A New Cross-Coupling-Based Synthesis of Carpanone
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Published in Organic letters (01.10.2009)
Published in Organic letters (01.10.2009)
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Discovery of a First-In-Class Small Molecule Antagonist against the Adrenomedullin‑2 Receptor: Structure–Activity Relationships and Optimization
Zirimwabagabo, Jean-Olivier, Jailani, Ameera B. A, Avgoustou, Paris, Tozer, Matthew J, Gibson, Karl R, Glossop, Paul A, Mills, James E. J, Porter, Roderick A, Blaney, Paul, Wang, Ning, Skerry, Timothy M, Richards, Gareth O, Harrity, Joseph P. A
Published in Journal of medicinal chemistry (25.03.2021)
Published in Journal of medicinal chemistry (25.03.2021)
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Discovery of a First-in-Class Potent Small Molecule Antagonist against the Adrenomedullin‑2 Receptor
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Published in ACS pharmacology & translational science (14.08.2020)
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AM2 수용체 억제제로서의 복소환식 스피로-화합물
GIBSON KARL RICHARD, GLOSSOP PAUL ALAN, SKERRY TIMOTHY M, PORTER RODERICK ALAN, ZIRIMWABAGABO JEAN OLIVIER, TOZER MATTHEW J, RICHARDS GARETH, HARRITY JOSEPH P.A
Year of Publication 17.09.2021
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Year of Publication 17.09.2021
Patent
AM2 수용체 억제제로서의 복소환식 스피로-화합물
GIBSON KARL RICHARD, GLOSSOP PAUL ALAN, SKERRY TIMOTHY M, PORTER RODERICK ALAN, ZIRIMWABAGABO JEAN OLIVIER, TOZER MATTHEW J, RICHARDS GARETH, HARRITY JOSEPH P.A
Year of Publication 19.08.2021
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Year of Publication 19.08.2021
Patent
Pd-Catalyzed kinetic resolution of cyclic enol ethers. An enantioselective route to functionalised pyransElectronic supplementary information (ESI) available: Experimental procedures, spectral data and stereochemical proofs. CCDC 979882. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c4cc00109e
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ChemInform Abstract: Palladium-Catalyzed Decarboxylative Generation and Asymmetric Allylation of α-Imino Anions
Qian, Xiaoyan, Ji, Pengfei, He, Chang, Zirimwabagabo, Jean-Olivier, Archibald, Michelle M., Yeagley, Andrew A., Chruma, Jason J.
Published in ChemInform (01.03.2015)
Published in ChemInform (01.03.2015)
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COMPOUNDS
GIBSON, Karl, Richard, BLANEY, Paul, Matthew, ZIRIMWABAGABO, Jean-Olivier, PORTER, Roderick, Alan, RICHARDS, Gareth, TOZER, Matthew, J, HARRITY, Joseph, P.A, GLOSSOP, Paul, Alan, SKERRY, Timothy, M
Year of Publication 03.07.2024
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Year of Publication 03.07.2024
Patent
Compounds
Gibson, Karl Richard, Harrity, Joseph P. A, Zirimwabagabo, Jean-Olivier, Porter, Roderick Alan, Richards, Gareth, Glossop, Paul Alan, Skerry, Timothy M, Blaney, Paul Matthew, Tozer, Matthew J
Year of Publication 02.08.2022
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Year of Publication 02.08.2022
Patent
HETEROCYCLIC SPIRO-COMPOUNDS AS AM2 RECEPTOR INHIBITORS
SKERRY, Timothy M, HARRITY, Joseph P.A, ZIRIMWABAGABO, Jean-Olivier, RICHARDS, Gareth, TOZER, Matthew, GLOSSOP, Paul, GIBSON, Karl, PORTER, Roderick
Year of Publication 29.06.2021
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Year of Publication 29.06.2021
Patent
HETEROCYCLIC SPIRO-COMPOUNDS AS AM2 RECEPTOR INHIBITORS
ZIRIMWABAGABO, Jean-Olivier, RICHARDS, Gareth, TOZER, Matthew, GLOSSOP, Paul, GIBSON, Karl, HARRITY, Josephy, SKERRY, Timothy, PORTER, Roderick
Year of Publication 29.06.2021
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Year of Publication 29.06.2021
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