Revisiting Pyrazolo[3,4‑d]pyrimidine Nucleosides as Anti-Trypanosoma cruzi and Antileishmanial Agents
Bouton, Jakob, Ferreira de Almeida Fiuza, Ludmila, Cardoso Santos, Camila, Mazzarella, Maria Angela, Soeiro, Maria de Nazaré Correia, Maes, Louis, Karalic, Izet, Caljon, Guy, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (08.04.2021)
Published in Journal of medicinal chemistry (08.04.2021)
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Activity of pyridyl-pyrazolone derivatives against Trypanosoma cruzi
Batista, Denise da Gama Jaen, de Almeida Fiuza, Ludmila Ferreira, Klupsch, Frédérique, da Costa, Krislayne Nunes, Batista, Marcos Meuser, da Conceição, Ketlym, Bouafia, Hassiba, Vergoten, Gérard, Millet, Régis, Thuru, Xavier, Bailly, Christian, Soeiro, Maria de Nazaré Correia
Published in Experimental parasitology (01.07.2024)
Published in Experimental parasitology (01.07.2024)
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Journal Article
Efficacy of Novel Pyrazolone Phosphodiesterase Inhibitors in Experimental Mouse Models of Trypanosoma cruzi
de Araújo, Julianna Siciliano, França da Silva, Cristiane, Batista, Denise da Gama Jaén, Nefertiti, Aline, Fiuza, Ludmila Ferreira de Almeida, Fonseca-Berzal, Cristina Rosa, Bernardino da Silva, Patrícia, Batista, Marcos Meuser, Sijm, Maarten, Kalejaiye, Titilola D, de Koning, Harry P, Maes, Louis, Sterk, Geert Jan, Leurs, Rob, Soeiro, Maria de Nazaré Correia
Published in Antimicrobial agents and chemotherapy (20.08.2020)
Published in Antimicrobial agents and chemotherapy (20.08.2020)
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Journal Article
6‐Methyl‐7‐Aryl‐7‐Deazapurine Nucleosides as Anti‐Trypanosoma cruzi Agents: Structure‐Activity Relationship and in vivo Efficacy
Lin, Cai, Ferreira de Almeida Fiuza, Ludmila, Cardoso Santos, Camila, Ferreira Nunes, Daniela, Cruz Moreira, Otacílio, Bouton, Jakob, Karalic, Izet, Maes, Louis, Caljon, Guy, Hulpia, Fabian, Nazaré C. Soeiro, Maria, Van Calenbergh, Serge
Published in ChemMedChem (20.07.2021)
Published in ChemMedChem (20.07.2021)
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Benign-by-Design SAHA Analogues for Human and Animal Vector-Borne Parasitic Diseases
Rossi, Michele, Martinengo, Bianca, Diamanti, Eleonora, Salerno, Alessandra, Rizzardi, Nicola, Fato, Romana, Bergamini, Christian, Souza de Oliveira, Andressa, de Araújo Marques Ferreira, Thais, Andrade Holanda, Cleonice, Romeiro, Luiz Antonio Soares, Soeiro, Maria de Nazaré Correia, Nunes, Krislayne, Ferreira de Almeida Fiuza, Ludmila, Meuser Batista, Marcos, Fraga, Carlos A M, E A Alkhalaf, Hamed, Elmahallawy, Ehab Kotb, Ebiloma, Godwin U, De Koning, Harry P, Vittorio, Serena, Vistoli, Giulio, Blanquart, Christophe, Bertrand, Philippe, Bolognesi, Maria Laura
Published in ACS medicinal chemistry letters (12.09.2024)
Published in ACS medicinal chemistry letters (12.09.2024)
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Journal Article
Identification of Pyrazolo[3,4-e][1,4]thiazepin based CYP51 inhibitors as potential Chagas disease therapeutic alternative: In vitro and in vivo evaluation, binding mode prediction and SAR exploration
Ferreira de Almeida Fiuza, Ludmila, Peres, Raiza Brandão, Simões-Silva, Marianne Rocha, da Silva, Patricia Bernardino, Batista, Denise da Gama Jaen, da Silva, Cristiane França, Nefertiti Silva da Gama, Aline, Krishna Reddy, Tummala Rama, Soeiro, Maria de Nazaré Correia
Published in European journal of medicinal chemistry (10.04.2018)
Published in European journal of medicinal chemistry (10.04.2018)
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Journal Article
Combination With Tomatidine Improves the Potency of Posaconazole Against Trypanosoma cruzi
Rocha-Hasler, Marianne, de Oliveira, Gabriel Melo, da Gama, Aline Nefertiti, Fiuza, Ludmila Ferreira de Almeida, Fesser, Anna Frieda, Cal, Monica, Rocchetti, Romina, Peres, Raiza Brandão, Guan, Xue Li, Kaiser, Marcel, Soeiro, Maria de Nazaré Correia, Mäser, Pascal
Published in Frontiers in cellular and infection microbiology (04.03.2021)
Published in Frontiers in cellular and infection microbiology (04.03.2021)
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7-Aryl-7-deazapurine 3′-deoxyribonucleoside derivative as a novel lead for Chagas’ disease therapy: in vitro and in vivo pharmacology
Cardoso-Santos, Camila, Ferreira de Almeida Fiuza, Ludmila, França da Silva, Cristiane, Mazzeti, Ana Lia, Donola Girão, Roberson, Melo de Oliveira, Gabriel, da Gama Jaen Batista, Denise, Cruz Moreira, Otacilio, Lins da Silva Gomes, Natália, Maes, Louis, Caljon, Guy, Hulpia, Fabian, Calenbergh, Serge V, Correia Soeiro, Maria de Nazaré
Published in JAC-antimicrobial resistance (01.12.2021)
Published in JAC-antimicrobial resistance (01.12.2021)
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In silico and in vitro assessment of anti-Trypanosoma cruzi efficacy, genotoxicity and pharmacokinetics of pentasubstituted pyrrolic Atorvastatin-aminoquinoline hybrid compounds
Araujo-Lima, Carlos Fernando, Carvalho, Rita de Cássia Castro, Peres, Raiza Brandão, Fiuza, Ludmila Ferreira de Almeida, Galvão, Bárbara Verena Dias, Castelo-Branco, Frederico S., Bastos, Mônica Macedo, Boechat, Nubia, Felzenszwalb, Israel, Soeiro, Maria de Nazaré Correia
Published in Acta tropica (01.06.2023)
Published in Acta tropica (01.06.2023)
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Journal Article
Benznidazole modulates release of inflammatory mediators by cardiac spheroids infected with Trypanosoma cruzi
de Almeida Fiuza, Ludmila Ferreira, Batista, Denise da Gama Jaen, Nunes, Daniela Ferreira, Moreira, Otacílio Cruz, Cascabulho, Cynthia, Soeiro, Maria de Nazaré Correia
Published in Experimental parasitology (01.02.2021)
Published in Experimental parasitology (01.02.2021)
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Journal Article
Identification and preliminary structure-activity relationship studies of novel pyridyl sulfonamides as potential Chagas disease therapeutic agents
Peres, Raiza Brandão, Ullah, Asma Inam, de Almeida Fiuza, Ludmila Ferreira, Silva, Patricia Bernardino, Batista, Marcos M., Corcoran, Olivia, Reddy, Tummala Rama Krishna, de Nazaré Correia Soeiro, Maria
Published in Bioorganic & medicinal chemistry letters (15.06.2018)
Published in Bioorganic & medicinal chemistry letters (15.06.2018)
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