Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: application of a bioisosteric scaffold hopping approach to flufenamic acid
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Published in European journal of medicinal chemistry (25.04.2018)
Published in European journal of medicinal chemistry (25.04.2018)
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Effects of the Molecular Weight of Hyaluronic Acid in a Carbon Nanotube Drug Delivery Conjugate
Arpicco, Silvia, Bartkowski, Michał, Barge, Alessandro, Zonari, Daniele, Serpe, Loredana, Milla, Paola, Dosio, Franco, Stella, Barbara, Giordani, Silvia
Published in Frontiers in chemistry (14.12.2020)
Published in Frontiers in chemistry (14.12.2020)
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Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3
Lolli, Marco L, Carnovale, Irene M, Pippione, Agnese C, Wahlgren, Weixiao Y, Bonanni, Davide, Marini, Elisabetta, Zonari, Daniele, Gallicchio, Margherita, Boscaro, Valentina, Goyal, Parveen, Friemann, Rosmarie, Rolando, Barbara, Bagnati, Renzo, Adinolfi, Salvatore, Oliaro-Bosso, Simonetta, Boschi, Donatella
Published in ACS medicinal chemistry letters (11.04.2019)
Published in ACS medicinal chemistry letters (11.04.2019)
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Mesoporous silica as topical nanocarriers for quercetin: characterization and in vitro studies
Sapino, Simona, Ugazio, Elena, Gastaldi, Lucia, Miletto, Ivana, Berlier, Gloria, Zonari, Daniele, Oliaro-Bosso, Simonetta
Published in European journal of pharmaceutics and biopharmaceutics (01.01.2015)
Published in European journal of pharmaceutics and biopharmaceutics (01.01.2015)
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Thermoresponsive mesoporous silica nanoparticles as a carrier for skin delivery of quercetin
Ugazio, Elena, Gastaldi, Lucia, Brunella, Valentina, Scalarone, Dominique, Jadhav, Sushilkumar A., Oliaro-Bosso, Simonetta, Zonari, Daniele, Berlier, Gloria, Miletto, Ivana, Sapino, Simona
Published in International journal of pharmaceutics (10.09.2016)
Published in International journal of pharmaceutics (10.09.2016)
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Hyaluronated mesoporous silica nanoparticles for active targeting: influence of conjugation method and hyaluronic acid molecular weight on the nanovector properties
Ricci, Valentina, Zonari, Daniele, Cannito, Stefania, Marengo, Alessandro, Scupoli, Maria Teresa, Malatesta, Manuela, Carton, Flavia, Boschi, Federico, Berlier, Gloria, Arpicco, Silvia
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Published in Journal of colloid and interface science (15.04.2018)
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New aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the hydroxytriazole scaffold
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Published in European journal of medicinal chemistry (05.07.2022)
Published in European journal of medicinal chemistry (05.07.2022)
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Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
Pippione, Agnese C., Giraudo, Alessandro, Bonanni, Davide, Carnovale, Irene M., Marini, Elisabetta, Cena, Clara, Costale, Annalisa, Zonari, Daniele, Pors, Klaus, Sadiq, Maria, Boschi, Donatella, Oliaro-Bosso, Simonetta, Lolli, Marco L.
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
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Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer
Pippione, Agnese Chiara, Kovachka, Sandra, Vigato, Chiara, Bertarini, Laura, Mannella, Iole, Sainas, Stefano, Rolando, Barbara, Denasio, Enrica, Piercy-Mycock, Helen, Romalho, Linda, Salladini, Edoardo, Adinolfi, Salvatore, Zonari, Daniele, Peraldo-Neia, Caterina, Chiorino, Giovanna, Passoni, Alice, Mirza, Osman Asghar, Frydenvang, Karla, Pors, Klaus, Lolli, Marco Lucio, Spyrakis, Francesca, Oliaro-Bosso, Simonetta, Boschi, Donatella
Published in European journal of medicinal chemistry (15.03.2024)
Published in European journal of medicinal chemistry (15.03.2024)
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SWCNT-porphyrin nano-hybrids selectively activated by ultrasound: an interesting model for sonodynamic applications
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Published in RSC advances (08.06.2020)
Published in RSC advances (08.06.2020)
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AI Based Discovery of a New AKR1C3 Inhibitor for Anticancer Applications
Pippione, Agnese C., Vigato, Chiara, Tucciarello, Cristina, Hussain, Samrina, Salladini, Edoardo, Truong, Ha H., Henriksen, Niel M., Vanzetti, Gaia, Giordano, Giorgia, Zonari, Daniele, Mirza, Osman Asghar, Frydenvang, Karla, Pignochino, Ymera, Oliaro-Bosso, Simonetta, Boschi, Donatella, Lolli, Marco L.
Published in ACS medicinal chemistry letters (08.08.2024)
Published in ACS medicinal chemistry letters (08.08.2024)
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Ruthenium polypyridyl squalene derivative: A novel self-assembling lipophilic probe for cellular imaging
Dosio, Franco, Stella, Barbara, Ferrero, Annalisa, Garino, Claudio, Zonari, Daniele, Arpicco, Silvia, Cattel, Luigi, Giordano, Susanna, Gobetto, Roberto
Published in International journal of pharmaceutics (20.01.2013)
Published in International journal of pharmaceutics (20.01.2013)
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