Search Results - "de Koning, Pieter D." :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Fit-for-Purpose Development of the Enabling Route to Crizotinib (PF-02341066)

Fit-for-Purpose Development of the Enabling Route to Crizotinib (PF-02341066)

by de Koning, Pieter D, McAndrew, Douglas, Moore, Robert, Moses, Ian B, Boyles, David C, Kissick, Kyle, Stanchina, Corey L, Cuthbertson, Timothy, Kamatani, Asayuki, Rahman, Leera, Rodriguez, Rick, Urbina, Armando, Sandoval (née Accacia), Alison, Rose, Peter R
Published in Organic process research & development (16.09.2011)

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An Enantioselective Synthesis of (S)-(+)-3-Aminomethyl-5-methylhexanoic Acid via Asymmetric Hydrogenation

An Enantioselective Synthesis of (S)-(+)-3-Aminomethyl-5-methylhexanoic Acid via Asymmetric Hydrogenation

by Burk, Mark J, de Koning, Pieter D, Grote, Todd M, Hoekstra, Marvin S, Hoge, Garrett, Jennings, Rex A, Kissel, William S, Le, Tung V, Lennon, Ian C, Mulhern, Thomas A, Ramsden, James A, Wade, Robert A
Published in Journal of organic chemistry (11.07.2003)

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Development of an Asymmetric Hydrogenation Route to (S)-N-Boc-2,6-dimethyltyrosine

Development of an Asymmetric Hydrogenation Route to (S)-N-Boc-2,6-dimethyltyrosine

by Praquin, Céline F. B, de Koning, Pieter D, Peach, Philip J, Howard, Roger M, Spencer, Sarah L
Published in Organic process research & development (16.09.2011)

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Work-Up Optimization en Route to an Improved Process To Prepare a Progesterone Receptor Antagonist

Work-Up Optimization en Route to an Improved Process To Prepare a Progesterone Receptor Antagonist

by de Koning, Pieter D, McManus, David J, Bandurek, George R
Published in Organic process research & development (16.09.2011)

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Development an Efficient Route to the 5-Lipoxygenase Inhibitor PF-04191834

Development an Efficient Route to the 5-Lipoxygenase Inhibitor PF-04191834

by de Koning, Pieter D, Murtagh, Lorraine, Lawson, Jon P, Vonder Embse, Richard A, Kunda, Sastry A, Kong, Wei
Published in Organic process research & development (16.09.2011)

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Use of Achiral (Diphosphine)RuCl2(Diamine) Precatalysts as a Practical Alternative to Sodium Borohydride for Ketone Reduction

Use of Achiral (Diphosphine)RuCl2(Diamine) Precatalysts as a Practical Alternative to Sodium Borohydride for Ketone Reduction

by de Koning, Pieter D, Jackson, Mark, Lennon, Ian C
Published in Organic process research & development (15.09.2006)

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A perspective on synthetic and solid-form enablement of inhalation candidates

A perspective on synthetic and solid-form enablement of inhalation candidates

by Selby, Matthew D, de Koning, Pieter D, Roberts, Dannielle F
Published in Future medicinal chemistry (01.10.2011)

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Enzymatic Desymmetrization Route to Ethyl [3-(2-Amino-2-methylpropyl)phenyl]acetate

Enzymatic Desymmetrization Route to Ethyl [3-(2-Amino-2-methylpropyl)phenyl]acetate

by de Koning, Pieter D, Gladwell, Iain R, Morrison, Natalie A, Moses, Ian B, Panesar, Maninder S, Pettman, Alan J, Thomson, Nicholas M, Yazbeck, Daniel R
Published in Organic process research & development (15.07.2011)

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Practical Synthesis of (1s,4s)-4-(Methylamino)-1′H-spiro[cyclohexane-1,3′-furo[3,4-c]pyridin]-1′-one

Practical Synthesis of (1s,4s)-4-(Methylamino)-1′H-spiro[cyclohexane-1,3′-furo[3,4-c]pyridin]-1′-one

by Bish, Gerwyn, de Koning, Pieter D, Dubant, Stephané P. A, Fengas, David, Fray, M. Jonathan
Published in Organic process research & development (17.09.2010)

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Development of a Practical Synthesis of the Progesterone Receptor Antagonist 4-{[3-Cyclopropyl-1-(mesylmethyl)-5-methyl-1H-pyrazol-4-yl]oxy}-2,6-dimethylbenzonitrile

