ATP-competitive DNA gyrase and topoisomerase IV inhibitors as antibacterial agents
Durcik, Martina, Tomašič, Tihomir, Zidar, Nace, Zega, Anamarija, Kikelj, Danijel, Mašič, Lucija Peterlin, Ilaš, Janez
Published in Expert opinion on therapeutic patents (04.03.2019)
Published in Expert opinion on therapeutic patents (04.03.2019)
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Rational design of balanced dual-targeting antibiotics with limited resistance
Nyerges, Akos, Tomašič, Tihomir, Durcik, Martina, Revesz, Tamas, Szili, Petra, Draskovits, Gabor, Bogar, Ferenc, Skok, Žiga, Zidar, Nace, Ilaš, Janez, Zega, Anamarija, Kikelj, Danijel, Daruka, Lejla, Kintses, Balint, Vasarhelyi, Balint, Foldesi, Imre, Kata, Diána, Welin, Martin, Kimbung, Raymond, Focht, Dorota, Mašič, Lucija Peterlin, Pal, Csaba
Published in PLoS biology (05.10.2020)
Published in PLoS biology (05.10.2020)
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Crystallographic Study of Peptidoglycan Biosynthesis Enzyme MurD: Domain Movement Revisited
Šink, Roman, Kotnik, Miha, Zega, Anamarija, Barreteau, Hélène, Gobec, Stanislav, Blanot, Didier, Dessen, Andréa, Contreras-Martel, Carlos
Published in PloS one (31.03.2016)
Published in PloS one (31.03.2016)
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Evaluation of the published kinase inhibitor set to identify multiple inhibitors of bacterial ATP-dependent mur ligases
Hrast, Martina, Rožman, Kaja, Ogris, Iza, Škedelj, Veronika, Patin, Delphine, Sova, Matej, Barreteau, Hélène, Gobec, Stanislav, Grdadolnik, Simona Golič, Zega, Anamarija
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Hybrid Inhibitors of DNA Gyrase A and B: Design, Synthesis and Evaluation
Durcik, Martina, Skok, Žiga, Ilaš, Janez, Zidar, Nace, Zega, Anamarija, Szili, Petra Éva, Draskovits, Gábor, Révész, Tamás, Kikelj, Danijel, Nyerges, Akos, Pál, Csaba, Mašič, Lucija Peterlin, Tomašič, Tihomir
Published in Pharmaceutics (22.12.2020)
Published in Pharmaceutics (22.12.2020)
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Efficient Synthesis of Hydroxy-Substituted 2‑Aminobenzo[d]thiazole-6-carboxylic Acid Derivatives as New Building Blocks in Drug Discovery
Durcik, Martina, Toplak, Žan, Zidar, Nace, Ilaš, Janez, Zega, Anamarija, Kikelj, Danijel, Mašič, Lucija Peterlin, Tomašič, Tihomir
Published in ACS omega (14.04.2020)
Published in ACS omega (14.04.2020)
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Practical Synthesis and Application of Halogen-Doped Pyrrole Building Blocks
Cotman, Andrej Emanuel, Guérin, Thomas, Kovačević, Ivana, Benedetto Tiz, Davide, Durcik, Martina, Fulgheri, Federica, Možina, Štefan, Secci, Daniela, Sterle, Maša, Ilaš, Janez, Zega, Anamarija, Zidar, Nace, Mašič, Lucija Peterlin, Tomašič, Tihomir, Leroux, Frédéric R, Hanquet, Gilles, Kikelj, Danijel
Published in ACS omega (13.04.2021)
Published in ACS omega (13.04.2021)
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6-Arylpyrido[2,3-d]pyrimidines as novel ATP-competitive inhibitors of bacterial D-alanine:D-alanine ligase
Škedelj, Veronika, Arsovska, Emilija, Tomašić, Tihomir, Kroflič, Ana, Hodnik, Vesna, Hrast, Martina, Bešter-Rogač, Marija, Anderluh, Gregor, Gobec, Stanislav, Bostock, Julieanne, Chopra, Ian, O'Neill, Alex J, Randall, Christopher, Zega, Anamarija
Published in PloS one (02.08.2012)
Published in PloS one (02.08.2012)
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NMR in the design of antibacterials
Arsovska, Emilija, Mali, Gregor, Golič Grdadolnik, Simona, Zega, Anamarija
