Development of a [18F]PD-L1 radiotracer to profile cancer patient response to immunotherapy
Zecca, Henry, Seo, Wone Woo, Voll, Ronald, Birnbaum, Lacey, Kelvin, James, Dreaden, Erik, Jui, Nathan, Goodman, Mark
Published in Nuclear medicine and biology (01.05.2022)
Published in Nuclear medicine and biology (01.05.2022)
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Journal Article
P-256 - Development of a [18F]PD-L1 radiotracer to profile cancer patient response to immunotherapy
Zecca, Henry, Seo, Wone Woo, Voll, Ronald, Birnbaum, Lacey, Kelvin, James, Dreaden, Erik, Jui, Nathan, Goodman, Mark
Published in Nuclear medicine and biology (01.05.2022)
Published in Nuclear medicine and biology (01.05.2022)
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Constitutively Synergistic Multiagent Drug Formulations Targeting MERTK, FLT3, and BCL-2 for Treatment of AML
Kelvin, James M., Jain, Juhi, Thapa, Aashis, Qui, Min, Birnbaum, Lacey A., Moore, Samuel G., Zecca, Henry, Summers, Ryan J., Switchenko, Jeffrey M., Costanza, Emma, Uricoli, Biaggio, Wang, Xiaodong, Jui, Nathan T., Fu, Haian, Du, Yuhong, DeRyckere, Deborah, Graham, Douglas K., Dreaden, Erik C.
Published in Pharmaceutical research (01.09.2023)
Published in Pharmaceutical research (01.09.2023)
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Journal Article
Development of constitutively synergistic nanoformulations to enhance chemosensitivity in T-cell leukemia
Kelvin, James M., Chimenti, Madison L., Zhang, Dan Y., Williams, Evelyn K., Moore, Samuel G., Humber, Gabrielle M., Baxter, Travon A., Birnbaum, Lacey A., Qui, Min, Zecca, Henry, Thapa, Aashis, Jain, Juhi, Jui, Nathan T., Wang, Xiaodong, Fu, Haian, Du, Yuhong, Kemp, Melissa L., Lam, Wilbur A., Graham, Douglas K., DeRyckere, Deborah, Dreaden, Erik C.
Published in Journal of controlled release (01.09.2023)
Published in Journal of controlled release (01.09.2023)
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Discovery of Tetrahydropyridopyrimidines as Irreversible Covalent Inhibitors of KRAS-G12C with In Vivo Activity
Fell, Jay B, Fischer, John P, Baer, Brian R, Ballard, Joshua, Blake, James F, Bouhana, Karyn, Brandhuber, Barbara J, Briere, David M, Burgess, Laurence E, Burkard, Michael R, Chiang, Harrah, Chicarelli, Mark J, Davidson, Kevin, Gaudino, John J, Hallin, Jill, Hanson, Lauren, Hee, Kenneth, Hicken, Erik J, Hinklin, Ronald J, Marx, Matthew A, Mejia, Macedonio J, Olson, Peter, Savechenkov, Pavel, Sudhakar, Niranjan, Tang, Tony P, Vigers, Guy P, Zecca, Henry, Christensen, James G
Published in ACS medicinal chemistry letters (13.12.2018)
Published in ACS medicinal chemistry letters (13.12.2018)
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Novel 1,2-dihydroquinazolin-2-ones: Design, synthesis, and biological evaluation against Trypanosoma brucei
Pham, ThanhTruc, Walden, Madeline, Butler, Christopher, Diaz-Gonzalez, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, Gomez-Pérez, Veronica, García-Hernández, Raquel, Zecca, Henry, Krakoff, Emma, Kopec, Brian, Ichire, Ogar, Mackenzie, Caden, Pitot, Marika, Ruiz, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Navarro, Miguel, Dounay, Amy B.