Development of a Practical Synthesis of the Progesterone Receptor Antagonist 4-{[3-Cyclopropyl-1-(mesylmethyl)-5-methyl-1H-pyrazol-4-yl]oxy}-2,6-dimethylbenzonitrile

by Bradley, Paul A, de Koning, Pieter D, Johnson, Patrick S, Lecouturier, Yann C, McManus, David J, Robin, Aurelie, Underwood, Toby J
Published in Organic process research & development (18.09.2009)

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Bidirectional Asymmetric Allylboration. A Convenient Asymmetric Synthesis of C 2-Symmetric 3-Methylenepentane-1,5-diols and Rapid Access to C 2-Symmetric Spiroketals

Bidirectional Asymmetric Allylboration. A Convenient Asymmetric Synthesis of C 2-Symmetric 3-Methylenepentane-1,5-diols and Rapid Access to C 2-Symmetric Spiroketals

by Barrett, Anthony G. M, Braddock, D. Christopher, de Koning, Pieter D, White, Andrew J. P, Williams, David J
Published in Journal of organic chemistry (28.01.2000)

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Efficient Synthesis of an Imidazole-Substituted δ-Amino Acid by the Integration of Chiral Technologies

Efficient Synthesis of an Imidazole-Substituted δ-Amino Acid by the Integration of Chiral Technologies

by Appleby, Ian, Boulton, Lee T, Cobley, Christopher J, Hill, Catherine, Hughes, Mike L, de Koning, Pieter D, Lennon, Ian C, Praquin, Céline, Ramsden, James A, Samuel, Helen J, Willis, Niamh
Published in Organic letters (12.05.2005)

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Synthetic Routes to 11-Oxygenated 14α,17α-Ethanoestradiols

Synthetic Routes to 11-Oxygenated 14α,17α-Ethanoestradiols

by Bull, James R., de Koning, Pieter D.
Published in European journal of organic chemistry (01.03.2001)

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ChemInform Abstract: Synthetic and Solid-Form Enablement of Inhalation Candidates

ChemInform Abstract: Synthetic and Solid-Form Enablement of Inhalation Candidates

by Selby, Matthew D., de Koning, Pieter D., Roberts, Dannielle F.
Published in ChemInform (15.05.2012)

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Development of an Enabling Route to PF-00610355: A Novel Inhaled β2-Adrenoreceptor Agonist

Development of an Enabling Route to PF-00610355: A Novel Inhaled β2-Adrenoreceptor Agonist

by de Koning, Pieter D., Gladwell, Iain R., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)

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Development of an Enabling Route to PF-00610355: A Novel Inhaled beta(2)-Adrenoreceptor Agonist

Development of an Enabling Route to PF-00610355: A Novel Inhaled beta(2)-Adrenoreceptor Agonist

by de Koning, Pieter D., Gladwell, Iain R., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (01.11.2011)

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Hydration and related reactions of 14,17-ethenoestradiol methyl ethers: a comparative study in selectivity

Hydration and related reactions of 14,17-ethenoestradiol methyl ethers: a comparative study in selectivity

by Bull, James R., De Koning, Pieter D., Hoadley, Clarissa & Reddie, Kim
Published in South African journal of chemistry (01.12.1998)

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Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled beta(2)-Adrenoreceptor Agonist

Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled beta(2)-Adrenoreceptor Agonist

by de Koning, Pieter D., Castro, Nieves, Gladwell, Iain R., Morrison, Natalie A., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (01.11.2011)

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Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled β2-Adrenoreceptor Agonist

Development of a Potential Manufacturing Route to PF-00610355: A Novel Inhaled β2-Adrenoreceptor Agonist

by de Koning, Pieter D., Castro, Nieves, Gladwell, Iain R., Morrison, Natalie A., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)

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Development of an Enabling Route to PF-00610355: A Novel Inhaled β 2 -Adrenoreceptor Agonist

Development of an Enabling Route to PF-00610355: A Novel Inhaled β 2 -Adrenoreceptor Agonist

by de Koning, Pieter D., Gladwell, Iain R., Moses, Ian B., Panesar, Maninder S., Pettman, Alan J., Thomson, Nicholas M.
Published in Organic process research & development (18.11.2011)

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