Quinolin-6-Yloxyacetamides Are Microtubule Destabilizing Agents That Bind to the Colchicine Site of Tubulin
Sharma, Ashwani, Sáez-Calvo, Gonzalo, Olieric, Natacha, de Asís Balaguer, Francisco, Barasoain, Isabel, Lamberth, Clemens, Díaz, J Fernando, Steinmetz, Michel O
Published in International journal of molecular sciences (22.06.2017)
Published in International journal of molecular sciences (22.06.2017)
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Journal Article
Synthesis of Thicolchicine‐Based Conjugates: Investigation towards Bivalent Tubulin/Microtubules Binders
Bonandi, Elisa, Foschi, Francesca, Marucci, Cristina, Dapiaggi, Federico, Sironi, Maurizio, Pieraccini, Stefano, Christodoulou, Michael S., de Asís Balaguer, Francisco, Díaz, J. Fernando, Zidar, Nace, Passarella, Daniele
Published in ChemPlusChem (Weinheim, Germany) (01.01.2019)
Published in ChemPlusChem (Weinheim, Germany) (01.01.2019)
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Journal Article
Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands
Balaguer, Francisco de Asís, Mühlethaler, Tobias, Estévez-Gallego, Juan, Calvo, Enrique, Giménez-Abián, Juan Francisco, Risinger, April L, Sorensen, Erik J, Vanderwal, Christopher D, Altmann, Karl-Heinz, Mooberry, Susan L, Steinmetz, Michel O, Oliva, María Ángela, Prota, Andrea E, Díaz, J Fernando
Published in International journal of molecular sciences (20.03.2019)
Published in International journal of molecular sciences (20.03.2019)
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Journal Article
Structure-activity relationships, biological evaluation and structural studies of novel pyrrolonaphthoxazepines as antitumor agents
Brindisi, Margherita, Ulivieri, Cristina, Alfano, Gloria, Gemma, Sandra, de Asís Balaguer, Francisco, Khan, Tuhina, Grillo, Alessandro, Chemi, Giulia, Menchon, Grégory, Prota, Andrea E., Olieric, Natacha, Lucena-Agell, Daniel, Barasoain, Isabel, Diaz, J. Fernando, Nebbioso, Angela, Conte, Mariarosaria, Lopresti, Ludovica, Magnano, Stefania, Amet, Rebecca, Kinsella, Paula, Zisterer, Daniela M., Ibrahim, Ola, O'Sullivan, Jeff, Morbidelli, Lucia, Spaccapelo, Roberta, Baldari, Cosima, Butini, Stefania, Novellino, Ettore, Campiani, Giuseppe, Altucci, Lucia, Steinmetz, Michel O., Brogi, Simone
Published in European journal of medicinal chemistry (15.01.2019)
Published in European journal of medicinal chemistry (15.01.2019)
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Journal Article
CTP promotes efficient ParB-dependent DNA condensation by facilitating one-dimensional diffusion from parS
Balaguer, Francisco de Asis, Aicart-Ramos, Clara, Fisher, Gemma LM, de Bragança, Sara, Martin-Cuevas, Eva M, Pastrana, Cesar L, Dillingham, Mark Simon, Moreno-Herrero, Fernando
Published in eLife (12.07.2021)
Published in eLife (12.07.2021)
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Journal Article
Structure, Thermodynamics, and Kinetics of Plinabulin Binding to Two Tubulin Isotypes
La Sala, Giuseppina, Olieric, Natacha, Sharma, Ashwani, Viti, Federica, de Asis Balaguer Perez, Francisco, Huang, Lan, Tonra, James R., Lloyd, G. Kenneth, Decherchi, Sergio, Díaz, José Fernando, Steinmetz, Michel O., Cavalli, Andrea
Published in Chem (14.11.2019)
Published in Chem (14.11.2019)
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Journal Article
Triazolopyrimidines Are Microtubule-Stabilizing Agents that Bind the Vinca Inhibitor Site of Tubulin
Sáez-Calvo, Gonzalo, Sharma, Ashwani, Balaguer, Francisco de Asís, Barasoain, Isabel, Rodríguez-Salarichs, Javier, Olieric, Natacha, Muñoz-Hernández, Hugo, Berbís, Manuel Álvaro, Wendeborn, Sebastian, Peñalva, Miguel Angel, Matesanz, Ruth, Canales, Ángeles, Prota, Andrea Enrico, Jímenez-Barbero, Jesús, Andreu, José Manuel, Lamberth, Clemens, Steinmetz, Michel Olivier, Díaz, José Fernando
Published in Cell chemical biology (22.06.2017)
Published in Cell chemical biology (22.06.2017)
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Journal Article
Development of a Novel Class of Microtubule Destabilizing Agents with Selectivity Against Diffuse Large B-Cell Lymphoma (DLBCL) with B-Cell Receptor (BCR) Activation
Pera Gresely, Benet, Balaguer, Francisco de Asís, Cardenas, Mariano Gonzalo, Revuelta, Maria Victoria, Calvo Vidal, Maria Nieves, Marullo, Rossella, Zamponi, Nahuel, Rivera, Ildefonso Ismael Rodriguez, Ai, Yong, Glickman, Joseph Fraser, Barasoain, Isabel, Díaz, Fernando, Melnick, Ari, Xue, Fengtian, Cerchietti, Leandro
Published in Blood (08.12.2017)
Published in Blood (08.12.2017)
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Journal Article
CTP promotes efficient ParB-dependent DNA condensation by facilitating one-dimensional diffusion from par S
Balaguer, Francisco de Asis, Aicart-Ramos, Clara, Fisher, Gemma Lm, de Bragança, Sara, Martin-Cuevas, Eva M, Pastrana, Cesar L, Dillingham, Mark Simon, Moreno-Herrero, Fernando
Published in eLife (12.07.2021)
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Published in eLife (12.07.2021)
Journal Article
Cytidine triphosphate promotes efficient ParB-dependent DNA condensation by facilitating one-dimensional spreading from parS
Francisco De Asis Balaguer, Aicart-Ramos, Clara, Fisher, Gemma Lm, De Bragança, Sara, Pastrana, Cesar L, Dillingham, Mark S, Moreno-Herrero, Fernando
Published in bioRxiv (11.02.2021)
Published in bioRxiv (11.02.2021)
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