Search Results - "Zeinyeh, Wael" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Converting Potent Indeno[1,2‑b]indole Inhibitors of Protein Kinase CK2 into Selective Inhibitors of the Breast Cancer Resistance Protein ABCG2

Converting Potent Indeno[1,2‑b]indole Inhibitors of Protein Kinase CK2 into Selective Inhibitors of the Breast Cancer Resistance Protein ABCG2

by Jabor Gozzi, Gustavo, Bouaziz, Zouhair, Winter, Evelyn, Daflon-Yunes, Nathalia, Aichele, Dagmar, Nacereddine, Abdelhamid, Marminon, Christelle, Valdameri, Glaucio, Zeinyeh, Waël, Bollacke, Andre, Guillon, Jean, Lacoudre, Aline, Pinaud, Noël, Cadena, Silvia M., Jose, Joachim, Le Borgne, Marc, Di Pietro, Attilio
Published in Journal of medicinal chemistry (08.01.2015)

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Involvement of the Prion Protein in the Protection of the Human Bronchial Epithelial Barrier Against Oxidative Stress

Involvement of the Prion Protein in the Protection of the Human Bronchial Epithelial Barrier Against Oxidative Stress

by Kouadri, Amal, El Khatib, Mariam, Cormenier, Johanna, Chauvet, Sylvain, Zeinyeh, Wael, El Khoury, Micheline, Macari, Laurence, Richaud, Pierre, Coraux, Christelle, Michaud-Soret, Isabelle, Alfaidy, Nadia, Benharouga, Mohamed
Published in Antioxidants & redox signaling (01.07.2019)

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Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies

Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies

by Zeinyeh, Wael, Esvan, Yannick J., Josselin, Béatrice, Baratte, Blandine, Bach, Stéphane, Nauton, Lionel, Théry, Vincent, Ruchaud, Sandrine, Anizon, Fabrice, Giraud, Francis, Moreau, Pascale
Published in Bioorganic & medicinal chemistry (15.05.2019)

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Targeting different binding sites in the CFTR structures allows to synergistically potentiate channel activity

Targeting different binding sites in the CFTR structures allows to synergistically potentiate channel activity

by Froux, Lionel, Elbahnsi, Ahmad, Boucherle, Benjamin, Billet, Arnaud, Baatallah, Nesrine, Hoffmann, Brice, Alliot, Julien, Zelli, Renaud, Zeinyeh, Wael, Haudecoeur, Romain, Chevalier, Benoit, Fortuné, Antoine, Mirval, Sandra, Simard, Christophe, Lehn, Pierre, Mornon, Jean-Paul, Hinzpeter, Alexandre, Becq, Frédéric, Callebaut, Isabelle, Décout, Jean-Luc
Published in European journal of medicinal chemistry (15.03.2020)

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QSAR Model of Indeno[1,2- b ]indole Derivatives and Identification of N -isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3- b ]furan-3-carboxamide as a Potent CK2 Inhibitor

QSAR Model of Indeno[1,2- b ]indole Derivatives and Identification of N -isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3- b ]furan-3-carboxamide as a Potent CK2 Inhibitor

by Haidar, Samer, Marminon, Christelle, Aichele, Dagmar, Nacereddine, Abdelhamid, Zeinyeh, Wael, Bouzina, Abdeslem, Berredjem, Malika, Ettouati, Laurent, Bouaziz, Zouhair, Le Borgne, Marc, Jose, Joachim
Published in Molecules (Basel, Switzerland) (01.01.2020)

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Unsymmetrical α,ω-end-functionalized oligo(cyclohexylidenes): efficient synthesis and conformational analysis

Unsymmetrical α,ω-end-functionalized oligo(cyclohexylidenes): efficient synthesis and conformational analysis

by Zeinyeh, Waël, Radix, Sylvie, Terreux, Raphaël, Chemelle, Julie-Anne, Walchshofer, Nadia
Published in Tetrahedron (07.07.2016)

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Progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux: Design, synthesis, characterization and biological evaluation

Progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux: Design, synthesis, characterization and biological evaluation

by Zeinyeh, Waël, Mahiout, Zahia, Radix, Sylvie, Lomberget, Thierry, Dumoulin, Axel, Barret, Roland, Grenot, Catherine, Rocheblave, Luc, Matera, Eva-Laure, Dumontet, Charles, Walchshofer, Nadia
Published in Steroids (01.10.2012)

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A One-Pot Synthesis of Highly Functionalized Purines

A One-Pot Synthesis of Highly Functionalized Purines

by Zelli, Renaud, Zeinyeh, Waël, Haudecoeur, Romain, Alliot, Julien, Boucherle, Benjamin, Callebaut, Isabelle, Décout, Jean-Luc
Published in Organic letters (01.12.2017)

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18FRS-127445 radiosynthesis and evaluation as a 5-HT2B receptor PET radiotracer in rat brain

18FRS-127445 radiosynthesis and evaluation as a 5-HT2B receptor PET radiotracer in rat brain

by Richin, Violette, Bouillot, Caroline, Bouvard, Sandrine, Courault, Pierre, Lancelot, Sophie, Zimmer, Luc, Zeinyeh, Wael
Published in Bioorganic & medicinal chemistry letters (01.11.2024)

