Rational-Based Discovery of Novel β-Carboline Derivatives as Potential Antimalarials: From In Silico Identification of Novel Targets to Inhibition of Experimental Cerebral Malaria
Alves, Fernanda de Moura, Bellei, Jessica Correa Bezerra, Barbosa, Camila de Souza, Duarte, Caíque Lopes, Fonseca, Amanda Luisa da, Pinto, Ana Claudia de Souza, Raimundo, Felipe Oliveira, Carpinter, Bárbara Albuquerque, Lemos, Ari Sérgio de Oliveira, Coimbra, Elaine Soares, Taranto, Alex Gutterres, Rocha, Vinícius Novaes, de Pilla Varotti, Fernando, Ribeiro Viana, Gustavo Henrique, Scopel, Kézia K G
Published in Pathogens (Basel) (01.12.2022)
Published in Pathogens (Basel) (01.12.2022)
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Journal Article
Imidazo[1,2‑a]pyrimidine as a New Antileishmanial Pharmacophore against Leishmania amazonensis Promastigotes and Amastigotes
Kumar, Ravinder, Singh, Rahul, das Chagas Almeida, Ayla, da Trindade Granato, Juliana, de Oliveira Lemos, Ari Sérgio, Kumar, Kushvinder, Patil, Madhuri T., da Silva, Adilson D., Rode, Ambadas B., Coimbra, Elaine S., Salunke, Deepak B.
Published in ACS omega (31.10.2023)
Published in ACS omega (31.10.2023)
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Journal Article
Synthesis, biological evaluation and mechanism of action of benzothiazole derivatives with aromatic hydrazone moiety, a new class of antileishmanial compounds
Coimbra, Elaine Soares, Antinarelli, Luciana M. R., Oliveira Lemos, Ari Sérgio, Silva Neto, Adolfo Firmino, Pinheiro, Alessandra Campbell, Souza, Marcus Vinícius Nora
Published in Chemical biology & drug design (01.07.2024)
Published in Chemical biology & drug design (01.07.2024)
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Journal Article
Structural, physicochemical, and functional (antioxidant/anti-inflammatory) properties of β-cyclodextrin supramolecular complexation with Mitracarpus frigidus extract
Ferreira, Thayna Gomes, de Freitas Souza, Thalita, de Lima Paula, Priscila, de Oliveira Lemos, Ari Sérgio, Pinto, Nícolas de Castro Campos, Denadai, Ângelo Márcio Leite, Fabri, Rodrigo Luiz
Published in Journal of drug delivery science and technology (01.06.2023)
Published in Journal of drug delivery science and technology (01.06.2023)
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Journal Article
Development and in vivo evaluation of chitosan-gel containing Mitracarpus frigidus methanolic extract for vulvovaginal candidiasis treatment
Campos, Lara Melo, de Oliveira Lemos, Ari Sérgio, da Cruz, Luisa Ferreira, de Freitas Araújo, Marcelo Gonzaga, de Mello Botti, Giuly Cristina Rodrigues, Júnior, Janildo Ludolf Reis, Rocha, Vinícius Novaes, Denadai, Ângelo Márcio Leite, da Silva, Thiago Pereira, Tavares, Guilherme Diniz, Scio, Elita, Fabri, Rodrigo Luiz, Pinto, Priscila Faria
Published in Biomedicine & pharmacotherapy (01.10.2020)
Published in Biomedicine & pharmacotherapy (01.10.2020)
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Journal Article
Prospecção fitoquímica e avaliação das atividades antimicrobiana e antioxidante de espécies de Arecaceae
Fabri, Rodrigo Luiz, de Oliveira Lemos, Ari Sérgio, De Lima Paula, Priscila de Lima Paula, De Freitas Souza, Thalita, Gomes Ferreira, Thayná, Melo Campos, Lara, Torres Branca, Matheus
Published in H.U. revista (08.12.2022)
Published in H.U. revista (08.12.2022)
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Journal Article
Lantana camara L. induces a multi-targeted cell death process in Leishmania amazonensis
Lemos, Ari Sérgio de Oliveira, Granato, Juliana da Trindade, Antinarelli, Luciana Maria Ribeiro, Machado, Patrícia de Almeida, Campos, Lara Melo, Bastos, João Pedro Reis Costa, Midlej, Victor do Valle, Silva Neto, Adolfo Firmino da, Fabri, Rodrigo Luiz, Coimbra, Elaine Soares
