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Metabolism and Excretion of [14C]Mobocertinib, a Selective Covalent Inhibitor of Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion Mutations, in Healthy Male Subjects
Chen, Hao, Shah, Abhi, Kato, Suguru, Griffin, Robert, Zhang, Steven, Pusalkar, Sandeepraj, Cohen, Lawrence, Li, Yuexian, Chowdhury, Swapan K., Zhu, Sean Xiaochun
Published in Drug metabolism and disposition (01.10.2024)
Published in Drug metabolism and disposition (01.10.2024)
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A Scalable General Synthetic Approach toward Ultrathin Imine-Linked Two-Dimensional Covalent Organic Framework Nanosheets for Photocatalytic CO2 Reduction
Liu, Wenbo, Li, Xiaokang, Wang, Chiming, Pan, Houhe, Liu, Wenping, Wang, Kang, Zeng, Qingdao, Wang, Rongming, Jiang, Jianzhuang
Published in Journal of the American Chemical Society (30.10.2019)
Published in Journal of the American Chemical Society (30.10.2019)
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Metabolism and Excretion of 14CMobocertinib, a Selective Covalent Inhibitor of Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion Mutations, in Healthy Male Subjects
Chen, Hao, Shah, Abhi, Kato, Suguru, Griffin, Robert, Zhang, Steven, Pusalkar, Sandeepraj, Cohen, Lawrence, Li, Yuexian, Chowdhury, Swapan K, Zhu, Sean Xiaochun
Published in Drug metabolism and disposition (16.09.2024)
Published in Drug metabolism and disposition (16.09.2024)
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Safety, pharmacokinetics, and pharmacodynamics of sofnobrutinib, a novel non‐covalent BTK inhibitor, in healthy subjects: First‐in‐human phase I study
Miyamoto, Kyoko, Miller, Robert M., Voors‐Pette, Christine, Oosterhaven, Jart A. F., Dobbelsteen, Marieke, Mihara, Katsuhiro, Geldof, Marian, Sato, Yuji, Matsuda, Naomi, Kirita, Shirou, Sawa, Masaaki, Arimura, Akinori
Published in Clinical and translational science (01.11.2024)
Published in Clinical and translational science (01.11.2024)
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A Dual−Functional Cationic Covalent Organic Frameworks Modified Separator for High Energy Lithium Metal Batteries
Yao, Shiyan, Yang, Yan, Liang, Ziwei, Chen, Jiahe, Ding, Jieying, Li, Fangkun, Liu, Junhao, Xi, Lei, Zhu, Min, Liu, Jun
Published in Advanced functional materials (01.03.2023)
Published in Advanced functional materials (01.03.2023)
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Internal catalysis for dynamic covalent chemistry applications and polymer science
Van Lijsebetten, Filip, Holloway, Joshua O, Winne, Johan M, Du Prez, Filip E
Published in Chemical Society reviews (07.12.2020)
Published in Chemical Society reviews (07.12.2020)
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Chemoproteomic discovery of a covalent allosteric inhibitor of WRN helicase
Baltgalvis, Kristen A., Lamb, Kelsey N., Symons, Kent T., Wu, Chu-Chiao, Hoffman, Melissa A., Snead, Aaron N., Song, Xiaodan, Glaza, Thomas, Kikuchi, Shota, Green, Jason C., Rogness, Donald C., Lam, Betty, Rodriguez-Aguirre, Maria E., Woody, David R., Eissler, Christie L., Rodiles, Socorro, Negron, Seth M., Bernard, Steffen M., Tran, Eileen, Pollock, Jonathan, Tabatabaei, Ali, Contreras, Victor, Williams, Heather N., Pastuszka, Martha K., Sigler, John J., Pettazzoni, Piergiorgio, Rudolph, Markus G., Classen, Moritz, Brugger, Doris, Claiborne, Christopher, Plancher, Jean-Marc, Cuartas, Isabel, Seoane, Joan, Burgess, Laurence E., Abraham, Robert T., Weinstein, David S., Simon, Gabriel M., Patricelli, Matthew P., Kinsella, Todd M.
Published in Nature (London) (09.05.2024)
Published in Nature (London) (09.05.2024)
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Transformation Strategy for Highly Crystalline Covalent Triazine Frameworks: From Staggered AB to Eclipsed AA Stacking
Yang, Zhenzhen, Chen, Hao, Wang, Song, Guo, Wei, Wang, Tao, Suo, Xian, Jiang, De-en, Zhu, Xiang, Popovs, Ilja, Dai, Sheng
Published in Journal of the American Chemical Society (15.04.2020)
Published in Journal of the American Chemical Society (15.04.2020)
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A non-covalent “click chemistry” strategy to efficiently coat highly porous MOF nanoparticles with a stable polymeric shell
Aykaç, Ahmet, Noiray, Magali, Malanga, Milo, Agostoni, Valentina, Casas-Solvas, Juan Manuel, Fenyvesi, Éva, Gref, Ruxandra, Vargas-Berenguel, Antonio
Published in Biochimica et biophysica acta. General subjects (01.06.2017)
Published in Biochimica et biophysica acta. General subjects (01.06.2017)
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PB2200: FOOD AND ACID REDUCING AGENT EFFECTS ON PHARMACOKINETICS (PK) AND PHARMACODYNAMICS (PD) OF THE COVALENT BRUTON TYROSINE KINASE INHIBITOR (BTKI) TL‐895 IN HEALTHY SUBJECTS
Allard, Martine, Krejsa, Cecile, Williams, Isaiah, Podoll, Terry, Steinmann, Kim, Slatter, Greg
Published in HemaSphere (08.08.2023)
Published in HemaSphere (08.08.2023)
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Mutualistic Synthesis from Orthogonal Dynamic Covalent Reactions
Lyu, Yonglei, Hu, Ying, Yang, Jinghui, Wang, Xin, Li, Jianwei
Published in Angewandte Chemie International Edition (24.10.2024)
Published in Angewandte Chemie International Edition (24.10.2024)
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Phenothiazine-based covalent organic frameworks with low exciton binding energies for photocatalysis
Wang, Weitao, Wang, Haotian, Tang, Xiaohui, Huo, Jinlei, Su, Yan, Lu, Chuangye, Zhang, Yujian, Xu, Hong, Gu, Cheng
Published in Chemical science (Cambridge) (29.07.2022)
Published in Chemical science (Cambridge) (29.07.2022)
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A road map for prioritizing warheads for cysteine targeting covalent inhibitors
Ábrányi-Balogh, Péter, Petri, László, Imre, Tímea, Szijj, Péter, Scarpino, Andrea, Hrast, Martina, Mitrović, Ana, Fonovič, Urša Pečar, Németh, Krisztina, Barreteau, Hélène, Roper, David I., Horváti, Kata, Ferenczy, György G., Kos, Janko, Ilaš, Janez, Gobec, Stanislav, Keserű, György M.
Published in European journal of medicinal chemistry (05.12.2018)
Published in European journal of medicinal chemistry (05.12.2018)
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Covalent inhibition of histone deacetylase 8 by 3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazin-6-imine
Muth, Marius, Jänsch, Niklas, Kopranovic, Aleksandra, Krämer, Andreas, Wössner, Nathalie, Jung, Manfred, Kirschhöfer, Frank, Brenner-Weiß, Gerald, Meyer-Almes, Franz-Josef
Published in Biochimica et biophysica acta. General subjects (01.03.2019)
Published in Biochimica et biophysica acta. General subjects (01.03.2019)
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