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[18F]RS-127445 radiosynthesis and evaluation as a 5-HT2B receptor PET radiotracer in rat brain

[18F]RS-127445 radiosynthesis and evaluation as a 5-HT2B receptor PET radiotracer in rat brain

by Richin, Violette, Bouillot, Caroline, Bouvard, Sandrine, Courault, Pierre, Lancelot, Sophie, Zimmer, Luc, Zeinyeh, Wael
Published in Bioorganic & medicinal chemistry letters (01.11.2024)

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Amyloid-Beta Radiotracer [18F]BF-227 Does Not Bind to Cytoplasmic Glial Inclusions of Postmortem Multiple System Atrophy Brain Tissue

Amyloid-Beta Radiotracer [18F]BF-227 Does Not Bind to Cytoplasmic Glial Inclusions of Postmortem Multiple System Atrophy Brain Tissue

by Chauveau, Fabien, Zimmer, Luc, Quadrio, Isabelle, Billard, Thierry, Zeinyeh, Waël, Lancelot, Sophie, Levigoureux, Elise, Verdurand, Mathieu, Perret-Liaudet, Armand
Published in Contrast media and molecular imaging (01.01.2018)

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Basics of Fourier Transform Applied to NMR Spectroscopy: An Interactive Open-Source Web Application

Basics of Fourier Transform Applied to NMR Spectroscopy: An Interactive Open-Source Web Application

by Esvan, Yannick J, Zeinyeh, Wael
Published in Journal of chemical education (14.01.2020)

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Interactive Web Application as a Teaching Tool to Introduce Basics of Chromatography and the Plate Theory

Interactive Web Application as a Teaching Tool to Introduce Basics of Chromatography and the Plate Theory

by Jordheim, Lars Petter, Denuzière, Anne, Machon, Christelle, Zeinyeh, Wael
Published in Journal of chemical education (13.07.2021)

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Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity

Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity

by Zeinyeh, Wael, Esvan, Yannick J., Josselin, Béatrice, Defois, Mathilde, Baratte, Blandine, Knapp, Stefan, Chaikuad, Apirat, Anizon, Fabrice, Giraud, Francis, Ruchaud, Sandrine, Moreau, Pascale
Published in European journal of medicinal chemistry (05.06.2022)

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In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α‑Synuclein PET Imaging

In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α‑Synuclein PET Imaging

by Verdurand, Mathieu, Levigoureux, Elise, Zeinyeh, Wael, Berthier, Laurent, Mendjel-Herda, Meriem, Cadarossanesaib, Florence, Bouillot, Caroline, Iecker, Thibault, Terreux, Raphaël, Lancelot, Sophie, Chauveau, Fabien, Billard, Thierry, Zimmer, Luc
Published in Molecular pharmaceutics (06.08.2018)

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New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis

New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis

by Tazarki, Helmi, Zeinyeh, Wael, Esvan, Yannick J., Knapp, Stefan, Chatterjee, Deep, Schröder, Martin, Joerger, Andreas C., Khiari, Jameleddine, Josselin, Béatrice, Baratte, Blandine, Bach, Stéphane, Ruchaud, Sandrine, Anizon, Fabrice, Giraud, Francis, Moreau, Pascale
Published in European journal of medicinal chemistry (15.03.2019)

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Design, synthesis and evaluation of progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux

Design, synthesis and evaluation of progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux

by Zeinyeh, Waël, Alameh, Ghina, Radix, Sylvie, Grenot, Catherine, Dumontet, Charles, Walchshofer, Nadia
Published in Bioorganic & medicinal chemistry letters (15.05.2010)

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Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co–crystal structure

Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co–crystal structure

by Esvan, Yannick J., Zeinyeh, Wael, Boibessot, Thibaut, Nauton, Lionel, Théry, Vincent, Knapp, Stefan, Chaikuad, Apirat, Loaëc, Nadège, Meijer, Laurent, Anizon, Fabrice, Giraud, Francis, Moreau, Pascale
Published in European journal of medicinal chemistry (08.08.2016)

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Synthesis and modulation properties of imidazo[4,5- b]pyridin-7-one and indazole-4,7-dione derivatives towards the Cryptosporidium parvum CpABC3 transporter

Synthesis and modulation properties of imidazo[4,5- b]pyridin-7-one and indazole-4,7-dione derivatives towards the Cryptosporidium parvum CpABC3 transporter

by Zeinyeh, Waël, Xia, Hexue, Lawton, Philippe, Radix, Sylvie, Marminon, Christelle, Nebois, Pascal, Walchshofer, Nadia
Published in European journal of medicinal chemistry (01.06.2010)

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Synthesis and preliminary in vitro kinase inhibition evaluation of new diversely substituted pyrido[3,4-g]quinazoline derivatives

Synthesis and preliminary in vitro kinase inhibition evaluation of new diversely substituted pyrido[3,4-g]quinazoline derivatives

by Zeinyeh, Wael, Esvan, Yannick J., Nauton, Lionel, Loaëc, Nadège, Meijer, Laurent, Théry, Vincent, Anizon, Fabrice, Giraud, Francis, Moreau, Pascale
Published in Bioorganic & medicinal chemistry letters (01.09.2016)

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