Identification of Novel Isoform-Selective Inhibitors within Class I Histone Deacetylases
Hu, Erding, Dul, Edward, Sung, Chiu-Mei, Chen, Zunxuan, Kirkpatrick, Robert, Zhang, Gui-Feng, Johanson, Kyung, Liu, Ronggang, Lago, Amparo, Hofmann, Glenn, Macarron, Ricardo, de los Frailes, Maite, Perez, Paloma, Krawiec, John, Winkler, James, Jaye, Michael
Published in The Journal of pharmacology and experimental therapeutics (01.11.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2003)
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Journal Article
Discovery of Substituted Maleimides as Liver X Receptor Agonists and Determination of a Ligand-Bound Crystal Structure
Jaye, Michael C, Krawiec, John A, Campobasso, Nino, Smallwood, Angela, Qiu, Chunyan, Lu, Quinn, Kerrigan, John J, De Los Frailes Alvaro, Maite, Laffitte, Bryan, Liu, Wu-Schyong, Marino, Joseph P, Meyer, Craig R, Nichols, Jason A, Parks, Derek J, Perez, Paloma, Sarov-Blat, Lea, Seepersaud, Sheila D, Steplewski, Klaudia M, Thompson, Scott K, Wang, Ping, Watson, Mike A, Webb, Christine L, Haigh, David, Caravella, Justin A, Macphee, Colin H, Willson, Timothy M, Collins, Jon L
Published in Journal of medicinal chemistry (25.08.2005)
Published in Journal of medicinal chemistry (25.08.2005)
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Journal Article
Discovery of Novel Inhibitors of the Tautomerase Activity of Macrophage Migration Inhibitory Factor (MIF)
Zapatero, Maria Cleofé, Pérez, Paloma, Vázquez, María Jesús, Colmenarejo, Gonzalo, de Los Frailes, Maite, Ramón, Fernando
Published in Journal of biomolecular screening (01.06.2016)
Published in Journal of biomolecular screening (01.06.2016)
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Journal Article
Discovery of Enhancers of the Secretion of Leukemia Inhibitory Factor for the Treatment of Multiple Sclerosis
Vela, Laura, Caballero, Iván, Fang, Leiping, Liu, Qin, Ramón, Fernando, Díez, Emilio, de Los Frailes, Maite
Published in Journal of biomolecular screening (01.06.2016)
Published in Journal of biomolecular screening (01.06.2016)
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Journal Article
Screening technologies for G protein-coupled receptors: from HTS to uHTS
De los Frailes, Maite, Diez, Emilio
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2009)
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2009)
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Journal Article
Discovery of 3-Aryl-4-isoxazolecarboxamides as TGR5 Receptor Agonists
Evans, Karen A, Budzik, Brian W, Ross, Sean A, Wisnoski, David D, Jin, Jian, Rivero, Ralph A, Vimal, Mythily, Szewczyk, George R, Jayawickreme, Channa, Moncol, David L, Rimele, Thomas J, Armour, Susan L, Weaver, Susan P, Griffin, Robert J, Tadepalli, Sarva M, Jeune, Michael R, Shearer, Todd W, Chen, Zibin B, Chen, Lihong, Anderson, Donald L, Becherer, J. David, De Los Frailes, Maite, Colilla, Francisco Javier
Published in Journal of medicinal chemistry (24.12.2009)
Published in Journal of medicinal chemistry (24.12.2009)
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The identification of structurally novel, selective, orally bioavailable positive modulators of mGluR2
D’Alessandro, Pier L., Corti, Corrado, Roth, Adelheid, Ugolini, Annarosa, Sava, Anna, Montanari, Dino, Bianchi, Federica, Garland, Stephen L., Powney, Ben, Koppe, Emma L., Rocheville, Magalie, Osborne, Greg, Perez, Paloma, de la Fuente, Jesús, De Los Frailes, Maite, Smith, Paul W., Branch, Clive, Nash, David, Watson, Stephen P.
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
Potent achiral agonists of the ghrelin (growth hormone secretagogue) receptor. Part I: Lead identification
Heightman, Tom D., Scott, Jackie S., Longley, Mark, Bordas, Vincent, Dean, David K., Elliott, Richard, Hutley, Gail, Witherington, Jason, Abberley, Lee, Passingham, Barry, Berlanga, Manuela, de los Frailes, Maite, Wise, Alan, Powney, Ben, Muir, Alison, McKay, Fiona, Butler, Sharon, Winborn, Kim, Gardner, Christopher, Darton, Jill, Campbell, Colin, Sanger, Gareth
Published in Bioorganic & medicinal chemistry letters (01.12.2007)
Published in Bioorganic & medicinal chemistry letters (01.12.2007)
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Journal Article
Organic compounds produced by micro-organisms, particularly exophiala pisciphila, are used as inhibitors of interaction of CD28 and its specific receptors
ELSON STEVE W, SANCHEZ PUELLES JOSE MARIA, DIEZ MONEDERO EMILIO, DE LOS FRAILES ALVAREZ MAITE, HUESO RODRIGUEZ JUAN A, DE LA FUENTE CARRALERO JESUS
Year of Publication 01.08.2000
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Year of Publication 01.08.2000
Patent
COMPUESTOS ORGANICOS PRODUCIDOS POR MICROORGANISMOS, EN PARTICULAR EXOPHIALA PISCIPHILA, Y SU USO COMO INHIBIDORES DE LA INTERACCION DE CD28 Y SUS RECEPTORES ESPECIFICOS
ELSON STEVE W, SANCHEZ PUELLES JOSE MARIA, DIEZ MONEDERO EMILIO, DE LOS FRAILES ALVAREZ MAITE, HUESO RODRIGUEZ JUAN A, DE LA FUENTE CARRALERO JESUS
Year of Publication 01.02.2001
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Year of Publication 01.02.2001
Patent
DERIVADOS DE HIDROCARBUROS AROMATICOS CARBOCICLICOS PRODUCIDOS POR HAPALOSPHAERIA DEFORMANS, INHIBIDORES DE LA INTERACCION DE CD28 Y SUS RE CEPTORES ESPECIFICOS
ELSON STEVE W, SANCHEZ PUELLES JOSE MARIA, DIEZ MONEDERO EMILIO, DE LOS FRAILES ALVAREZ MAITE, HUESO RODRIGUEZ JUAN A, DE LA FUENTE CARRALERO JESUS
Year of Publication 01.02.2001
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Year of Publication 01.02.2001
Patent