Highly potent p21(WAF1)-derived peptide inhibitors of CDK-mediated pRb phosphorylation: delineation and structural insight into their interactions with cyclin A
Zheleva, D I, McInnes, C, Gavine, A-L, Zhelev, N Z, Fischer, P M, Lane, D P
Published in The journal of peptide research (01.11.2002)
Published in The journal of peptide research (01.11.2002)
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A Quantitative Study of the in Vitro Binding of the C-Terminal Domain of p21 to PCNA: Affinity, Stoichiometry, and Thermodynamics
Zheleva, Daniella I, Zhelev, Nikolai Z, Fischer, Peter M, Duff, Susan V, Warbrick, Emma, Blake, David G, Lane, David P
Published in Biochemistry (Easton) (27.06.2000)
Published in Biochemistry (Easton) (27.06.2000)
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Journal Article
Use of Peptides from p21 (Waf1/Cip1) to Investigate PCNA Function in Xenopus Egg Extracts
Mattock, Heidi, Jares, Pedro, Zheleva, Daniella I., Lane, David P., Warbrick, Emma, Blow, J.Julian
Published in Experimental cell research (01.05.2001)
Published in Experimental cell research (01.05.2001)
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Journal Article
Structural and Biochemical Studies of Human Proliferating Cell Nuclear Antigen Complexes Provide a Rationale for Cyclin Association and Inhibitor Design
Kontopidis, George, Wu, Su-Ying, Zheleva, Daniella I., Taylor, Paul, McInnes, Campbell, Lane, David P., Fischer, Peter M., Walkinshaw, Malcolm D., Fersht, Alan
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2005)
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2005)
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Discovery of a Novel Family of CDK Inhibitors with the Program LIDAEUS: Structural Basis for Ligand-Induced Disordering of the Activation Loop
Wu, Su Ying, McNae, Iain, Kontopidis, George, McClue, Steven J, McInnes, Campbell, Stewart, Kevin J, Wang, Shudong, Zheleva, Daniella I, Marriage, Howard, Lane, David P, Taylor, Paul, Fischer, Peter M, Walkinshaw, Malcolm D
Published in Structure (London) (01.04.2003)
Published in Structure (London) (01.04.2003)
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Insights into Cyclin Groove Recognition: Complex Crystal Structures and Inhibitor Design through Ligand Exchange
Kontopidis, George, Andrews, Martin J.I., McInnes, Campbell, Cowan, Angela, Powers, Helen, Innes, Lorraine, Plater, Andy, Griffiths, Gary, Paterson, Dougie, Zheleva, Daniella I., Lane, David P., Green, Stephen, Walkinshaw, Malcolm D., Fischer, Peter M.
Published in Structure (London) (01.12.2003)
Published in Structure (London) (01.12.2003)
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Journal Article
Peptide inhibitors of CDK2-cyclin A that target the cyclin recruitment-Site: structural variants of the C-Terminal Phe
Atkinson, Gail E, Cowan, Angela, McInnes, Campbell, Zheleva, Daniella I, Fischer, Peter M, Chan, Weng C
Published in Bioorganic & medicinal chemistry letters (16.09.2002)
Published in Bioorganic & medicinal chemistry letters (16.09.2002)
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Discovery and Characterization of 2-Anilino-4- (Thiazol-5-yl)Pyrimidine Transcriptional CDK Inhibitors as Anticancer Agents
Wang, Shudong, Griffiths, Gary, Midgley, Carol A., Barnett, Anna L., Cooper, Michael, Grabarek, Joanna, Ingram, Laura, Jackson, Wayne, Kontopidis, George, McClue, Steven J., McInnes, Campbell, McLachlan, Janice, Meades, Christopher, Mezna, Mokdad, Stuart, Iain, Thomas, Mark P., Zheleva, Daniella I., Lane, David P., Jackson, Robert C., Glover, David M., Blake, David G., Fischer, Peter M.
Published in Chemistry & biology (29.10.2010)
Published in Chemistry & biology (29.10.2010)
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