Site-selective protein-modification chemistry for basic biology and drug development
Krall, Nikolaus, da Cruz, Filipa P., Boutureira, Omar, Bernardes, Gonçalo J. L.
Published in Nature chemistry (01.02.2016)
Published in Nature chemistry (01.02.2016)
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Novel Potent Metallocenes against Liver Stage Malaria
MATOS, Joana, DA CRUZ, Filipa P, CABRITA, Elia, GUT, Jiri, NOGUEIRA, Fátima, DO ROSARIO, Virgílio E, MOREIRA, Rui, ROSENTHAL, Philip J, PRUDENCIO, Miguel, GOMES, Paula
Published in Antimicrobial Agents and Chemotherapy (01.03.2012)
Published in Antimicrobial Agents and Chemotherapy (01.03.2012)
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4-C-Me-DAB and 4-C-Me-LAB—enantiomeric alkyl-branched pyrrolidine iminosugars—are specific and potent α-glucosidase inhibitors; acetone as the sole protecting group
Cruz, Filipa P. da, Newberry, Scott, Jenkinson, Sarah F., Wormald, Mark R., Butters, Terry D., Alonzi, Dominic S., Nakagawa, Shinpei, Becq, Frederic, Norez, Caroline, Nash, Robert J., Kato, Atsushi, Fleet, George W.J.
Published in Tetrahedron letters (12.01.2011)
Published in Tetrahedron letters (12.01.2011)
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Controlled masking and targeted release of redox-cycling ortho-quinones via a C–C bond-cleaving 1,6-elimination
Dunsmore, Lavinia, Navo, Claudio D., Becher, Julie, de Montes, Enrique Gil, Guerreiro, Ana, Hoyt, Emily, Brown, Libby, Zelenay, Viviane, Mikutis, Sigitas, Cooper, Jonathan, Barbieri, Isaia, Lawrinowitz, Stefanie, Siouve, Elise, Martin, Esther, Ruivo, Pedro R., Rodrigues, Tiago, da Cruz, Filipa P., Werz, Oliver, Vassiliou, George, Ravn, Peter, Jiménez-Osés, Gonzalo, Bernardes, Gonçalo J. L.
Published in Nature chemistry (01.07.2022)
Published in Nature chemistry (01.07.2022)
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Drug Screen Targeted at Plasmodium Liver Stages Identifies a Potent Multistage Antimalarial Drug
da Cruz, Filipa P., Martin, Cécilie, Buchholz, Kathrin, Lafuente-Monasterio, Maria J., Rodrigues, Tiago, Sönnichsen, Birte, Moreira, Rui, Gamo, Francisco-Javier, Marti, Matthias, Mota, Maria M., Hannus, Michael, Prudêncio, Miguel
Published in The Journal of infectious diseases (15.04.2012)
Published in The Journal of infectious diseases (15.04.2012)
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Dual-stage triterpenoids from an African medicinal plant targeting the malaria parasite
Ramalhete, Cátia, da Cruz, Filipa P., Mulhovo, Silva, Sousa, Inês J., Fernandes, Miguel X., Prudêncio, Miguel, Ferreira, Maria-José U.
Published in Bioorganic & medicinal chemistry (01.08.2014)
Published in Bioorganic & medicinal chemistry (01.08.2014)
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Quinolin-4(1H)‑imines are Potent Antiplasmodial Drugs Targeting the Liver Stage of Malaria
Rodrigues, Tiago, da Cruz, Filipa P, Lafuente-Monasterio, Maria J, Gonçalves, Daniel, Ressurreição, Ana S, Sitoe, Ana R, Bronze, Maria R, Gut, Jiri, Schneider, Gisbert, Mota, Maria M, Rosenthal, Philip J, Prudêncio, Miguel, Gamo, Francisco-Javier, Lopes, Francisca, Moreira, Rui
Published in Journal of medicinal chemistry (13.06.2013)
Published in Journal of medicinal chemistry (13.06.2013)
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Triterpenoids as inhibitors of erythrocytic and liver stages of Plasmodium infections
Ramalhete, Cátia, da Cruz, Filipa P., Lopes, Dinora, Mulhovo, Silva, Rosário, Virgílio E., Prudêncio, Miguel, Ferreira, Maria-José U.
Published in Bioorganic & medicinal chemistry (15.12.2011)
Published in Bioorganic & medicinal chemistry (15.12.2011)
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Flavones as isosteres of 4(1H)-quinolones: Discovery of ligand efficient and dual stage antimalarial lead compounds
Rodrigues, Tiago, Ressurreição, Ana S., da Cruz, Filipa P., Albuquerque, Inês S., Gut, Jiri, Carrasco, Marta P., Gonçalves, Daniel, Guedes, Rita C., dos Santos, Daniel J.V.A., Mota, Maria M., Rosenthal, Philip J., Moreira, Rui, Prudêncio, Miguel, Lopes, Francisca
Published in European journal of medicinal chemistry (01.11.2013)
Published in European journal of medicinal chemistry (01.11.2013)
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Towards the biotechnological isomerization of branched sugars: d-tagatose-3-epimerase equilibrates both enantiomers of 4- C-methyl-ribulose with both enantiomers of 4- C-methyl-xylulose
Rao, Devendar, Yoshihara, Akihide, Gullapalli, Pushpakiran, Morimoto, Kenji, Takata, Goro, da Cruz, Filipa P., Jenkinson, Sarah F., Wormald, Mark R., Dwek, Raymond A., Fleet, George W.J., Izumori, Ken
Published in Tetrahedron letters (12.05.2008)
Published in Tetrahedron letters (12.05.2008)
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Carbon-branched carbohydrate chirons: practical access to both enantiomers of 2- C-methyl-ribono-1,4-lactone and 2- C-methyl-arabinonolactone
Booth, Kathrine V., da Cruz, Filipa P., Hotchkiss, David J., Jenkinson, Sarah F., Jones, Nigel A., Weymouth-Wilson, Alexander C., Clarkson, Robert, Heinz, Thomas, Fleet, George W.J.
Published in Tetrahedron: asymmetry (20.10.2008)
Published in Tetrahedron: asymmetry (20.10.2008)
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