Reversible and regionally selective downregulation of brain cannabinoid CB1 receptors in chronic daily cannabis smokers
HIRVONEN, J, GOODWIN, R. S, LI, C.-T, TERRY, G. E, ZOGHBI, S. S, MORSE, C, PIKE, V. W, VOLKOW, N. D, HUESTIS, M. A, INNIS, R. B
Published in Molecular psychiatry (01.06.2012)
Published in Molecular psychiatry (01.06.2012)
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cAMP signaling in brain is decreased in unmedicated depressed patients and increased by treatment with a selective serotonin reuptake inhibitor
Fujita, M, Richards, E M, Niciu, M J, Ionescu, D F, Zoghbi, S S, Hong, J, Telu, S, Hines, C S, Pike, V W, Zarate, C A, Innis, R B
Published in Molecular psychiatry (01.05.2017)
Published in Molecular psychiatry (01.05.2017)
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[11C]deschloroclozapine is an improved PET radioligand for quantifying a human muscarinic DREADD expressed in monkey brain
Yan, Xuefeng, Telu, Sanjay, Dick, Rachel M, Liow, Jeih-San, Zanotti-Fregonara, Paolo, Morse, Cheryl L, Manly, Lester S, Gladding, Robert L, Shrestha, Stal, Lerchner, Walter, Nagai, Yuji, Minamimoto, Takafumi, Zoghbi, Sami S, Innis, Robert B, Pike, Victor W, Richmond, Barry J, Eldridge, Mark AG
Published in Journal of cerebral blood flow and metabolism (01.10.2021)
Published in Journal of cerebral blood flow and metabolism (01.10.2021)
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A Genetic Polymorphism for Translocator Protein 18 Kda Affects both in Vitro and in Vivo Radioligand Binding in Human Brain to this Putative Biomarker of Neuroinflammation
Kreisl, William C, Jenko, Kimberly J, Hines, Christina S, Lyoo, Chul Hyoung, Corona, Winston, Morse, Cheryl L, Zoghbi, Sami S, Hyde, Thomas, Kleinman, Joel E, Pike, Victor W, McMahon, Francis J, Innis, Robert B
Published in Journal of cerebral blood flow and metabolism (01.01.2013)
Published in Journal of cerebral blood flow and metabolism (01.01.2013)
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Reduced cannabinoid CB1 receptor binding in alcohol dependence measured with positron emission tomography
HIRVONEN, J, ZANOTTI-FREGONARA, P, MORSE, C, ZOGHBI, S. S, PIKE, V. W, INNIS, R. B, HEILIG, M, UMHAU, J. C, GEORGE, D. T, RALLIS-FRUTOS, D, LYOO, C. H, LI, C.-T, HINES, C. S, SUN, H, TERRY, G. E
Published in Molecular psychiatry (01.08.2013)
Published in Molecular psychiatry (01.08.2013)
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Neuroinflammation in Temporal Lobe Epilepsy Measured Using Positron Emission Tomographic Imaging of Translocator Protein
Gershen, Leah D, Zanotti-Fregonara, Paolo, Dustin, Irene H, Liow, Jeih-San, Hirvonen, Jussi, Kreisl, William C, Jenko, Kimberly J, Inati, Sara K, Fujita, Masahiro, Morse, Cheryl L, Brouwer, Chad, Hong, Jinsoo S, Pike, Victor W, Zoghbi, Sami S, Innis, Robert B, Theodore, William H
Published in JAMA neurology (01.08.2015)
Published in JAMA neurology (01.08.2015)
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In vivo‐ and in silico‐driven identification of novel synthetic quinoxalines as anticonvulsants and AMPA inhibitors
Abulkhair, Hamada S., Elmeligie, Salwa, Ghiaty, Adel, El‐Morsy, Ahmed, Bayoumi, Ashraf H., Ahmed, Hany E. A., El‐Adl, Khaled, Zayed, Mohamed F., Hassan, Memy H., Akl, Eman N., El‐Zoghbi, Mona S.
Published in Archiv der Pharmazie (Weinheim) (01.05.2021)
Published in Archiv der Pharmazie (Weinheim) (01.05.2021)
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The Inhibitor Ko143 Is Not Specific for ABCG2
Weidner, Lora D, Zoghbi, Sami S, Lu, Shuiyu, Shukla, Suneet, Ambudkar, Suresh V, Pike, Victor W, Mulder, Jan, Gottesman, Michael M, Innis, Robert B, Hall, Matthew D
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)
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Evaluation of Two Potent and Selective PET Radioligands to Image COX-1 and COX-2 in Rhesus Monkeys
Kim, Min-Jeong, Shrestha, Stal S, Cortes, Michelle, Singh, Prachi, Morse, Cheryl, Liow, Jeih-San, Gladding, Robert L, Brouwer, Chad, Henry, Katharine, Gallagher, Evan, Tye, George L, Zoghbi, Sami S, Fujita, Masahiro, Pike, Victor W, Innis, Robert B
Published in Journal of Nuclear Medicine (01.12.2018)
Published in Journal of Nuclear Medicine (01.12.2018)
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New Pyrimidine-5-Carbonitriles as COX-2 Inhibitors: Design, Synthesis, Anticancer Screening, Molecular Docking, and In Silico ADME Profile Studies
AL-Ghulikah, Hanan A, El-Sebaey, Samiha A, Bass, Amr K. A, El-Zoghbi, Mona S
Published in Molecules (Basel, Switzerland) (01.11.2022)
Published in Molecules (Basel, Switzerland) (01.11.2022)
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Synthesis and preclinical evaluation of [11C]uPSEM792 for PSAM4-GlyR based chemogenetics
Nerella, Sridhar Goud, Telu, Sanjay, Liow, Jeih-San, Jenkins, Madeline D., Zoghbi, Sami S., Gomez, Juan L., Michaelides, Michael, Eldridge, Mark A. G., Richmond, Barry J., Innis, Robert B., Pike, Victor W.
