Design, Synthesis, and Activity of 2-Imidazol-1-ylpyrimidine Derived Inducible Nitric Oxide Synthase Dimerization Inhibitors
Davey, David D, Adler, Marc, Arnaiz, Damian, Eagen, Keith, Erickson, Shawn, Guilford, William, Kenrick, Margaret, Morrissey, Michael M, Ohlmeyer, Mike, Pan, Gonghua, Paradkar, Vidyadhar M, Parkinson, John, Polokoff, Mark, Saionz, Kurt, Santos, Cecile, Subramanyam, Babu, Vergona, Ron, Wei, Robert G, Whitlow, Marc, Ye, Bin, Zhao, Zuchun (Spring), Devlin, James J, Phillips, Gary
Published in Journal of medicinal chemistry (22.03.2007)
Published in Journal of medicinal chemistry (22.03.2007)
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Identification and Characterization of a Potent, Selective, and Orally Active Antagonist of the CC Chemokine Receptor-1
Liang, Meina, Mallari, Cornell, Rosser, Mary, Ng, Howard P., May, Karen, Monahan, Sean, Bauman, John G., Islam, Imadul, Ghannam, Ameen, Buckman, Brad, Shaw, Ken, Wei, Guo-Ping, Xu, Wei, Zhao, Zuchun, Ho, Elena, Shen, Jun, Oanh, Huynh, Subramanyam, Babu, Vergona, Ron, Taub, Dennis, Dunning, Laura, Harvey, Susan, Snider, R.Michael, Hesselgesser, Joseph, Morrissey, Michael M., Perez, H.Daniel, Horuk, Richard
Published in The Journal of biological chemistry (23.06.2000)
Published in The Journal of biological chemistry (23.06.2000)
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Thiophene-Anthranilamides as Highly Potent and Orally Available Factor Xa Inhibitors
Ye, Bin, Arnaiz, Damian O, Chou, Yuo-Ling, Griedel, Brian D, Karanjawala, Rushad, Lee, Wheeseong, Morrissey, Michael M, Sacchi, Karna L, Sakata, Steven T, Shaw, Kenneth J, Wu, Shung C, Zhao, Zuchun, Adler, Marc, Cheeseman, Sarah, Dole, William P, Ewing, Janice, Fitch, Richard, Lentz, Dao, Liang, Amy, Light, David, Morser, John, Post, Joseph, Rumennik, Galina, Subramanyam, Babu, Sullivan, Mark E, Vergona, Ron, Walters, Janette, Wang, Yi-Xin, White, Kathy A, Whitlow, Marc, Kochanny, Monica J
Published in Journal of medicinal chemistry (28.06.2007)
Published in Journal of medicinal chemistry (28.06.2007)
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Substituted thiophene-anthranilamides as potent inhibitors of human factor Xa
Kochanny, Monica J., Adler, Marc, Ewing, Janice, Griedel, Brian D., Ho, Elena, Karanjawala, Rushad, Lee, Wheeseong, Lentz, Dao, Liang, Amy M., Morrissey, Michael M., Phillips, Gary B., Post, Joseph, Sacchi, Karna L., Sakata, Steven T., Subramanyam, Babu, Vergona, Ron, Walters, Janette, White, Kathy A., Whitlow, Marc, Ye, Bin, Zhao, Zuchun, Shaw, Kenneth J.
Published in Bioorganic & medicinal chemistry (01.03.2007)
Published in Bioorganic & medicinal chemistry (01.03.2007)
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Synthesis and biological evaluation of piperazine-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)
Ye, Bin, Chou, Yuo-Ling, Karanjawala, Rushad, Lee, Wheeseong, Lu, Shou-Fu, Shaw, Kenneth J., Jones, Steven, Lentz, Dao, Liang, Amy, Tseng, Jih-Lie, Wu, Qingyu, Zhao, Zuchun
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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Synthesis and biological evaluation of menthol-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)
Ye, Bin, Bauer, Shawn, Buckman, Brad O., Ghannam, Ameen, Griedel, Brian D., Khim, Seock-Kyu, Lee, Wheeseong, Sacchi, Karna L., Shaw, Kenneth J., Liang, Amy, Wu, Qingyu, Zhao, Zuchun
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Crystallographic analysis of potent and selective factor Xa inhibitors complexed to bovine trypsin
Whitlow, Marc, Arnaiz, Damain O., Buckman, Brad O., Davey, David D., Griedel, Brain, Guilford, William J., Koovakkat, Sunil K., Liang, Amy, Mohan, Raju, Phillips, Gary B., Seto, Marian, Shaw, Kenneth J., Xu, Wei, Zhao, Zuchun, Light, David R., Morrissey, Michael M.
Published in Acta crystallographica. Section D, Biological crystallography. (01.08.1999)
Published in Acta crystallographica. Section D, Biological crystallography. (01.08.1999)
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Benzimidazole-Based fXa inhibitors with improved thrombin and trypsin selectivity
Shaw, Kenneth J., Guilford, William J., Griedel, Brian D., Sakata, Steve, Trinh, Lan, Wu, Shung, Xu, Wei, Zhao, Zuchun, Morrissey, Michael M.
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
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Design and synthesis of aminophenol-Based factor xa inhibitors
Wu, Shung, Guilford, William J, Chou, Yuo-Ling, Griedel, Brian D, Liang, Amy, Sakata, Steve, Shaw, Kenneth J, Trinh, Lan, Xu, Wei, Zhao, Zuchun, Morrissey, Michael M
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
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Inhibition of PAI-1: a new anti-thrombotic approach
Wu, Qingyu, Zhao, Zuchun
Published in Current drug targets. Cardiovascular & hematological disorders (01.06.2002)
Published in Current drug targets. Cardiovascular & hematological disorders (01.06.2002)
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Design, synthesis, and in vitro biological activity of benzimidazole based factor Xa inhibitors
Zhao, Z, Arnaiz, D O, Griedel, B, Sakata, S, Dallas, J L, Whitlow, M, Trinh, L, Post, J, Liang, A, Morrissey, M M, Shaw, K J
Published in Bioorganic & medicinal chemistry letters (01.05.2000)
Published in Bioorganic & medicinal chemistry letters (01.05.2000)
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