecular sciences (15.06.2021)
Published in International journal of molecular sciences (15.06.2021)
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Comparative Antiseizure Analysis of Diverse Natural Coumarin Derivatives in Zebrafish
Kozioł, Ewelina, Jóźwiak, Krzysztof, Budzyńska, Barbara, de Witte, Peter A M, Copmans, Daniëlle, Skalicka-Woźniak, Krystyna
Published in International journal of molecular sciences (22.10.2021)
Published in International journal of molecular sciences (22.10.2021)
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Inhibition of glutamate decarboxylase (GAD) by ethyl ketopentenoate (EKP) induces treatment-resistant epileptic seizures in zebrafish
Zhang, Yifan, Vanmeert, Michiel, Siekierska, Aleksandra, Ny, Annelii, John, Jubi, Callewaert, Geert, Lescrinier, Eveline, Dehaen, Wim, de Witte, Peter A M, Kaminski, Rafal M
Published in Scientific reports (03.08.2017)
Published in Scientific reports (03.08.2017)
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Zebrafish bioassay-guided natural product discovery: isolation of angiogenesis inhibitors from East African medicinal plants
Crawford, Alexander D, Liekens, Sandra, Kamuhabwa, Appolinary R, Maes, Jan, Munck, Sebastian, Busson, Roger, Rozenski, Jef, Esguerra, Camila V, de Witte, Peter A M
Published in PloS one (17.02.2011)
Published in PloS one (17.02.2011)
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Identification of GSK‑3 as a Potential Therapeutic Entry Point for Epilepsy
Aourz, Najat, Serruys, Ann-Sophie K, Chabwine, Joëlle N, Balegamire, Pascal Byenda, Afrikanova, Tatiana, Edrada-Ebel, RuAngelie, Grey, Alexander I, Kamuhabwa, Appolinary R, Walrave, Laura, Esguerra, Camila V, van Leuven, Fred, de Witte, Peter A. M, Smolders, Ilse, Crawford, Alexander D
Published in ACS chemical neuroscience (17.04.2019)
Published in ACS chemical neuroscience (17.04.2019)
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Insights from zebrafish and mouse models on the activity and safety of ar-turmerone as a potential drug candidate for the treatment of epilepsy
Orellana-Paucar, Adriana Monserrath, Afrikanova, Tatiana, Thomas, Joice, Aibuldinov, Yelaman K, Dehaen, Wim, de Witte, Peter A M, Esguerra, Camila V
Published in PloS one (13.12.2013)
Published in PloS one (13.12.2013)
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Integration of Microfractionation, qNMR and zebrafish screening for the in vivo bioassay-guided isolation and quantitative bioactivity analysis of natural products
Bohni, Nadine, Cordero-Maldonado, María Lorena, Maes, Jan, Siverio-Mota, Dany, Marcourt, Laurence, Munck, Sebastian, Kamuhabwa, Appolinary R, Moshi, Mainen J, Esguerra, Camila V, de Witte, Peter A M, Crawford, Alexander D, Wolfender, Jean-Luc
Published in PloS one (21.05.2013)
Published in PloS one (21.05.2013)
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Zebrafish-Based Discovery of Antiseizure Compounds from the North Sea: Isoquinoline Alkaloids TMC-120A and TMC-120B
Copmans, Daniëlle, Kildgaard, Sara, Rasmussen, Silas A, Ślęzak, Monika, Dirkx, Nina, Partoens, Michèle, Esguerra, Camila V, Crawford, Alexander D, Larsen, Thomas O, de Witte, Peter A M
Published in Marine drugs (25.10.2019)
Published in Marine drugs (25.10.2019)
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Pharmacokinetics in Zebrafish Embryos (ZFE) Following Immersion and Intrayolk Administration: A Fluorescence-Based Analysis
Guarin, Marlly, Ny, Annelii, De Croze, Noémie, Maes, Jan, Léonard, Marc, Annaert, Pieter, de Witte, Peter
