Structural Optimization and Biological Activity of Pyrazole Derivatives: Virtual Computational Analysis, Recovery Assay and 3D Culture Model as Potential Predictive Tools of Effectiveness against Trypanosoma cruzi
Orlando, Lorraine Martins Rocha, Lechuga, Guilherme Curty, da Silva Lara, Leonardo, Ferreira, Byanca Silva, Pereira, Cynthia Nathalia, Silva, Rafaela Corrêa, Dos Santos, Maurício Silva, Pereira, Mirian Claudia S
Published in Molecules (Basel, Switzerland) (08.11.2021)
Published in Molecules (Basel, Switzerland) (08.11.2021)
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Synthesis by Microwave Irradiation, Molecular Structural Analysis and Trypanocidal Activity of Novel Pyrazole-tetrahydropyrimidine Derivatives
Pereira, Cynthia Nathalia, de Oliveira, Júlia Akihoshi, da Silva Lara, Leonardo, Rocha Orlando, Lorraine Martins, de Souza Pereira, Mirian Claudia, Dos Santos, Maurício Silva
Published in Current organic synthesis (01.01.2023)
Published in Current organic synthesis (01.01.2023)
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Synthesis and Anti-Trypanosoma cruzi Activity of New Pyrazole-Thiadiazole Scaffolds
Souza, Thamyris Perez de, Orlando, Lorraine Martins Rocha, Lara, Leonardo da Silva, Paes, Vitoria Barbosa, Dutra, Lucas Penha, dos Santos, Mauricio Silva, Pereira, Mirian Claudia de Souza
Published in Molecules (Basel, Switzerland) (01.08.2024)
Published in Molecules (Basel, Switzerland) (01.08.2024)
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Trypanosoma cruzi infection of human induced pluripotent stem cell-derived cardiomyocytes: an in vitro model for drug screening for Chagas disease
da Silva Lara, Leonardo, Andrade-Lima, Leonardo, Magalhães Calvet, Claudia, Borsoi, Juliana, Lopes Alberto Duque, Thabata, Henriques-Pons, Andrea, Souza Pereira, Mirian Claudia, Veiga Pereira, Lygia
Published in Microbes and infection (01.05.2018)
Published in Microbes and infection (01.05.2018)
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N‑Nitrosulfonamides as Carbonic Anhydrase Inhibitors: A Promising Chemotype for Targeting Chagas Disease and Leishmaniasis
Bonardi, Alessandro, Vermelho, Alane Beatriz, da Silva Cardoso, Veronica, de Souza Pereira, Mirian Claudia, da Silva Lara, Leonardo, Selleri, Silvia, Gratteri, Paola, Supuran, Claudiu T, Nocentini, Alessio
Published in ACS medicinal chemistry letters (11.04.2019)
Published in ACS medicinal chemistry letters (11.04.2019)
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Antitrypanosomal Activity of 1,2,3-Triazole-Based Hybrids Evaluated Using In Vitro Preclinical Translational Models
Orlando, Lorraine Martins Rocha, Lara, Leonardo da Silva, Lechuga, Guilherme Curty, Rodrigues, Giseli Capaci, Pandoli, Omar Ginoble, de Sá, Druval Santos, Pereira, Mirian Claudia de Souza
Published in Biology (Basel, Switzerland) (01.09.2023)
Published in Biology (Basel, Switzerland) (01.09.2023)
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Bioactivity of Novel Pyrazole-Thiazolines Scaffolds against Trypanosoma cruzi : Computational Approaches and 3D Spheroid Model on Drug Discovery for Chagas Disease
Lara, Leonardo da Silva, Lechuga, Guilherme Curty, Orlando, Lorraine Martins Rocha, Ferreira, Byanca Silva, Souto, Bernardo Araújo, Dos Santos, Maurício Silva, Pereira, Mirian Claudia de Souza
Published in Pharmaceutics (05.05.2022)
Published in Pharmaceutics (05.05.2022)
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Synthesis by microwave irradiation of new pyrazole-imidazoline-pyrimidine analogs: Physicochemical and photophysical properties and their biological activity against Trypanosoma cruzi
Pereira, Cynthia Nathalia, Rosa, José Otávio, Lara, Leonardo da Silva, Orlando, Lorraine Martins Rocha, Figueiredo, Nathália da Silva, Pereira, Mirian Claudia de Souza, Junior, Roberto Shigueru Nobuyasu, Santos, Maurício Silva dos
Published in Journal of molecular structure (15.10.2023)
Published in Journal of molecular structure (15.10.2023)
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