Synthesis, Structure−Activity Relationships, and Biological Properties of 1-Heteroaryl-4-[ω-(1H-indol-3-yl)alkyl]piperazines, Novel Potential Antipsychotics Combining Potent Dopamine D2 Receptor Antagonism with Potent Serotonin Reuptake Inhibition
Smid, Pieter, Coolen, Hein K. A. C, Keizer, Hiskias G, van Hes, Rolf, de Moes, Jan-Peter, den Hartog, Arnold P, Stork, Bob, Plekkenpol, Rob H, Niemann, Leonarda C, Stroomer, Cees N. J, Tulp, Martin Th. M, van Stuivenberg, Herman H, McCreary, Andrew C, Hesselink, Mayke B, Herremans, Arnoud H. J, Kruse, Chris G
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
Get full text
Journal Article
Allosteric Inhibition of the Neuropeptidase Neurolysin
Hines, Christina S., Ray, Kallol, Schmidt, Jack J., Xiong, Fei, Feenstra, Rolf W., Pras-Raves, Mia, de Moes, Jan Peter, Lange, Jos H.M., Melikishvili, Manana, Fried, Michael G., Mortenson, Paul, Charlton, Michael, Patel, Yogendra, Courtney, Stephen M., Kruse, Chris G., Rodgers, David W.
Published in The Journal of biological chemistry (19.12.2014)
Published in The Journal of biological chemistry (19.12.2014)
Get full text
Journal Article
Synthesis, Structure−Activity Relationships, and Biological Properties of 1-Heteroaryl-4-[ω-(1 H -indol-3-yl)alkyl]piperazines, Novel Potential Antipsychotics Combining Potent Dopamine D 2 Receptor Antagonism with Potent Serotonin Reuptake Inhibition
Smid, Pieter, Coolen, Hein K. A. C., Keizer, Hiskias G., van Hes, Rolf, de Moes, Jan-Peter, den Hartog, Arnold P., Stork, Bob, Plekkenpol, Rob H., Niemann, Leonarda C., Stroomer, Cees N. J., Tulp, Martin Th. M., van Stuivenberg, Herman H., McCreary, Andrew C., Hesselink, Mayke B., Herremans, Arnoud H. J., Kruse, Chris G.
Published in Journal of medicinal chemistry (01.11.2005)
Published in Journal of medicinal chemistry (01.11.2005)
Get full text
Journal Article