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
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Journal Article
KRAS G12C 억제제
HINKLIN RONALD JAY, MEJIA MACEDONIO J, VIGERS GUY P.A, FISCHER JOHN P, LEE MATTHEW RANDOLF, FELL JAY BRADFORD, GAUDINO JOHN J, ZECCA HENRY J, TANG TONY P, BLAKE JAMES F, CHRISTENSEN JAMES GAIL, HICKEN ERIK JAMES, MARX MATTHEW ARNOLD, CHICARELLI MARK JOSEPH, BURGESS LAURENCE E, SAVECHENKOV PAVEL
Year of Publication 12.04.2019
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Year of Publication 12.04.2019
Patent
Constitutively synergistic multiagent drug formulations targeting MERTK, FLT3, and BCL-2 for treatment of AML
Kelvin, James M, Jain, Juhi, Thapa, Aashis, Qui, Min, Birnbaum, Lacey A, Moore, Samuel G, Zecca, Henry, Summers, Ryan J, Costanza, Emma, Uricoli, Biaggio, Wang, Xiaodong, Jui, Nathan T, Fu, Haian, Du, Yuhong, DeRyckere, Deborah, Graham, Douglas K, Dreaden, Erik C
Published in bioRxiv : the preprint server for biology (15.03.2023)
Published in bioRxiv : the preprint server for biology (15.03.2023)
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MODULATORS OF LIVER RECEPTOR HOMOLOGUE 1 (LRH-1) AND USES
CATO, Michael Lee, FLYNN, Autumn, JUI, Nathan, ORTLUND, Eric, ZECCA, Henry, SPURLIN, Racheal
Year of Publication 02.05.2024
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Year of Publication 02.05.2024
Patent
KRas G12C inhibitors
Hicken, Erik James, Blake, James F, Chicarelli, Mark Joseph, Vigers, Guy P. A, Tang, Tony, Fischer, John P, Marx, Matthew Arnold, Zecca, Henry J, Lee, Matthew Randolph, Fell, Jay Bradford, Savechenkov, Pavel
Year of Publication 19.03.2024
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Year of Publication 19.03.2024
Patent
KRAS G12C INHIBITORS
FELL, Jay, Bradford, TANG, Tony, VIGERS, Guy, P.A, HICKEN, Erik, James, MARX, Matthew, Arnold, LEE, Matthew, Randolph, ZECCA, Henry, J, BLAKE, James, F, FISHER, John, P, CHICARELLI, Mark, Joseph, SAVENCHENKOV, Pavel
Year of Publication 09.03.2022
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Year of Publication 09.03.2022
Patent
KRAS G12C INHIBITORS
Vigers, Guy P.A, Hicken, Erik James, Blake, James F, Chicarelli, Mark Joseph, Tang, Tony, Fischer, John P, Marx, Matthew Arnold, Zecca, Henry J, Lee, Matthew Randolph, Fell, Jay Bradford, Savechenkov, Pavel
Year of Publication 09.12.2021
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Year of Publication 09.12.2021
Patent
Screening and Development of Constitutively Synergistic Combination Drug Formulations for T Cell Acute Lymphoblastic Leukemia
Kelvin, James M, Zhang, Dan Y, Williams, Evelyn K, Moore, Samuel G, Birnbaum, Lacey A, Zecca, Henry, Wang, Xiaodong, Jain, Juhi, Qui, Min, Jui, Nathan T, Fu, Haian, Du, Yuhong, Kemp, Melissa L, Lam, Wilbur A, Deryckere, Deborah, Graham, Douglas K, Dreaden, Erik C
Published in bioRxiv (22.09.2022)
Published in bioRxiv (22.09.2022)
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Paper
KRAS G12C inhibitors
Burgess, Laurence E, Hicken, Erik James, Blake, James F, Vigers, Guy P. A, Gaudino, John J, Hinklin, Ronald Jay, Fischer, John P, Marx, Matthew Arnold, Lee, Matthew Randolph, Savechenkov, Pavel, Tang, Tony P, Mejia, Macedonio J, Christensen, James Gail, Chicarelli, Mark Joseph, Zecca, Henry J, Fell, Jay Bradford
Year of Publication 08.03.2022
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Year of Publication 08.03.2022
Patent
KRAS G12C INHIBITORS
FELL, Jay, Bradford, TANG, Tony, VIGERS, Guy, P.A, HICKEN, Erik, James, MARX, Matthew, Arnold, LEE, Matthew, Randolph, ZECCA, Henry, J, BLAKE, James, F, FISHER, John, P, CHICARELLI, Mark, Joseph, SAVENCHENKOV, Pavel
Year of Publication 17.03.2021
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Year of Publication 17.03.2021
Patent
KRAS G12C INHIBITORS
TANG, Tony, HINKEN, Erik, FELL, Jay, MARX, Matthew, ZECCA, Henry, BLAKE, James, FISHER, John, CHICARELLI, Mark, LEE, Matthew, SAVENCHENKOV, Pavel, VIGERS, Guy
Year of Publication 14.11.2019
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Year of Publication 14.11.2019
Patent
KRas G12C inhibitors
Burgess, Laurence E, Hicken, Erik James, Lee, Matthew Randolf, Blake, James F, Gaudino, John J, Hinklin, Ronald Jay, Fischer, John P, Marx, Matthew Arnold, Savechenkov, Pavel, Tang, Tony P, Mejia, Macedonio J, Vigers, Guy P.A, Christensen, James Gail, Chicarelli, Mark Joseph, Zecca, Henry J, Fell, Jay Bradford
Year of Publication 02.09.2021
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Year of Publication 02.09.2021
Patent
KRAS G12C INHIBITORS
SAVECHENKOV, Pavel, BLAKE, James F, LEE, Matthew Randolf, HINKLIN, Ronald Jay, MEJIA, Macedonio J, VIGERS, Guy P.A, CHRISTENSEN, James Gail, FISCHER, John P, CHICARELLI, Mark Joseph, HICKEN, Erik James, ZECCA, Henry J, BURGESS, Laurence E, FELL, Jay Bradford, GAUDINO, John J, MARX, Matthew Arnold, TANG, Tony P
Year of Publication 02.09.2021
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Year of Publication 02.09.2021
Patent
KRAS G12C INHIBITORS
HINKLIN, Ronald, Jay, BURGESS, Laurence, E, SAVECHENKOV, Pavel, VIGERS, Guy, P.A, MARX, Matthew, Arnold, ZECCA, Henry, J, BLAKE, James, F, TANG, Tony, P, FELL, Jay, Bradford, LEE, Matthew, Randolf, MEJIA, Macedonio, J, HICKEN, Erik, James, GAUDINO, John, J, CHRISTENSEN, James, Gail, FISCHER, John, P, CHICARELLI, Mark, Joseph
Year of Publication 17.02.2021
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Year of Publication 17.02.2021
Patent