Published in Pharmaceuticals (Basel, Switzerland) (16.06.2021)
Published in Pharmaceuticals (Basel, Switzerland) (16.06.2021)
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Zebrafish Bioassay-Guided Microfractionation Identifies Anticonvulsant Steroid Glycosides from the Philippine Medicinal Plant Solanum torvum
Challal, Soura, Buenafe, Olivia E. M, Queiroz, Emerson F, Maljevic, Snezana, Marcourt, Laurence, Bock, Merle, Kloeti, Werner, Dayrit, Fabian M, Harvey, Alan L, Lerche, Holger, Esguerra, Camila V, de Witte, Peter A. M, Wolfender, Jean-Luc, Crawford, Alexander D
Published in ACS chemical neuroscience (15.10.2014)
Published in ACS chemical neuroscience (15.10.2014)
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From the North Sea to Drug Repurposing, the Antiseizure Activity of Halimide and Plinabulin
Copmans, Daniëlle, Kildgaard, Sara, Roux, Emma, Partoens, Michèle, Steurs, Gert, Wang, Xinhui, De Borggraeve, Wim M, Esguerra, Camila V, Crawford, Alexander D, Larsen, Thomas O, de Witte, Peter A M
Published in Pharmaceuticals (Basel, Switzerland) (18.02.2022)
Published in Pharmaceuticals (Basel, Switzerland) (18.02.2022)
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Optimization and pharmacological validation of a leukocyte migration assay in zebrafish larvae for the rapid in vivo bioactivity analysis of anti-inflammatory secondary metabolites
Cordero-Maldonado, María Lorena, Siverio-Mota, Dany, Vicet-Muro, Liliana, Wilches-Arizábala, Isabel María, Esguerra, Camila V, de Witte, Peter A M, Crawford, Alexander D
Published in PloS one (04.10.2013)
Published in PloS one (04.10.2013)
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Journal Article
Fishing for Drugs from Nature: Zebrafish as a Technology Platform for Natural Product Discovery
Crawford, Alexander D., Esguerra, Camila V., de Witte, Peter A.
Published in Planta medica (01.05.2008)
Published in Planta medica (01.05.2008)
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Stress-induced inflammation evoked by immunogenic cell death is blunted by the IRE1α kinase inhibitor KIRA6 through HSP60 targeting
Rufo, Nicole, Korovesis, Dimitris, Van Eygen, Sofie, Derua, Rita, Garg, Abhishek D, Finotello, Francesca, Vara-Perez, Monica, Rožanc, Jan, Dewaele, Michael, de Witte, Peter A, Alexopoulos, Leonidas G, Janssens, Sophie, Sinkkonen, Lasse, Sauter, Thomas, Verhelst, Steven H L, Agostinis, Patrizia
Published in Cell death and differentiation (01.01.2022)
Published in Cell death and differentiation (01.01.2022)
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Journal Article
Efficacy of Fenfluramine and Norfenfluramine Enantiomers and Various Antiepileptic Drugs in a Zebrafish Model of Dravet Syndrome
Li, Jing, Nelis, Maxim, Sourbron, Jo, Copmans, Daniëlle, Lagae, Lieven, Cabooter, Deirdre, de Witte, Peter A. M.
Published in Neurochemical research (01.09.2021)
Published in Neurochemical research (01.09.2021)
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Fishing Anti-Inflammatories from Known Drugs: In Silico Repurposing, Design, Synthesis and Biological Evaluation of Bisacodyl Analogues
Veitía, Maité Sylla-Iyarreta, Mota, Dany Siverio, Lerari, Vanessa, Marín, Marta, Giner, Rosa M, Muro, Liliana Vicet, Guerra, Yankier Rivero, Dumas, Françoise, Ferroud, Clotilde, de Witte, Peter A M, Crawford, Alexander D, Arán, Vicente J, Ponce, Yovani Marrero
Published in Current topics in medicinal chemistry (01.10.2017)
Published in Current topics in medicinal chemistry (01.10.2017)
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