Discovery of triazolinone non-nucleoside inhibitors of HIV reverse transcriptase
Sweeney, Zachary K., Acharya, Sahaja, Briggs, Andrew, Dunn, James P., Elworthy, Todd R., Fretland, Jennifer, Giannetti, Anthony M., Heilek, Gabrielle, Li, Yu, Kaiser, Ann C., Martin, Michael, Saito, Y. David, Smith, Mark, Suh, Judy M., Swallow, Steven, Wu, Jeffrey, Hang, Julie Q., Zhou, Amy S., Klumpp, Klaus
Published in Bioorganic & medicinal chemistry (01.08.2008)
Published in Bioorganic & medicinal chemistry (01.08.2008)
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Journal Article
Design of Annulated Pyrazoles as Inhibitors of HIV-1 Reverse Transcriptase
Sweeney, Zachary K, Harris, Seth F, Arora, Nidhi, Javanbakht, Hassan, Li, Yu, Fretland, Jennifer, Davidson, James P, Billedeau, J. Roland, Gleason, Shelley K, Hirschfeld, Donald, Kennedy-Smith, Joshua J, Mirzadegan, Taraneh, Roetz, Ralf, Smith, Mark, Sperry, Sarah, Suh, Judy M, Wu, Jeffrey, Tsing, Stan, Villaseñor, Armando G, Paul, Amber, Su, Guoping, Heilek, Gabrielle, Hang, Julie Q, Zhou, Amy S, Jernelius, Jesper A, Zhang, Fang-Jie, Klumpp, Klaus
Published in Journal of medicinal chemistry (11.12.2008)
Published in Journal of medicinal chemistry (11.12.2008)
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Journal Article
Discovery and optimization of pyridazinone non-nucleoside inhibitors of HIV-1 reverse transcriptase
Sweeney, Zachary K., Dunn, James P., Li, Yu, Heilek, Gabrielle, Dunten, Pete, Elworthy, Todd R., Han, Xiaochun, Harris, Seth F., Hirschfeld, Donald R., Hogg, J. Heather, Huber, Walter, Kaiser, Ann C., Kertesz, Denis J., Kim, Woongki, Mirzadegan, Taraneh, Roepel, Michael G., Saito, Y. David, Silva, Tania M.P.C., Swallow, Steven, Tracy, Jahari L., Villasenor, Armando, Vora, Harit, Zhou, Amy S., Klumpp, Klaus
Published in Bioorganic & medicinal chemistry (01.08.2008)
Published in Bioorganic & medicinal chemistry (01.08.2008)
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Journal Article
Orally bioavailable prodrugs of a BCS class 2 molecule, an inhibitor of HIV-1 reverse transcriptase
Elworthy, Todd R., Dunn, James P., Hogg, J. Heather, Lam, Grace, Saito, Y. David, Silva, Tania M.P.C., Stefanidis, Dimitrios, Woroniecki, Witold, Zhornisky, Eugenia, Zhou, Amy S., Klumpp, Klaus
Published in Bioorganic & medicinal chemistry (15.12.2008)
Published in Bioorganic & medicinal chemistry (15.12.2008)
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Journal Article