Ligand Dependent Switch from RXR Homo- to RXR-NURR1 Heterodimerization
Scheepstra, Marcel, Andrei, Sebastian A, de Vries, Rens M. J. M, Meijer, Femke A, Ma, Jian-Nong, Burstein, Ethan S, Olsson, Roger, Ottmann, Christian, Milroy, Lech-Gustav, Brunsveld, Luc
Published in ACS chemical neuroscience (20.09.2017)
Published in ACS chemical neuroscience (20.09.2017)
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Characterization and small-molecule stabilization of the multisite tandem binding between 14-3-3 and the R domain of CFTR
Stevers, Loes M., Lam, Chan V., Leysen, Seppe F. R., Meijer, Femke A., van Scheppingen, Daphne S., de Vries, Rens M. J. M., Carlile, Graeme W., Milroy, Lech G., Thomas, David Y., Brunsveld, Luc, Ottmann, Christian
Published in Proceedings of the National Academy of Sciences - PNAS (01.03.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (01.03.2016)
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Journal Article
Elucidation of an Allosteric Mode of Action for a Thienopyrazole RORγt Inverse Agonist
Vries, Rens M. J. M., Doveston, Richard G., Meijer, Femke A., Brunsveld, Luc
Published in ChemMedChem (03.04.2020)
Published in ChemMedChem (03.04.2020)
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Journal Article
Allosteric small molecule modulators of nuclear receptors
Meijer, Femke A., Leijten-van de Gevel, Iris A., de Vries, Rens M.J.M., Brunsveld, Luc
Published in Molecular and cellular endocrinology (05.04.2019)
Published in Molecular and cellular endocrinology (05.04.2019)
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Journal Article
Structural interface between LRRK2 and 14-3-3 protein
Stevers, Loes M, de Vries, Rens M J M, Doveston, Richard G, Milroy, Lech-Gustav, Brunsveld, Luc, Ottmann, Christian
Published in Biochemical journal (01.04.2017)
Published in Biochemical journal (01.04.2017)
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Journal Article
Ligand-Based Design of Allosteric Retinoic Acid Receptor-Related Orphan Receptor γt (RORγt) Inverse Agonists
Meijer, Femke A, Doveston, Richard G, de Vries, Rens M.J.M, Vos, Gaël M, Vos, Alex A.A, Leysen, Seppe, Scheepstra, Marcel, Ottmann, Christian, Milroy, Lech-Gustav, Brunsveld, Luc
Published in Journal of medicinal chemistry (09.01.2020)
Published in Journal of medicinal chemistry (09.01.2020)
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Journal Article
Indazole MRL-871 interacts with PPARγ via a binding mode that induces partial agonism
Leijten-van de Gevel, Iris A., van Herk, Kim H.N., de Vries, Rens M.J.M., Ottenheym, Nicolaas J., Ottmann, Christian, Brunsveld, Luc
Published in Bioorganic & medicinal chemistry (15.08.2022)
Published in Bioorganic & medicinal chemistry (15.08.2022)
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Journal Article
Structure–Activity Relationship Studies of Trisubstituted Isoxazoles as Selective Allosteric Ligands for the Retinoic-Acid-Receptor-Related Orphan Receptor γt
Meijer, Femke A, Saris, Annet O.W.M, Doveston, Richard G, Oerlemans, Guido J.M, de Vries, Rens M.J.M, Somsen, Bente A, Unger, Anke, Klebl, Bert, Ottmann, Christian, Cossar, Peter J, Brunsveld, Luc
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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