Published in Scientific reports (22.01.2024)
Published in Scientific reports (22.01.2024)
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Design, synthesis, docking, and anticancer evaluations of new thiazolo[3,2-a] pyrimidines as topoisomerase II inhibitors
El-Zoghbi, Mona S., El-Sebaey, Samiha A., AL-Ghulikah, Hanan A., Sobh, Eman A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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PET measurement of cyclooxygenase-2 using a novel radioligand: upregulation in primate neuroinflammation and first-in-human study
Shrestha, Stal, Kim, Min-Jeong, Eldridge, Mark, Lehmann, Michael L, Frankland, Michael, Liow, Jeih-San, Yu, Zu-Xi, Cortes-Salva, Michelle, Telu, Sanjay, Henter, Ioline D, Gallagher, Evan, Lee, Jae-Hoon, Fredericks, J Megan, Poffenberger, Chelsie, Tye, George, Ruiz-Perdomo, Yanira, Anaya, Fernanda Juarez, Montero Santamaria, Jose A, Gladding, Robert L, Zoghbi, Sami S, Fujita, Masahiro, Katz, James D, Pike, Victor W, Innis, Robert B
Published in Journal of neuroinflammation (02.05.2020)
Published in Journal of neuroinflammation (02.05.2020)
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Distinct patterns of increased translocator protein in posterior cortical atrophy and amnestic Alzheimer’s disease
Kreisl, William C, Lyoo, Chul Hyoung, Liow, Jeih-San, Snow, Joseph, Page, Emily, Jenko, Kimberly J, Morse, Cheryl L, Zoghbi, Sami S, Pike, Victor W, Turner, R. Scott, Innis, Robert B
Published in Neurobiology of aging (01.03.2017)
Published in Neurobiology of aging (01.03.2017)
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Prediction of Dopamine Transporter Binding Availability by Genotype: A Preliminary Report
Jacobsen, Leslie K., Staley, Julie K., Zoghbi, Sami S., Seibyl, John P., Kosten, Thomas R., Innis, Robert B., Gelernter, Joel
Published in The American journal of psychiatry (01.10.2000)
Published in The American journal of psychiatry (01.10.2000)
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Kinetic analysis in healthy humans of a novel positron emission tomography radioligand to image the peripheral benzodiazepine receptor, a potential biomarker for inflammation
Fujita, Masahiro, Imaizumi, Masao, Zoghbi, Sami S., Fujimura, Yota, Farris, Amanda G., Suhara, Tetsuya, Hong, Jinsoo, Pike, Victor W., Innis, Robert B.
Published in NeuroImage (Orlando, Fla.) (01.03.2008)
Published in NeuroImage (Orlando, Fla.) (01.03.2008)
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3‑Substituted 1,5-Diaryl‑1H‑1,2,4-triazoles as Prospective PET Radioligands for Imaging Brain COX‑1 in Monkey. Part 1: Synthesis and Pharmacology
Singh, Prachi, Shrestha, Stal, Cortes-Salva, Michelle Y, Jenko, Kimberly J, Zoghbi, Sami S, Morse, Cheryl L, Innis, Robert B, Pike, Victor W
Published in ACS chemical neuroscience (21.11.2018)
Published in ACS chemical neuroscience (21.11.2018)
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Comparison of two PET radioligands, [11C]FPEB and [11C]SP203, for quantification of metabotropic glutamate receptor 5 in human brain
Lohith, Talakad G, Tsujikawa, Tetsuya, Siméon, Fabrice G, Veronese, Mattia, Zoghbi, Sami S, Lyoo, Chul Hyoung, Kimura, Yasuyuki, Morse, Cheryl L, Pike, Victor W, Fujita, Masahiro, Innis, Robert B
Published in Journal of cerebral blood flow and metabolism (01.07.2017)
Published in Journal of cerebral blood flow and metabolism (01.07.2017)
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Evaluation of 11C-NR2B-SMe and Its Enantiomers as PET Radioligands for Imaging the NR2B Subunit Within the NMDA Receptor Complex in Rats
Cai, Lisheng, Liow, Jeih-San, Morse, Cheryl L, Telu, Sanjay, Davies, Riley, Frankland, Michael P, Zoghbi, Sami S, Cheng, Ken, Hall, Matthew D, Innis, Robert B, Pike, Victor W
Published in The Journal of nuclear medicine (1978) (01.08.2020)
Published in The Journal of nuclear medicine (1978) (01.08.2020)
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