Structure-Based Design and Synthesis of Covalent Inhibitors for Deubiquitinase and Acetyltransferase ChlaDUB1 of Chlamydia trachomatis
Zimmermann, Thomas, Feng, Jiachen, de Campos, Luana Janaína, Knight, Lindsey A., Schlötzer, Jan, Ramirez, Yesid A., Schwickert, Kevin, Zehe, Markus, Adler, Thomas B., Schirmeister, Tanja, Kisker, Caroline, Sotriffer, Christoph, Conda-Sheridan, Martin, Decker, Michael
Published in Journal of medicinal chemistry (11.07.2024)
Published in Journal of medicinal chemistry (11.07.2024)
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Design, Biological Evaluation, and Computer-Aided Analysis of Dihydrothiazepines as Selective Antichlamydial Agents
de Campos, Luana Janaína, Seleem, Mohamed A., Feng, Jiachen, Pires de Oliveira, Kelly Mari, de Andrade dos Santos, João Víctor, Hayer, Shivdeep, Clayton, Jonathan B., Kathi, Sharvath, Fisher, Derek J., Ouellette, Scot P., Conda-Sheridan, Martin
Published in Journal of medicinal chemistry (09.02.2023)
Published in Journal of medicinal chemistry (09.02.2023)
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Pharmacophore modeling, molecular docking, and molecular dynamics studies to identify new 5-HT2AR antagonists with the potential for design of new atypical antipsychotics
Martins, Allana Faustino, de Campos, Luana Janaína, Conda-Sheridan, Martin, de Melo, Eduardo Borges
Published in Molecular diversity (01.10.2023)
Published in Molecular diversity (01.10.2023)
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Design, synthesis and in vivo evaluation of 1,4-dioxo-2-butenyl aryl amine derivatives as a promising anti-inflammatory drug prototype
da Silveira, Ingridhy O.M.F., Moslaves, Iluska S.B., Muller, Jéssica A.I., Hortelan, Cristiane R.W., Juliano Oliveira, Rodrigo, Okuyama, Tatiane T., Fernandes, Juliana, Badenoch, Bretton, Janaína de Campos, Luana, Almeida, Leandro D., Mohammad, Jiyan, Martins, Allana C.F., Beatriz, Adilson, da Silva Júnior, Eufrânio N., Cristina Toffoli-Kadri, Mônica, da Silva Gomes, Roberto
Published in Bioorganic chemistry (01.07.2022)
Published in Bioorganic chemistry (01.07.2022)
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Engineering a nanoantibiotic system displaying dual mechanism of action
Xing, Huihua, de Campos, Luana Janaína, Pereira, Aramis Jose, Fiora, Maria Mercedes, Aguiar-Alves, Fabio, Tagliazucchi, Mario, Conda-Sheridan, Martin
Published in Proceedings of the National Academy of Sciences - PNAS (16.04.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (16.04.2024)
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Orphan GPRC5B activation modulates airway contractility
Varadharajan, Subashini, Balraj, Premanand, Kale, Narendra, Campos, Luana Janaina de, Conda Sheridan, Martin, Mallik, Sanku, Pabelick, Christina M, YS, Prakash, Sathish, Venkatachalem
Published in Physiology (Bethesda, Md.) (01.05.2023)
Published in Physiology (Bethesda, Md.) (01.05.2023)
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