Published in Current medicinal chemistry (01.01.2014)
Published in Current medicinal chemistry (01.01.2014)
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Dual Inhibitor of MurD and MurE Ligases from Escherichia coli and Staphylococcus aureus
Tomašić, Tihomir, Šink, Roman, Zidar, Nace, Fic, Anja, Contreras-Martel, Carlos, Dessen, Andréa, Patin, Delphine, Blanot, Didier, Müller-Premru, Manica, Gobec, Stanislav, Zega, Anamarija, Kikelj, Danijel, Mašič, Lucija Peterlin
Published in ACS medicinal chemistry letters (09.08.2012)
Published in ACS medicinal chemistry letters (09.08.2012)
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Data on biosynthesis of BPAF glucuronide, enzyme kinetics of BPAF glucuronidation, and molecular modeling
Gramec Skledar, Darja, Trontelj, Jurij, Troberg, Johanna, Tomašič, Tihomir, Zega, Anamarija, Finel, Moshe, Peterlin Mašič, Lucija
Published in Data in brief (01.02.2019)
Published in Data in brief (01.02.2019)
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Hydrogen-Bonding Ability of Noyori-Ikariya Catalysts Enables Stereoselective Access to CF 3 -Substituted syn -1,2-Diols via Dynamic Kinetic Resolution
Sterle, Maša, Huš, Matej, Lozinšek, Matic, Zega, Anamarija, Cotman, Andrej Emanuel
Published in ACS catalysis (05.05.2023)
Published in ACS catalysis (05.05.2023)
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Direct thrombin inhibitors built on the azaphenylalanine scaffold provoke degranulation of mast cells
Peternel, Luka, Stempelj, Mateja, Cerne, Manica, Zega, Anamarija, Obreza, Ales, Oblak, Marko, Drevensek, Gorazd, Budihna, Metka V, Stanovnik, Lovro, Urleb, Uros
Published in Thrombosis and haemostasis (01.02.2006)
Published in Thrombosis and haemostasis (01.02.2006)
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Antithrombotic potential of new direct thrombin inhibitors built on the azaphenylalanine scaffold in two rat venous thrombosis models
Peternel, Luka, Stegnar, Mojca, Drevensek, Gorazd, Budihna, Metka V, Bozic, Mojca, Zega, Anamarija, Stalc, Anton, Cerne, Manica, Urleb, Uros
Published in Thrombosis and haemostasis (01.03.2005)
Published in Thrombosis and haemostasis (01.03.2005)
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Hydrogen-Bonding Ability of Noyori–Ikariya Catalysts Enables Stereoselective Access to CF3‑Substituted syn-1,2-Diols via Dynamic Kinetic Resolution
Sterle, Maša, Huš, Matej, Lozinšek, Matic, Zega, Anamarija, Cotman, Andrej Emanuel
Published in ACS catalysis (05.05.2023)
Published in ACS catalysis (05.05.2023)
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Endocrine activities and adipogenic effects of bisphenol AF and its main metabolite
Skledar, Darja Gramec, Carino, Adriana, Trontelj, Jurij, Troberg, Johanna, Distrutti, Eleonora, Marchianò, Silvia, Tomašič, Tihomir, Zega, Anamarija, Finel, Moshe, Fiorucci, Stefano, Mašič, Lucija Peterlin
Published in Chemosphere (Oxford) (01.01.2019)
Published in Chemosphere (Oxford) (01.01.2019)
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ATP-competitive inhibitors of human DNA topoisomerase II? with improved antiproliferative activity based on N-phenylpyrrolamide scaffold
Skok, Ziga, Durcik, Martina, Zajex, Ziva, Skledar, Darja Gramec, Bozovic, Kristof, Pis, Anja, Tomas, Tihomir, Zega, Anamarija, Mas, Lucija Peterlin, Kikelj, Danijel, Zidar, Nace, Ilas, Janez
Published in European journal of medicinal chemistry (05.03.2023)
Published in European journal of medicinal chemistry (05.03.2023)
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