Published in Journal of ethnopharmacology (30.01.2025)
Published in Journal of ethnopharmacology (30.01.2025)
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Journal Article
Antibiofilm potential of Annona muricata L. ethanolic extract against multi-drug resistant Candida albicans
Campos, Lara Melo, Silva, Thiago P., de Oliveira Lemos, Ari Sérgio, Mendonça Diniz, Irley Olívia, Palazzi, Cinthia, Novaes da Rocha, Vinícius, de Freitas Araújo, Marcelo Gonzaga, Melo, Rossana C.N., Fabri, Rodrigo Luiz
Published in Journal of ethnopharmacology (28.10.2023)
Published in Journal of ethnopharmacology (28.10.2023)
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Journal Article
Exploring the antifungal potential of Annona muricata leaf extract-loaded hydrogel in treating vulvovaginal candidiasis
Campos, Lara Melo, de Oliveira Lemos, Ari Sérgio, de Lima Paula, Priscila, da Rocha, Vinícius Novaes, de Freitas Araújo, Marcelo Gonzaga, Tavares, Guilherme Diniz, Barradas, Thais Nogueira, Nascimento, Wesley William Gonçalves, Denadai, Angelo Mácio Leite, de Oliveira, Luiz Fernando Cappa, Fabri, Rodrigo Luiz
Published in Colloids and surfaces, B, Biointerfaces (01.06.2024)
Published in Colloids and surfaces, B, Biointerfaces (01.06.2024)
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Journal Article
Pharmacological investigation of antioxidant and anti-inflammatory activities of leaves and branches extracts from Plinia cauliflora (Jaboticaba)
de Lima Paula, Priscila, de Oliveira Lemos, Ari Sérgio, Campos, Lara Melo, Ferreira, Thayná Gomes, Freitas de Souza, Thalita, Queiroz, Lucas Sales, Machado Resende Guedes, Maria Clara, Martins, Mário Machado, Goulart Filho, Luiz Ricardo, Macedo, Gilson Costa, Tavares, Guilherme Diniz, Rocha, Vinícius Novaes, Leite Denadai, Ângelo Márcio, Fabri, Rodrigo Luiz
Published in Journal of ethnopharmacology (15.11.2021)
Published in Journal of ethnopharmacology (15.11.2021)
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Journal Article
Assessment of lipid profile in fat body and eggs of Rhipicephalus microplus engorged females exposed to (E)-cinnamaldehyde and α-bisabolol, potential acaricide compounds
Marchesini, Paula, Lemos, Ari Sérgio de Oliveira, Bitencourt, Ricardo de Oliveira Barbosa, Fiorotti, Jéssica, Angelo, Isabele da Costa, Fabri, Rodrigo Luiz, Costa-Júnior, Lívio Martins, Lopes, Welber Daniel Zaneti, Bittencourt, Vânia Rita Elias Pinheiro, Monteiro, Caio
Published in Veterinary parasitology (01.12.2021)
Published in Veterinary parasitology (01.12.2021)
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Journal Article
4‐Quinolinylhydrazone analogues kill Leishmania (Leishmania) amazonensis by inducing apoptosis and mitochondria‐dependent pathway cell death
Granato, Juliana da Trindade, Silva, Emerson Teixeira da, Lemos, Ari Sérgio de Oliveira, Machado, Patrícia de Almeida, Midlej, Victor do Valle, Antinarelli, Luciana Maria Ribeiro, Silva Neto, Adolfo Firmino da, Souza, Marcus Vinícius Nora, Coimbra, Elaine Soares
Published in Chemical biology & drug design (01.05.2024)
Published in Chemical biology & drug design (01.05.2024)
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Journal Article
Development and characterization of chitosan film containing hydroethanolic extract of Coffea arabica leaves for wound dressing application
Silva, Allana Carvalho, Valle, Ana Beatriz Caribé dos Santos, Lemos, Ari Sérgio de Oliveira, Campos, Lara Melo, Fabri, Rodrigo Luiz, Costa, Fabiano Freire, da Silva, Jeferson Gomes, Vilela, Fernanda Maria Pinto, Tavares, Guilherme Diniz, Rodarte, Mirian Pereira, Denadai, Ângelo Márcio Leite
