LLY-507, a Cell-active, Potent, and Selective Inhibitor of Protein-lysine Methyltransferase SMYD2
Nguyen, Hannah, Allali-Hassani, Abdellah, Antonysamy, Stephen, Chang, Shawn, Chen, Lisa Hong, Curtis, Carmen, Emtage, Spencer, Fan, Li, Gheyi, Tarun, Li, Fengling, Liu, Shichong, Martin, Joseph R., Mendel, David, Olsen, Jonathan B., Pelletier, Laura, Shatseva, Tatiana, Wu, Song, Zhang, Feiyu Fred, Arrowsmith, Cheryl H., Brown, Peter J., Campbell, Robert M., Garcia, Benjamin A., Barsyte-Lovejoy, Dalia, Mader, Mary, Vedadi, Masoud
Published in The Journal of biological chemistry (29.05.2015)
Published in The Journal of biological chemistry (29.05.2015)
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Abstract P142: Preclinical characterization of LOX-22783, a highly potent, mutant-selective and brain-penetrant allosteric PI3Kα H1047R inhibitor
Klippel, Anke, Wang, Rui, Puca, Loredana, Faber, Andrew Lee, Shen, Weihua, Bhagwat, Shripad V., Karukurichi, Kannan, Zhang, Feiyu Fred, Perez, Carmen, Rama, Ramon, Ramos, Ana, Zheng, Yi, Bonday, Zahid, Thomas, James, Brooks, Harold B., Kindler, Lisa J., Bogner, Sarah M., Zolfaghari, Parisa, II, Mark Hicks, Callies, Sophie, Mattioni, Brian, LeBrun, Laurie, Durbin, Jim, Anderson, Erin, Mayne, Chris, Kesicki, Edward, Kolakowski, Gabrielle, Andrews, Steven W., Brandhuber, Barbara J.
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Thermodynamic benchmark study using Biacore technology
Navratilova, Iva, Papalia, Giuseppe A., Rich, Rebecca L., Bedinger, Daniel, Brophy, Susan, Condon, Brad, Deng, Ta, Emerick, Anne W., Guan, Hann-Wen, Hayden, Tanya, Heutmekers, Thomas, Hoorelbeke, Bart, McCroskey, Mark C., Murphy, Mary M., Nakagawa, Terry, Parmeggiani, Fabio, Qin, Xiaochun, Rebe, Sabina, Tomasevic, Nenad, Tsang, Tiffany, Waddell, M. Brett, Zhang, Fred Feiyu, Leavitt, Stephanie, Myszka, David G.
Published in Analytical biochemistry (01.05.2007)
Published in Analytical biochemistry (01.05.2007)
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Structural Bases of PAS Domain-regulated Kinase (PASK) Activation in the Absence of Activation Loop Phosphorylation
Kikani, Chintan K., Antonysamy, Stephen A., Bonanno, Jeffrey B., Romero, Rich, Zhang, Feiyu Fred, Russell, Marijane, Gheyi, Tarun, Iizuka, Miyo, Emtage, Spencer, Sauder, J. Michael, Turk, Benjamin E., Burley, Stephen K., Rutter, Jared
Published in The Journal of biological chemistry (24.12.2010)
Published in The Journal of biological chemistry (24.12.2010)
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