Published in Materials today communications (01.03.2024)
Published in Materials today communications (01.03.2024)
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Journal Article
Supramolecular complexes between Plinia cauliflora (DC.) Kausel extracts and β-cyclodextrin: Physicochemical characterization and antioxidant and anti-inflammatory properties
de Lima Paula, Priscila, Lemos, Ari Sérgio de Oliveira, Queiroz, Lucas Sales, Rocha, Vinícius Novaes, Coimbra, Elaine Soares, Fabri, Rodrigo Luiz, Denadai, Ângelo Márcio Leite
Published in Journal of drug delivery science and technology (01.06.2023)
Published in Journal of drug delivery science and technology (01.06.2023)
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Journal Article
Avaliação do perfil químico e citotóxico de Jatropha multifida L. (Euphorbiaceae) / Chemical and citotoxic perfil evaluation of Jatropha multifida L. (Euphorbiaceae)
Lemos, Ari Sérgio de Oliveira, De Oliveira, Naiara Norberto Tavares, Netto, Lívia Lacerda, Reis, Samara Evangelista, De Medeiros, Valquíria Pereira, Fabri, Rodrigo Luiz, Chedier, Luciana Moreira
Published in Brazilian Journal of Development (05.10.2021)
Published in Brazilian Journal of Development (05.10.2021)
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Journal Article
Potencial antimicrobiano, citotóxico e leishmanicida do extrato em diclorometano das partes aéreas de Mitracarpus frigidus (Rubiaceae)
Fabri, Rodrigo Luiz, Da Cunha, Paula Spagnol, Campos, Lara Melo, Lemos, Ari Sérgio de Oliveira, Coimbra, Elaine Soares, Scio, Elita
Published in Revista eletrônica de Farmácia (24.09.2020)
Published in Revista eletrônica de Farmácia (24.09.2020)
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Journal Article
Plantago major L. (Plantaginaceae) pode ser utilizado como agente antimicrobiano para emprego em produtos para uso oral?
Nogueira, Maria Luiza, Lima, Leandro Martins, Lemos, Ari Sérgio de Oliveira, Diogo, Marcel Arruda, De Freitas Souza, Thalita, Santana da Silva, João Paulo, Alves da Silva Filho, Ademar, Moreira Chedier, Luciana, Fabri, Rodrigo Luiz, De Faria Pinto, Priscila
Published in Revista Fitos (30.09.2021)
Published in Revista Fitos (30.09.2021)
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Journal Article
FORMULAÇÃO FITOTERÁPICA NANOESTRUTURADA À BASE DE MITRACARPUS FRIGIDUS COM CICLODEXTRINA, PROCESSO DE OBTENÇÃO, COMPOSIÇÕES E USOS
PRISCILA DE LIMA PAULA, JAIR ADRIANO KOPKE DE AGUIAR, LARA MELO CAMPOS, ARI SÉRGIO DE OLIVEIRA LEMOS, RODRIGO LUIZ FABRI, THALITA DE FREITAS SOUZA, GUILHERME DINIZ TAVARES, ÂNGELO MÁRCIO LEITE DENADAI, THAYNÁ GOMES FERREIRA
Year of Publication 28.03.2023
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Year of Publication 28.03.2023
Patent
Processo de obtenção de formulações fitoterápicas nanoestruturadas à base de plinia cauliflora (dc.) kausel (jabuticaba) com ciclodextrinas, composições e usos
PRISCILA DE LIMA PAULA, LARA MELO CAMPOS, MARIA CLARA MACHADO RESENDE GUEDES, ARI SÉRGIO DE OLIVEIRA LEMOS, RODRIGO LUIZ FABRI, GILSON COSTA MACEDO, LUCAS SALES QUEIROZ, ÂNGELO MÁRCIO LEITE DENADAI
Year of Publication 22.03.2022
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Year of Publication 22.03.2022
Patent
FORMULAÇÃO GELIFICADA PARA USO VAGINAL À BASE DE QUITOSANA COM MITRACARPUS FRIGIDUS, PROCESSO DE OBTENÇÃO, COMPOSIÇÕES E USOS
PRISCILA DE LIMA PAULA, LARA MELO CAMPOS, PRISCILA DE FARIA PINTO, ARI SÉRGIO DE OLIVEIRA LEMOS, RODRIGO LUIZ FABRI, VINÍCIUS NOVAES ROCHA, ANA CAROLINA MORAIS APOLÔNIO, GUILHERME DINIZ TAVARES, MARCELO GONZAGA DE FREITAS ARAÚJO, ÂNGELO MÁRCIO LEITE DENADAI
Year of Publication 29.11.2022
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Year of Publication 29.11.2022
Patent